SI3150610T1 - Soli in polimorfi 8-fluoro-2-(4-(metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona - Google Patents

Soli in polimorfi 8-fluoro-2-(4-(metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona

Info

Publication number
SI3150610T1
SI3150610T1 SI201131808T SI201131808T SI3150610T1 SI 3150610 T1 SI3150610 T1 SI 3150610T1 SI 201131808 T SI201131808 T SI 201131808T SI 201131808 T SI201131808 T SI 201131808T SI 3150610 T1 SI3150610 T1 SI 3150610T1
Authority
SI
Slovenia
Prior art keywords
azepino
polymorphs
indol
methylamino
tetrahydro
Prior art date
Application number
SI201131808T
Other languages
English (en)
Inventor
Patricia Ann Basford
Anthony Michael Campeta
Adam Gillmore
Matthew Cameron Jones
Eleftherios Kougoulos
Suman Luthra
Robert Walton
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43859823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI3150610(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of SI3150610T1 publication Critical patent/SI3150610T1/sl

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/19—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
    • C07C57/13—Dicarboxylic acids
    • C07C57/145—Maleic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
SI201131808T 2010-02-12 2011-02-10 Soli in polimorfi 8-fluoro-2-(4-(metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona SI3150610T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30427710P 2010-02-12 2010-02-12
EP16183844.6A EP3150610B1 (en) 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one

Publications (1)

Publication Number Publication Date
SI3150610T1 true SI3150610T1 (sl) 2019-12-31

Family

ID=43859823

Family Applications (2)

Application Number Title Priority Date Filing Date
SI201131808T SI3150610T1 (sl) 2010-02-12 2011-02-10 Soli in polimorfi 8-fluoro-2-(4-(metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona
SI201131051A SI2534153T1 (sl) 2010-02-12 2011-02-10 Soli in polimorfi 8-fluoro-2-(4-((metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI201131051A SI2534153T1 (sl) 2010-02-12 2011-02-10 Soli in polimorfi 8-fluoro-2-(4-((metilamino)metil)fenil)-1,3,4,5-tetrahidro-6H-azepino (5,4,3-cd)indol-6-ona

Country Status (30)

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US (5) US8754072B2 (sl)
EP (4) EP4166558A1 (sl)
JP (6) JP5745283B2 (sl)
KR (2) KR102108226B1 (sl)
CN (2) CN104876937B (sl)
AR (2) AR080164A1 (sl)
AU (1) AU2011213944B2 (sl)
CA (2) CA2787881C (sl)
CY (3) CY1118319T1 (sl)
DK (2) DK2534153T3 (sl)
ES (2) ES2607806T3 (sl)
HK (1) HK1176617A1 (sl)
HR (2) HRP20161742T1 (sl)
HU (3) HUE030969T2 (sl)
IL (1) IL220921B (sl)
LT (3) LT3150610T (sl)
LU (1) LUC00093I2 (sl)
MX (1) MX343383B (sl)
NL (1) NL300958I2 (sl)
NO (1) NO2018039I1 (sl)
NZ (1) NZ601445A (sl)
PL (2) PL3150610T3 (sl)
PT (2) PT2534153T (sl)
RS (2) RS55487B1 (sl)
RU (1) RU2570198C2 (sl)
SG (2) SG10201406805RA (sl)
SI (2) SI3150610T1 (sl)
SM (1) SMT201600462B (sl)
TW (1) TWI545123B (sl)
WO (1) WO2011098971A1 (sl)

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CN114341162A (zh) 2019-07-10 2022-04-12 赛博克萨2公司 作为治疗剂的细胞毒素的肽缀合物
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