SG11201403345UA - Substituted annulated pyrimidines and triazines, and use thereof - Google Patents

Substituted annulated pyrimidines and triazines, and use thereof

Info

Publication number
SG11201403345UA
SG11201403345UA SG11201403345UA SG11201403345UA SG11201403345UA SG 11201403345U A SG11201403345U A SG 11201403345UA SG 11201403345U A SG11201403345U A SG 11201403345UA SG 11201403345U A SG11201403345U A SG 11201403345UA SG 11201403345U A SG11201403345U A SG 11201403345UA
Authority
SG
Singapore
Prior art keywords
triazines
pyrimidines
substituted annulated
annulated
substituted
Prior art date
Application number
SG11201403345UA
Other languages
English (en)
Inventor
Markus Follmann
Johannes-Peter Stasch
Gorden Redlich
Nils Griebenow
Dieter Lang
Frank Wunder
Walter Hübsch
Alexandros Vakalopoulos
Adrian Tersteegen
Original Assignee
Bayer Pharma AG
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47559479&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201403345U(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Pharma AG, Bayer Ip Gmbh filed Critical Bayer Pharma AG
Publication of SG11201403345UA publication Critical patent/SG11201403345UA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SG11201403345UA 2012-01-11 2013-01-10 Substituted annulated pyrimidines and triazines, and use thereof SG11201403345UA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102012200349A DE102012200349A1 (de) 2012-01-11 2012-01-11 Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung
PCT/EP2013/050381 WO2013104703A1 (de) 2012-01-11 2013-01-10 Substituierte annellierte pyrimidine und triazine und ihre verwendung

Publications (1)

Publication Number Publication Date
SG11201403345UA true SG11201403345UA (en) 2014-09-26

Family

ID=47559479

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201605655UA SG10201605655UA (en) 2012-01-11 2013-01-10 Substituted annulated pyrimidines and triazines, and use thereof
SG11201403345UA SG11201403345UA (en) 2012-01-11 2013-01-10 Substituted annulated pyrimidines and triazines, and use thereof

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG10201605655UA SG10201605655UA (en) 2012-01-11 2013-01-10 Substituted annulated pyrimidines and triazines, and use thereof

Country Status (29)

Country Link
US (2) US20140357637A1 (pt)
EP (1) EP2802592A1 (pt)
JP (1) JP6251183B2 (pt)
KR (1) KR20140114416A (pt)
CN (1) CN104812762B (pt)
AP (1) AP2014007844A0 (pt)
AU (1) AU2013208968A1 (pt)
BR (1) BR112014016971A8 (pt)
CA (1) CA2860855A1 (pt)
CL (1) CL2014001779A1 (pt)
CO (1) CO7000776A2 (pt)
CR (1) CR20140327A (pt)
CU (1) CU20140082A7 (pt)
DE (1) DE102012200349A1 (pt)
DO (1) DOP2014000160A (pt)
EA (1) EA025837B1 (pt)
EC (1) ECSP14008556A (pt)
GT (1) GT201400147A (pt)
HK (1) HK1211585A1 (pt)
IL (1) IL233460A0 (pt)
MA (1) MA35844B1 (pt)
MX (1) MX2014008201A (pt)
NZ (1) NZ626394A (pt)
PE (1) PE20142293A1 (pt)
PH (1) PH12014501595A1 (pt)
SG (2) SG10201605655UA (pt)
TN (1) TN2014000298A1 (pt)
WO (1) WO2013104703A1 (pt)
ZA (1) ZA201405042B (pt)

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DE102012200352A1 (de) 2012-01-11 2013-07-11 Bayer Intellectual Property Gmbh Substituierte, annellierte Imidazole und Pyrazole und ihre Verwendung
EP2822951B1 (de) 2012-03-06 2017-07-26 Bayer Intellectual Property GmbH Substituierte azabicyclen und ihre verwendung
ES2616042T3 (es) 2013-03-01 2017-06-09 Bayer Pharma Aktiengesellschaft Pirazolopiridinas sustituidas con bencilo y su uso
KR20150121007A (ko) 2013-03-01 2015-10-28 바이엘 파마 악티엔게젤샤프트 트리플루오르메틸-치환된 고리-융합된 피리미딘 및 그의 용도
MX2016000258A (es) 2013-07-10 2016-04-28 Bayer Pharma AG Bencil-1h-pirazolo[3,4-b]piridinas y su uso.

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DOP2014000160A (es) 2014-08-31
MA35844B1 (fr) 2014-12-01
US20150274754A1 (en) 2015-10-01
JP2015503605A (ja) 2015-02-02
CA2860855A1 (en) 2013-07-18
ECSP14008556A (es) 2015-12-31
CU20140082A7 (es) 2014-10-30
US20140357637A1 (en) 2014-12-04
ZA201405042B (en) 2016-08-31
NZ626394A (en) 2016-11-25
PH12014501595A1 (en) 2014-10-08
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WO2013104703A1 (de) 2013-07-18
SG10201605655UA (en) 2016-09-29
BR112014016971A2 (pt) 2017-06-13
AU2013208968A1 (en) 2014-07-24
JP6251183B2 (ja) 2017-12-20
CO7000776A2 (es) 2014-07-21
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CR20140327A (es) 2014-11-26
CN104812762B (zh) 2018-01-16
EP2802592A1 (de) 2014-11-19
HK1211585A1 (en) 2016-05-27
CN104812762A (zh) 2015-07-29
AP2014007844A0 (en) 2014-07-31
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MX2014008201A (es) 2014-08-08
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US9505786B2 (en) 2016-11-29
KR20140114416A (ko) 2014-09-26
EA025837B1 (ru) 2017-02-28
EA201491339A1 (ru) 2015-01-30
TN2014000298A1 (en) 2015-12-21
CL2014001779A1 (es) 2014-11-03

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