SE440780B - Nya 11beta-substituerade mellanprodukter till anvendning vid framstellning av steroidderivat - Google Patents

Nya 11beta-substituerade mellanprodukter till anvendning vid framstellning av steroidderivat

Info

Publication number
SE440780B
SE440780B SE7714612A SE7714612A SE440780B SE 440780 B SE440780 B SE 440780B SE 7714612 A SE7714612 A SE 7714612A SE 7714612 A SE7714612 A SE 7714612A SE 440780 B SE440780 B SE 440780B
Authority
SE
Sweden
Prior art keywords
hydroxy
group
methyl
compound
estr
Prior art date
Application number
SE7714612A
Other languages
English (en)
Swedish (sv)
Other versions
SE7714612L (sv
Inventor
J G Teutsch
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of SE7714612L publication Critical patent/SE7714612L/
Publication of SE440780B publication Critical patent/SE440780B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/006—Ketals at position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
SE7714612A 1977-01-13 1977-12-21 Nya 11beta-substituerade mellanprodukter till anvendning vid framstellning av steroidderivat SE440780B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7700857A FR2377417A1 (fr) 1977-01-13 1977-01-13 Nouveaux derives steroides substitues en 11b, ainsi que leur procede de preparation

Publications (2)

Publication Number Publication Date
SE7714612L SE7714612L (sv) 1978-07-14
SE440780B true SE440780B (sv) 1985-08-19

Family

ID=9185436

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7714612A SE440780B (sv) 1977-01-13 1977-12-21 Nya 11beta-substituerade mellanprodukter till anvendning vid framstellning av steroidderivat

Country Status (14)

Country Link
US (1) US4147695A (fr)
JP (1) JPS5390253A (fr)
BE (1) BE862868A (fr)
CA (1) CA1122971A (fr)
CH (1) CH629823A5 (fr)
DE (1) DE2801415A1 (fr)
DK (1) DK164324C (fr)
FR (1) FR2377417A1 (fr)
GB (1) GB1595131A (fr)
HU (1) HU175290B (fr)
IE (1) IE46300B1 (fr)
LU (1) LU78860A1 (fr)
NL (1) NL7800365A (fr)
SE (1) SE440780B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE23167T1 (de) * 1981-01-09 1986-11-15 Roussel Uclaf In stellung 11 substituierte steroidzwischenprodukte und verfahren zu ihrer herstellung.
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1 (fr) * 1982-03-01 1986-02-14 Roussel Uclaf Nouveaux produits derives de la structure 3-ceto 4,9 19-nor steroides, leur procede de preparation et leur application comme medicaments
FR2586021B1 (fr) * 1985-08-09 1988-10-14 Roussel Uclaf Nouveaux produits derives de la structure 5a-oh d 9(10) 19-nor steroides
US5929262A (en) * 1995-03-30 1999-07-27 The United States Of America As Represented By The Department Of Health And Human Services Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2880233A (en) * 1956-01-05 1959-03-31 Sterling Drug Inc Compounds of the perhydrochrysene and related series and preparation thereof
US3299108A (en) * 1965-10-18 1967-01-17 Searle & Co 17alpha-alkynyl/alkenyl-13beta-alkyl-11-alkylgona-1, 3, 5 (10)-triene-3, 17beta-diols, ethers and esters thereof and intermediates thereto
US3346602A (en) * 1966-10-12 1967-10-10 Searle & Co 13beta-alkyl-11-alkylgona-1, 3, 5 (10)-trien-17-ones, ethers and esters thereof
FR2235949B1 (fr) * 1973-06-18 1978-03-17 Roussel Uclaf
FR2237906A1 (en) * 1973-06-26 1975-02-14 Roussel Uclaf 11-oxo estr-9-ene derivs. - intermediates in the synthesis of steroids

Also Published As

Publication number Publication date
DE2801415A1 (de) 1978-07-20
BE862868A (fr) 1978-07-12
FR2377417B1 (fr) 1979-04-20
FR2377417A1 (fr) 1978-08-11
IE780077L (en) 1978-07-13
JPS5390253A (en) 1978-08-08
NL7800365A (nl) 1978-07-17
DK13778A (da) 1978-07-14
CA1122971A (fr) 1982-05-04
HU175290B (hu) 1980-06-28
DK164324C (da) 1992-11-02
JPS631320B2 (fr) 1988-01-12
IE46300B1 (en) 1983-04-20
CH629823A5 (fr) 1982-05-14
LU78860A1 (fr) 1978-09-18
DK164324B (da) 1992-06-09
SE7714612L (sv) 1978-07-14
GB1595131A (en) 1981-08-05
US4147695A (en) 1979-04-03

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