SI0770622T1 - Cyclic adhesion inhibitors - Google Patents

Cyclic adhesion inhibitors

Info

Publication number
SI0770622T1
SI0770622T1 SI9630172T SI9630172T SI0770622T1 SI 0770622 T1 SI0770622 T1 SI 0770622T1 SI 9630172 T SI9630172 T SI 9630172T SI 9630172 T SI9630172 T SI 9630172T SI 0770622 T1 SI0770622 T1 SI 0770622T1
Authority
SI
Slovenia
Prior art keywords
adhesion inhibitors
cyclic adhesion
cyclic
inhibitors
adhesion
Prior art date
Application number
SI9630172T
Other languages
English (en)
Slovenian (sl)
Inventor
Alfred Dr. Jonczyk
Simon Dr. Goodman
Beate Dr. Diefenbach
Arne Dr. Sutter
G�nter Dr. H�lzmann
Horst Prof. Kessler
Michael Dechantsreiter
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SI0770622T1 publication Critical patent/SI0770622T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Toxicology (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SI9630172T 1995-09-15 1996-08-31 Cyclic adhesion inhibitors SI0770622T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19534177A DE19534177A1 (de) 1995-09-15 1995-09-15 Cyclische Adhäsionsinhibitoren
EP96113972A EP0770622B1 (de) 1995-09-15 1996-08-31 Cyclische Adhäsionsinhibitoren

Publications (1)

Publication Number Publication Date
SI0770622T1 true SI0770622T1 (en) 2000-08-31

Family

ID=7772215

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9630172T SI0770622T1 (en) 1995-09-15 1996-08-31 Cyclic adhesion inhibitors

Country Status (29)

Country Link
US (1) US6001961A (es)
EP (1) EP0770622B1 (es)
JP (3) JP4115550B2 (es)
KR (1) KR100438244B1 (es)
CN (1) CN1203090C (es)
AR (1) AR003574A1 (es)
AT (1) ATE189461T1 (es)
AU (1) AU717574B2 (es)
BR (1) BR9603751A (es)
CA (1) CA2185489C (es)
CO (1) CO4750841A1 (es)
CZ (1) CZ286713B6 (es)
DE (2) DE19534177A1 (es)
DK (1) DK0770622T3 (es)
ES (1) ES2144179T3 (es)
GR (1) GR3033293T3 (es)
HU (1) HU224614B1 (es)
ID (1) ID18770A (es)
MX (1) MX9604100A (es)
NO (1) NO316946B1 (es)
PL (1) PL185125B1 (es)
PT (1) PT770622E (es)
RU (1) RU2157379C2 (es)
SI (1) SI0770622T1 (es)
SK (1) SK282391B6 (es)
TR (1) TR199600716A2 (es)
TW (1) TW517064B (es)
UA (1) UA49799C2 (es)
ZA (1) ZA967768B (es)

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US4792525A (en) * 1982-08-04 1988-12-20 La Jolla Cancer Research Foundation Tetrapeptide
US4517686A (en) * 1982-08-04 1985-05-21 La Jolla Cancer Research Foundation Polypeptide
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JP2945680B2 (ja) * 1988-09-09 1999-09-06 旭硝子株式会社 ペプチド誘導体およびその用途
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Also Published As

Publication number Publication date
TR199600716A3 (es) 1997-04-22
KR970015598A (ko) 1997-04-28
TW517064B (en) 2003-01-11
HUP9602507A3 (en) 1998-01-28
RU2157379C2 (ru) 2000-10-10
CA2185489A1 (en) 1997-03-16
HU224614B1 (hu) 2005-11-28
PL185125B1 (pl) 2003-02-28
AU717574B2 (en) 2000-03-30
ES2144179T3 (es) 2000-06-01
DE59604363D1 (de) 2000-03-09
AU6558096A (en) 1997-03-20
US6001961A (en) 1999-12-14
NO316946B1 (no) 2004-07-05
DE19534177A1 (de) 1997-03-20
BR9603751A (pt) 1998-06-02
HU9602507D0 (en) 1996-11-28
CZ264396A3 (en) 1997-04-16
PL316071A1 (en) 1997-03-17
MX9604100A (es) 1997-08-30
TR199600716A2 (tr) 1997-04-22
NO963853L (no) 1997-03-17
EP0770622A3 (de) 1997-07-02
DK0770622T3 (da) 2000-07-03
GR3033293T3 (en) 2000-09-29
SK116796A3 (en) 2001-05-10
CN1203090C (zh) 2005-05-25
PT770622E (pt) 2000-07-31
ZA967768B (en) 1997-04-07
JP2007186525A (ja) 2007-07-26
KR100438244B1 (ko) 2004-08-25
HUP9602507A2 (en) 1997-08-28
CN1149588A (zh) 1997-05-14
CO4750841A1 (es) 1999-03-31
JPH09132593A (ja) 1997-05-20
CA2185489C (en) 2007-05-08
UA49799C2 (uk) 2002-10-15
SK282391B6 (sk) 2002-01-07
EP0770622B1 (de) 2000-02-02
JP4115550B2 (ja) 2008-07-09
NO963853D0 (no) 1996-09-13
ATE189461T1 (de) 2000-02-15
AR003574A1 (es) 1998-08-05
EP0770622A2 (de) 1997-05-02
JP2007016042A (ja) 2007-01-25
ID18770A (id) 1998-05-07
JP4116062B2 (ja) 2008-07-09
CZ286713B6 (en) 2000-06-14

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