SG11201805368YA - Anthelmintic depsipeptide compounds - Google Patents

Anthelmintic depsipeptide compounds

Info

Publication number
SG11201805368YA
SG11201805368YA SG11201805368YA SG11201805368YA SG11201805368YA SG 11201805368Y A SG11201805368Y A SG 11201805368YA SG 11201805368Y A SG11201805368Y A SG 11201805368YA SG 11201805368Y A SG11201805368Y A SG 11201805368YA SG 11201805368Y A SG11201805368Y A SG 11201805368YA
Authority
SG
Singapore
Prior art keywords
international
animals
compounds
duluth
blvd
Prior art date
Application number
SG11201805368YA
Other languages
English (en)
Inventor
Hir De Fallois Loic Le
Gregory Pacofsky
Alan Long
Charles Meng
Hyoung Lee
Original Assignee
Merial Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Inc filed Critical Merial Inc
Publication of SG11201805368YA publication Critical patent/SG11201805368YA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K11/00Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
SG11201805368YA 2015-12-28 2016-12-14 Anthelmintic depsipeptide compounds SG11201805368YA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562272040P 2015-12-28 2015-12-28
PCT/US2016/066497 WO2017116702A1 (en) 2015-12-28 2016-12-14 Anthelmintic depsipeptide compounds

Publications (1)

Publication Number Publication Date
SG11201805368YA true SG11201805368YA (en) 2018-07-30

Family

ID=57868331

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201805368YA SG11201805368YA (en) 2015-12-28 2016-12-14 Anthelmintic depsipeptide compounds

Country Status (23)

Country Link
US (3) US10344056B2 (enExample)
EP (1) EP3397638B1 (enExample)
JP (1) JP6943859B2 (enExample)
KR (2) KR102427124B1 (enExample)
CN (1) CN108699052B (enExample)
AR (1) AR107249A1 (enExample)
AU (2) AU2016380868B2 (enExample)
BR (1) BR112018013369A2 (enExample)
CA (1) CA3009867C (enExample)
CL (1) CL2018001744A1 (enExample)
CO (1) CO2018006527A2 (enExample)
HK (1) HK1255391A1 (enExample)
HU (1) HUE065907T2 (enExample)
IL (1) IL260262B2 (enExample)
MX (1) MX2018007948A (enExample)
MY (1) MY194716A (enExample)
NZ (1) NZ743913A (enExample)
PH (1) PH12018501367B1 (enExample)
RU (2) RU2715556C2 (enExample)
SG (1) SG11201805368YA (enExample)
TW (1) TWI787165B (enExample)
UY (1) UY37050A (enExample)
WO (1) WO2017116702A1 (enExample)

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CN108699052B (zh) 2015-12-28 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
WO2018039508A1 (en) 2016-08-25 2018-03-01 Merial, Inc. Method for reducing unwanted effects in parasiticidal treatments
JP2020504710A (ja) 2016-11-16 2020-02-13 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性デプシペプチド化合物
PT3579696T (pt) 2017-02-08 2023-07-19 Boehringer Ingelheim Animal Health Usa Inc Modelo in vivo para infeção por vermes parasitários e métodos para avaliação de compostos antiparasíticos, que incluem compostos ativos contra a dirofilariose canina
EP3480195A1 (en) 2017-11-07 2019-05-08 Bayer Animal Health GmbH Method for the synthesis of cyclic depsipeptides
WO2019091975A1 (en) 2017-11-07 2019-05-16 Bayer Animal Health Gmbh Method for the synthesis of cyclic depsipeptides
NZ764359A (en) * 2017-11-29 2023-03-31 Zoetis Services Llc Endoparasitic depsipeptides
WO2019157241A1 (en) 2018-02-08 2019-08-15 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal compositions comprising eprinomectin and praziquantel, methods and uses thereof
AU2020205960B2 (en) 2019-01-10 2024-04-18 Zoetis Services Llc Anthelmintic laboratory animal model for heartworm
WO2020191091A1 (en) 2019-03-19 2020-09-24 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic aza-benzothiophene and aza-benzofuran compounds
EP4114358A4 (en) * 2020-03-06 2024-03-27 Lifemax Laboratories, Inc. TOPICAL PHARMACEUTICAL FORMULATIONS OF A CYCLIC DEPSIPEPTIDE
US11964977B2 (en) 2020-05-29 2024-04-23 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic heterocyclic compounds
US12161089B2 (en) 2020-12-21 2024-12-10 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal collar comprising isoxazoline compounds
US12258193B2 (en) 2022-02-17 2025-03-25 Boehringer Ingelheim Vetmedica Gmbh Method and system for providing a fluid product mailer
WO2025057117A1 (en) * 2023-09-15 2025-03-20 Animol Discovery, Inc. Antiparasitic cyclic depsipeptides

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Also Published As

Publication number Publication date
KR20180100349A (ko) 2018-09-10
PH12018501367B1 (en) 2022-10-21
TW201726670A (zh) 2017-08-01
JP2019504050A (ja) 2019-02-14
US11230571B2 (en) 2022-01-25
KR102427124B1 (ko) 2022-07-28
NZ743913A (en) 2019-04-26
UY37050A (es) 2017-07-31
AU2016380868A1 (en) 2018-07-19
US20170233438A1 (en) 2017-08-17
RU2018127195A3 (enExample) 2020-01-30
KR20220003663A (ko) 2022-01-10
IL260262A (en) 2018-07-31
US12018048B2 (en) 2024-06-25
AU2020200854B2 (en) 2021-08-05
EP3397638B1 (en) 2023-08-23
CO2018006527A2 (es) 2018-07-10
TWI787165B (zh) 2022-12-21
BR112018013369A2 (pt) 2019-02-19
EP3397638A1 (en) 2018-11-07
US10344056B2 (en) 2019-07-09
HUE065907T2 (hu) 2024-06-28
RU2018127195A (ru) 2020-01-30
CN108699052A (zh) 2018-10-23
CA3009867A1 (en) 2017-07-06
US20220098241A1 (en) 2022-03-31
CL2018001744A1 (es) 2018-08-17
US20190248840A1 (en) 2019-08-15
CA3009867C (en) 2022-05-31
RU2020107484A (ru) 2020-03-19
AU2020200854A1 (en) 2020-02-27
MY194716A (en) 2022-12-15
PH12018501367A1 (en) 2019-02-27
CN108699052B (zh) 2022-04-29
AU2016380868B2 (en) 2019-11-28
HK1255391A1 (zh) 2019-08-16
IL260262B2 (en) 2023-06-01
WO2017116702A1 (en) 2017-07-06
JP6943859B2 (ja) 2021-10-06
RU2715556C2 (ru) 2020-03-02
AR107249A1 (es) 2018-04-11
MX2018007948A (es) 2018-08-01

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