SG10201903532XA - 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor - Google Patents

1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor

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Publication number
SG10201903532XA
SG10201903532XA SG10201903532XA SG10201903532XA SG10201903532XA SG 10201903532X A SG10201903532X A SG 10201903532XA SG 10201903532X A SG10201903532X A SG 10201903532XA SG 10201903532X A SG10201903532X A SG 10201903532XA SG 10201903532X A SG10201903532X A SG 10201903532XA
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Singapore
Prior art keywords
methylpyrimidin
pyrazol
pyrrolidin
methoxyethyl
fluorophenyl
Prior art date
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SG10201903532XA
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English (en)
Inventor
Shelley Allen
Steven W Andrews
Brian Baer
Zackary Crane
Weidong Liu
Daniel John Watson
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Array Biopharma Inc
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Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of SG10201903532XA publication Critical patent/SG10201903532XA/en

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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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SG10201903532XA 2014-05-15 2015-05-14 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor SG10201903532XA (en)

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SG10201903532XA SG10201903532XA (en) 2014-05-15 2015-05-14 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor

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RS53350B (en) 2008-09-22 2014-10-31 Array Biopharma, Inc. SUBSTITUTED COMPOUNDS OF IMIDASO [1,2-B] PYRIDASINE AS INK KINASE INHIBITORS
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CN109970614B (zh) 2023-01-13
SG11201609550PA (en) 2016-12-29
EP3564236A1 (en) 2019-11-06
PT3154959T (pt) 2019-09-24
PH12016502242A1 (en) 2017-01-09
US10835533B2 (en) 2020-11-17
WO2015175788A1 (en) 2015-11-19
PH12016502242B1 (en) 2017-01-09
CN109970614A (zh) 2019-07-05
DK3154959T3 (da) 2019-09-30
CN106459013A (zh) 2017-02-22
JP2017518981A (ja) 2017-07-13
RU2719489C2 (ru) 2020-04-17
AU2015259075B2 (en) 2019-01-24
MX2016014945A (es) 2017-03-27
PH12020500171A1 (en) 2021-02-08
JP2019085427A (ja) 2019-06-06
RS59286B1 (sr) 2019-10-31
RU2016149233A (ru) 2018-06-20
JP6499672B2 (ja) 2019-04-10
RU2016149233A3 (hu) 2018-12-03
CN106459013B (zh) 2019-10-25

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