MA35844B1 - Pyrimidines et triazines annelées substituées et leur utilisation - Google Patents

Pyrimidines et triazines annelées substituées et leur utilisation

Info

Publication number
MA35844B1
MA35844B1 MA37178A MA37178A MA35844B1 MA 35844 B1 MA35844 B1 MA 35844B1 MA 37178 A MA37178 A MA 37178A MA 37178 A MA37178 A MA 37178A MA 35844 B1 MA35844 B1 MA 35844B1
Authority
MA
Morocco
Prior art keywords
triazines
pyrimidines
substituted
ringed
prophylaxis
Prior art date
Application number
MA37178A
Other languages
English (en)
Inventor
Nils Griebenow
Frank Wunder
Gorden Redlich
Walter Hübsch
Markus Follmann
Johannes-Peter Stasch
Dieter Lang
Alexandros Vakalopoulos
Adrian Tersteegen
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47559479&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA35844(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of MA35844B1 publication Critical patent/MA35844B1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Abstract

La présente invention concerne de nouvelles pyrimidines et triazines annelées substituées, leur procédé de fabrication, leur utilisation seules ou en combinaisons pour le traitement et/ou la prophylaxie de maladies, ainsi que leur utilisation pour fabriquer des médicaments destinés au traitement et/ou à la prophylaxie de maladies, notamment au traitement et/ou à la prophylaxie de maladies cardiovasculaires.
MA37178A 2012-01-11 2014-07-07 Pyrimidines et triazines annelées substituées et leur utilisation MA35844B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102012200349A DE102012200349A1 (de) 2012-01-11 2012-01-11 Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung
PCT/EP2013/050381 WO2013104703A1 (fr) 2012-01-11 2013-01-10 Pyrimidines et triazines annelées substituées et leur utilisation

Publications (1)

Publication Number Publication Date
MA35844B1 true MA35844B1 (fr) 2014-12-01

Family

ID=47559479

Family Applications (1)

Application Number Title Priority Date Filing Date
MA37178A MA35844B1 (fr) 2012-01-11 2014-07-07 Pyrimidines et triazines annelées substituées et leur utilisation

Country Status (29)

Country Link
US (2) US20140357637A1 (fr)
EP (1) EP2802592A1 (fr)
JP (1) JP6251183B2 (fr)
KR (1) KR20140114416A (fr)
CN (1) CN104812762B (fr)
AP (1) AP2014007844A0 (fr)
AU (1) AU2013208968A1 (fr)
BR (1) BR112014016971A8 (fr)
CA (1) CA2860855A1 (fr)
CL (1) CL2014001779A1 (fr)
CO (1) CO7000776A2 (fr)
CR (1) CR20140327A (fr)
CU (1) CU20140082A7 (fr)
DE (1) DE102012200349A1 (fr)
DO (1) DOP2014000160A (fr)
EA (1) EA025837B1 (fr)
EC (1) ECSP14008556A (fr)
GT (1) GT201400147A (fr)
HK (1) HK1211585A1 (fr)
IL (1) IL233460A0 (fr)
MA (1) MA35844B1 (fr)
MX (1) MX2014008201A (fr)
NZ (1) NZ626394A (fr)
PE (1) PE20142293A1 (fr)
PH (1) PH12014501595A1 (fr)
SG (2) SG10201605655UA (fr)
TN (1) TN2014000298A1 (fr)
WO (1) WO2013104703A1 (fr)
ZA (1) ZA201405042B (fr)

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Also Published As

Publication number Publication date
AU2013208968A1 (en) 2014-07-24
EA025837B1 (ru) 2017-02-28
AP2014007844A0 (en) 2014-07-31
SG11201403345UA (en) 2014-09-26
NZ626394A (en) 2016-11-25
US20150274754A1 (en) 2015-10-01
GT201400147A (es) 2015-04-06
US9505786B2 (en) 2016-11-29
CO7000776A2 (es) 2014-07-21
BR112014016971A8 (pt) 2017-07-04
EA201491339A1 (ru) 2015-01-30
WO2013104703A1 (fr) 2013-07-18
CL2014001779A1 (es) 2014-11-03
DE102012200349A1 (de) 2013-07-11
JP2015503605A (ja) 2015-02-02
PH12014501595A1 (en) 2014-10-08
CN104812762B (zh) 2018-01-16
JP6251183B2 (ja) 2017-12-20
US20140357637A1 (en) 2014-12-04
CA2860855A1 (fr) 2013-07-18
IL233460A0 (en) 2014-08-31
PE20142293A1 (es) 2014-12-19
BR112014016971A2 (pt) 2017-06-13
SG10201605655UA (en) 2016-09-29
CU20140082A7 (es) 2014-10-30
CR20140327A (es) 2014-11-26
EP2802592A1 (fr) 2014-11-19
KR20140114416A (ko) 2014-09-26
ECSP14008556A (es) 2015-12-31
MX2014008201A (es) 2014-08-08
DOP2014000160A (es) 2014-08-31
CN104812762A (zh) 2015-07-29
TN2014000298A1 (en) 2015-12-21
HK1211585A1 (en) 2016-05-27
ZA201405042B (en) 2016-08-31

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