SK10342002A3 - Pyrimidínkarboxamidy užitočné ako selektívne inhibítory izozymov PDE4 - Google Patents

Pyrimidínkarboxamidy užitočné ako selektívne inhibítory izozymov PDE4 Download PDF

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Publication number
SK10342002A3
SK10342002A3 SK1034-2002A SK10342002A SK10342002A3 SK 10342002 A3 SK10342002 A3 SK 10342002A3 SK 10342002 A SK10342002 A SK 10342002A SK 10342002 A3 SK10342002 A3 SK 10342002A3
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SK
Slovakia
Prior art keywords
formula
group
carboxamide
inhibitors
asthma
Prior art date
Application number
SK1034-2002A
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English (en)
Slovak (sk)
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
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Pfizer Products Inc.
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Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of SK10342002A3 publication Critical patent/SK10342002A3/sk

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Virology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
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  • Urology & Nephrology (AREA)
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  • Pain & Pain Management (AREA)
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  • Hospice & Palliative Care (AREA)
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SK1034-2002A 2000-01-31 2001-01-30 Pyrimidínkarboxamidy užitočné ako selektívne inhibítory izozymov PDE4 SK10342002A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31
PCT/IB2001/000125 WO2001057025A1 (en) 2000-01-31 2001-01-30 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
SK10342002A3 true SK10342002A3 (sk) 2003-12-02

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SK1034-2002A SK10342002A3 (sk) 2000-01-31 2001-01-30 Pyrimidínkarboxamidy užitočné ako selektívne inhibítory izozymov PDE4

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US (1) US6740655B2 (enExample)
EP (1) EP1252157B1 (enExample)
JP (1) JP2003522165A (enExample)
KR (1) KR20020071029A (enExample)
CN (1) CN1404480A (enExample)
AP (1) AP2002002590A0 (enExample)
AR (1) AR027336A1 (enExample)
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CA (1) CA2396458C (enExample)
CO (1) CO5271669A1 (enExample)
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PT (1) PT1252157E (enExample)
PY (1) PY0102108A (enExample)
SK (1) SK10342002A3 (enExample)
SV (1) SV2001000298A (enExample)
TN (1) TNSN01019A1 (enExample)
TR (1) TR200402292T4 (enExample)
UY (1) UY26570A1 (enExample)
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Families Citing this family (86)

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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
US20030032632A1 (en) * 1999-12-24 2003-02-13 Crispps Leslie Alan Pharmaceutical aerosol formulation of salmeterol and fluticasone propionate
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
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