MX2018007948A - Compuestos depsipeptidicos como anthelminticos. - Google Patents

Compuestos depsipeptidicos como anthelminticos.

Info

Publication number
MX2018007948A
MX2018007948A MX2018007948A MX2018007948A MX2018007948A MX 2018007948 A MX2018007948 A MX 2018007948A MX 2018007948 A MX2018007948 A MX 2018007948A MX 2018007948 A MX2018007948 A MX 2018007948A MX 2018007948 A MX2018007948 A MX 2018007948A
Authority
MX
Mexico
Prior art keywords
compounds
animals
depsipeptide compounds
compositions
birds
Prior art date
Application number
MX2018007948A
Other languages
English (en)
Inventor
Ik Lee Hyoung
Long Alan
Pacofsky Gregory
Meng Charles
Le Hir De Fallois Loic
Original Assignee
Merial Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Inc filed Critical Merial Inc
Publication of MX2018007948A publication Critical patent/MX2018007948A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Compuestos depsipeptídicos cíclicos de fórmula (I) y composiciones que comprenden los compuestos que son eficaces contra parásitos que dañan a los animales, incluyendo a los humanos. Los compuestos y las composiciones se pueden usar para combatir parásitos dentro o sobre los animales incluyendo a mamíferos y aves. La invención también provee un método mejorado para erradicar, controlar y prevenir una infestación por parásitos en animales, incluyendo aves y mamíferos.
MX2018007948A 2015-12-28 2016-12-14 Compuestos depsipeptidicos como anthelminticos. MX2018007948A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562272040P 2015-12-28 2015-12-28
PCT/US2016/066497 WO2017116702A1 (en) 2015-12-28 2016-12-14 Anthelmintic depsipeptide compounds

Publications (1)

Publication Number Publication Date
MX2018007948A true MX2018007948A (es) 2018-08-01

Family

ID=57868331

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018007948A MX2018007948A (es) 2015-12-28 2016-12-14 Compuestos depsipeptidicos como anthelminticos.

Country Status (22)

Country Link
US (3) US10344056B2 (es)
EP (1) EP3397638B1 (es)
JP (1) JP6943859B2 (es)
KR (2) KR102427124B1 (es)
CN (1) CN108699052B (es)
AR (1) AR107249A1 (es)
AU (2) AU2016380868B2 (es)
BR (1) BR112018013369A2 (es)
CA (1) CA3009867C (es)
CL (1) CL2018001744A1 (es)
CO (1) CO2018006527A2 (es)
HK (1) HK1255391A1 (es)
IL (1) IL260262B2 (es)
MX (1) MX2018007948A (es)
MY (1) MY194716A (es)
NZ (1) NZ743913A (es)
PH (1) PH12018501367A1 (es)
RU (2) RU2715556C2 (es)
SG (1) SG11201805368YA (es)
TW (1) TWI787165B (es)
UY (1) UY37050A (es)
WO (1) WO2017116702A1 (es)

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MX2021001566A (es) * 2015-05-20 2022-09-12 Boehringer Ingelheim Animal Health Usa Inc Compuestos depsipeptidicos como anthelminticos.
WO2018039508A1 (en) 2016-08-25 2018-03-01 Merial, Inc. Method for reducing unwanted effects in parasiticidal treatments
US11382949B2 (en) 2016-11-16 2022-07-12 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
HRP20230870T1 (hr) 2017-02-08 2023-11-10 Boehringer Ingelheim Animal Health USA Inc. Model in vivo za infekciju parazitnim crvima i postupak ocjenjivanja antiparazitnih spojeva, uključujući spojeve koji djeluju protiv pseće dirofilarioze
EP3480195A1 (en) 2017-11-07 2019-05-08 Bayer Animal Health GmbH Method for the synthesis of cyclic depsipeptides
CN111757880A (zh) 2017-11-07 2020-10-09 拜耳动物保健有限责任公司 用于合成环状缩肽的方法
UA125155C2 (uk) * 2017-11-29 2022-01-19 Зоетіс Сервісіс Ллк Анти-ендопаразитарні депсипептиди
WO2019157241A1 (en) 2018-02-08 2019-08-15 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal compositions comprising eprinomectin and praziquantel, methods and uses thereof
US20220071183A1 (en) 2019-01-10 2022-03-10 Zoetis Services Llc Anthelmintic laboratory animal model for heartworm
CA3133100A1 (en) 2019-03-19 2020-09-24 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic aza-benzothiophene and aza-benzofuran compounds
BR112022024156A2 (pt) 2020-05-29 2023-02-14 Boehringer Ingelheim Animal Health Usa Inc Compostos heterocílicos antelmínticos
US20220201983A1 (en) 2020-12-21 2022-06-30 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal collar comprising isoxazoline compounds
WO2023156938A1 (en) 2022-02-17 2023-08-24 Boehringer Ingelheim Vetmedica Gmbh Method and system for providing a fluid product mailer

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NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
DE122005000058I1 (de) 1992-03-17 2006-04-27 Astellas Pharma Inc Depsipeptide, Herstellung und Anwendung
CA2155871A1 (en) 1993-02-19 1994-09-01 Makoto Ohyama Derivatives of cyclodepsipeptide pf 1022
DE4317432A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
EP0718293B1 (en) 1993-09-06 2002-03-13 Fujisawa Pharmaceutical Co., Ltd. Cyclodepsipeptide compound
SE9303657D0 (sv) 1993-11-05 1993-11-05 Astra Ab Short-acting dihydropyridines
DE4400464A1 (de) 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
DE4437198A1 (de) 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
DE19520275A1 (de) 1995-06-02 1996-12-05 Bayer Ag Endoparasitizide Mittel
WO1997011064A1 (fr) 1995-09-22 1997-03-27 Meiji Seika Kaisha, Ltd. Nouveaux derives depsipeptides cycliques de pf1022
PT953563E (pt) 1996-10-07 2003-08-29 Fujisawa Pharmaceutical Co Processo para a preparacao de derivados de depsipeptidos e novos compostos intermediarios para essa preparacao
DE19713626A1 (de) 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
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DE102008031284A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102008031283A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
WO2011069995A1 (en) 2009-12-11 2011-06-16 Bayer Animal Health Gmbh Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
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MX2021001566A (es) * 2015-05-20 2022-09-12 Boehringer Ingelheim Animal Health Usa Inc Compuestos depsipeptidicos como anthelminticos.

Also Published As

Publication number Publication date
AU2020200854B2 (en) 2021-08-05
KR20220003663A (ko) 2022-01-10
KR20180100349A (ko) 2018-09-10
US10344056B2 (en) 2019-07-09
CA3009867A1 (en) 2017-07-06
AR107249A1 (es) 2018-04-11
UY37050A (es) 2017-07-31
CO2018006527A2 (es) 2018-07-10
EP3397638A1 (en) 2018-11-07
JP6943859B2 (ja) 2021-10-06
RU2715556C2 (ru) 2020-03-02
RU2018127195A (ru) 2020-01-30
CA3009867C (en) 2022-05-31
HK1255391A1 (zh) 2019-08-16
RU2020107484A (ru) 2020-03-19
AU2020200854A1 (en) 2020-02-27
TWI787165B (zh) 2022-12-21
US20170233438A1 (en) 2017-08-17
CN108699052B (zh) 2022-04-29
US20190248840A1 (en) 2019-08-15
MY194716A (en) 2022-12-15
US20220098241A1 (en) 2022-03-31
NZ743913A (en) 2019-04-26
IL260262B2 (en) 2023-06-01
EP3397638B1 (en) 2023-08-23
JP2019504050A (ja) 2019-02-14
US11230571B2 (en) 2022-01-25
BR112018013369A2 (pt) 2019-02-19
AU2016380868A1 (en) 2018-07-19
PH12018501367A1 (en) 2019-02-27
RU2018127195A3 (es) 2020-01-30
KR102427124B1 (ko) 2022-07-28
TW201726670A (zh) 2017-08-01
AU2016380868B2 (en) 2019-11-28
CN108699052A (zh) 2018-10-23
IL260262A (en) 2018-07-31
WO2017116702A1 (en) 2017-07-06
CL2018001744A1 (es) 2018-08-17
SG11201805368YA (en) 2018-07-30

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