RU94006013A - Производные оксазолидиндиона, их получение и применение - Google Patents

Производные оксазолидиндиона, их получение и применение

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Publication number
RU94006013A
RU94006013A RU94006013/04A RU94006013A RU94006013A RU 94006013 A RU94006013 A RU 94006013A RU 94006013/04 A RU94006013/04 A RU 94006013/04A RU 94006013 A RU94006013 A RU 94006013A RU 94006013 A RU94006013 A RU 94006013A
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Russia
Prior art keywords
oxazolidindion
derivatives
production
application
substituted
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Application number
RU94006013/04A
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English (en)
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RU2126797C1 (ru
Inventor
Сохда Такаси
Икеда Хитоси
Момосе Ю
Имаи Сатико
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Такеда Кемикал Индастриз, Лтд.
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Application filed by Такеда Кемикал Индастриз, Лтд. filed Critical Такеда Кемикал Индастриз, Лтд.
Publication of RU94006013A publication Critical patent/RU94006013A/ru
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Publication of RU2126797C1 publication Critical patent/RU2126797C1/ru

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Claims (1)

  1. Предложены новые соединения 2, 4 - оксазолидиндиона формулы:
    Figure 00000001

    где R является углеводородным остатком или гетероциклической группой, которые могут быть замещенными; Y представляет собой -CO-, CH(OH)- или NR3- (где R3 - алкил группа, которая может быть замещенной); m - 0 или 1; n - 0,1 или 2; X - CH или N; А - двухвалентный прямой или разветвленный остаток углеводородной цепи, содержащей 1 - 7 атомов углерода; R1 и R2 - каждый является водородом или алкил группой или R1 и R2 комбинируются друг с другом с образованием 5- - 6-членной гетероциклической группы, возможно содержащей азот, L и M каждый является водородом или L и M комбинируются друг с другом с образованием связи или его фармацевтически приемлемые соли, имеющие прекрасную гипогликемическую и гиполипидемическую активность, и пригодны для использования в качестве лекарственных препаратов для лечения диабета и гиперлипидемии.
RU94006013A 1993-02-26 1994-02-25 Производные 2,4-оксазолидиндиона или их фармацевтически приемлемая соль, способы их получения, лекарственная композиция, оказывающая гипогликемическое и гиполипидемическое действие, способ снижения содержания сахара и липидов в крови при лечении млекопитающих, страдающих диабетом или гиперлипидимией RU2126797C1 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP05-038236 1993-02-26
JP3823693 1993-02-26
JP05-197304 1993-08-09
JP19730493 1993-08-09

Publications (2)

Publication Number Publication Date
RU94006013A true RU94006013A (ru) 1995-09-27
RU2126797C1 RU2126797C1 (ru) 1999-02-27

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Family Applications (1)

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RU94006013A RU2126797C1 (ru) 1993-02-26 1994-02-25 Производные 2,4-оксазолидиндиона или их фармацевтически приемлемая соль, способы их получения, лекарственная композиция, оказывающая гипогликемическое и гиполипидемическое действие, способ снижения содержания сахара и липидов в крови при лечении млекопитающих, страдающих диабетом или гиперлипидимией

Country Status (18)

Country Link
US (4) US5665748A (ru)
EP (1) EP0612743B1 (ru)
JP (2) JP3328720B2 (ru)
KR (1) KR940019699A (ru)
CN (1) CN1098411A (ru)
AT (1) ATE157975T1 (ru)
AU (1) AU673034B2 (ru)
CA (1) CA2116387C (ru)
DE (1) DE69405425T2 (ru)
DK (1) DK0612743T3 (ru)
ES (1) ES2108375T3 (ru)
FI (1) FI940904A (ru)
GR (1) GR3025342T3 (ru)
HU (1) HUT70159A (ru)
NO (1) NO305079B1 (ru)
PH (1) PH31468A (ru)
RU (1) RU2126797C1 (ru)
TW (1) TW268952B (ru)

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