SE461591B - Daunorubicin- och doxorubicin-analoger, deras framstaellning och terapeutisk komposition innehaallande dem - Google Patents

Daunorubicin- och doxorubicin-analoger, deras framstaellning och terapeutisk komposition innehaallande dem

Info

Publication number
SE461591B
SE461591B SE8300324A SE8300324A SE461591B SE 461591 B SE461591 B SE 461591B SE 8300324 A SE8300324 A SE 8300324A SE 8300324 A SE8300324 A SE 8300324A SE 461591 B SE461591 B SE 461591B
Authority
SE
Sweden
Prior art keywords
hydrogen
formula
daunorubicin
methyl
doxorubicin
Prior art date
Application number
SE8300324A
Other languages
English (en)
Swedish (sv)
Other versions
SE8300324L (sv
SE8300324D0 (sv
Inventor
S Penco
G Franchi
F Arcamone
A M Casazza
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of SE8300324D0 publication Critical patent/SE8300324D0/xx
Publication of SE8300324L publication Critical patent/SE8300324L/xx
Publication of SE461591B publication Critical patent/SE461591B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SE8300324A 1982-01-26 1983-01-21 Daunorubicin- och doxorubicin-analoger, deras framstaellning och terapeutisk komposition innehaallande dem SE461591B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8202080 1982-01-26

Publications (3)

Publication Number Publication Date
SE8300324D0 SE8300324D0 (sv) 1983-01-21
SE8300324L SE8300324L (sv) 1983-07-27
SE461591B true SE461591B (sv) 1990-03-05

Family

ID=10527864

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8300324A SE461591B (sv) 1982-01-26 1983-01-21 Daunorubicin- och doxorubicin-analoger, deras framstaellning och terapeutisk komposition innehaallande dem

Country Status (28)

Country Link
JP (1) JPS58128396A (fi)
KR (1) KR900006214B1 (fi)
AT (1) AT378776B (fi)
AU (1) AU551700B2 (fi)
BE (1) BE895687A (fi)
CA (1) CA1197237A (fi)
CH (1) CH657622A5 (fi)
CS (1) CS235979B2 (fi)
DE (1) DE3301489A1 (fi)
DK (1) DK157322C (fi)
ES (1) ES8403140A1 (fi)
FI (1) FI74977C (fi)
FR (1) FR2520365B1 (fi)
GB (1) GB2116169B (fi)
GR (1) GR77890B (fi)
HU (1) HU192784B (fi)
IE (1) IE53750B1 (fi)
IL (1) IL67709A (fi)
IT (1) IT1210482B (fi)
NL (1) NL8300150A (fi)
NO (1) NO153456C (fi)
NZ (1) NZ203047A (fi)
PH (1) PH19130A (fi)
PT (1) PT76113A (fi)
SE (1) SE461591B (fi)
SU (1) SU1187724A3 (fi)
YU (1) YU43536B (fi)
ZA (1) ZA83450B (fi)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2182926B (en) * 1985-11-19 1989-10-04 Erba Farmitalia Nitro anthracyclines, process for their preparation and use thereof
GB8708927D0 (en) * 1987-04-14 1987-05-20 Erba Farmitalia Chiral synthesis of anthracyclines

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1509875A (en) * 1976-06-14 1978-05-04 Farmaceutici Italia Optically active anthracyclinones and anthracycline glycosides
GB1573037A (en) * 1977-05-05 1980-08-13 Farmaceutici Italia Anthracyclines
ATE4387T1 (de) * 1979-07-04 1983-08-15 Farmitalia Carlo Erba S.P.A. Anthracyclin-glycoside, verfahren zu ihrer herstellung und sie enthaltende therapeutische zusammensetzung.
DE3100968A1 (de) * 1980-01-16 1982-01-14 Farmitalia Carlo Erba S.p.A., 20159 Milano Anthracyclinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
GB8301178D0 (en) 1983-02-16
CS235979B2 (en) 1985-05-15
ATA15683A (de) 1985-02-15
NL8300150A (nl) 1983-08-16
KR840003262A (ko) 1984-08-20
FI74977B (fi) 1987-12-31
IE53750B1 (en) 1989-02-01
FI830155L (fi) 1983-07-27
ZA83450B (en) 1983-10-26
DK157322B (da) 1989-12-11
DE3301489A1 (de) 1983-08-04
DK157322C (da) 1990-05-07
PT76113A (en) 1983-02-01
NO153456B (no) 1985-12-16
FR2520365A1 (fr) 1983-07-29
AU551700B2 (en) 1986-05-08
ES519255A0 (es) 1984-03-01
IE830144L (en) 1983-07-26
ES8403140A1 (es) 1984-03-01
NO830234L (no) 1983-07-27
KR900006214B1 (ko) 1990-08-25
JPS58128396A (ja) 1983-07-30
SU1187724A3 (ru) 1985-10-23
CH657622A5 (it) 1986-09-15
SE8300324L (sv) 1983-07-27
IL67709A (en) 1986-03-31
FI74977C (fi) 1988-04-11
HU192784B (en) 1987-07-28
GB2116169A (en) 1983-09-21
FI830155A0 (fi) 1983-01-17
PH19130A (en) 1986-01-08
DK27683D0 (da) 1983-01-25
BE895687A (fr) 1983-05-16
NO153456C (no) 1986-03-26
IL67709A0 (en) 1983-05-15
GR77890B (fi) 1984-09-25
GB2116169B (en) 1985-09-04
IT1210482B (it) 1989-09-14
YU43536B (en) 1989-08-31
NZ203047A (en) 1985-10-11
YU8983A (en) 1986-02-28
AU1052583A (en) 1983-08-04
CA1197237A (en) 1985-11-26
AT378776B (de) 1985-09-25
JPS6328436B2 (fi) 1988-06-08
FR2520365B1 (fr) 1985-07-12
SE8300324D0 (sv) 1983-01-21
DK27683A (da) 1983-07-27
DE3301489C2 (fi) 1988-01-28
IT8319147A0 (it) 1983-01-18

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