RU2652987C2 - Производные пиридинона в качестве ингибиторов трансглутаминазы тканей - Google Patents

Производные пиридинона в качестве ингибиторов трансглутаминазы тканей Download PDF

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RU2652987C2
RU2652987C2 RU2015104969A RU2015104969A RU2652987C2 RU 2652987 C2 RU2652987 C2 RU 2652987C2 RU 2015104969 A RU2015104969 A RU 2015104969A RU 2015104969 A RU2015104969 A RU 2015104969A RU 2652987 C2 RU2652987 C2 RU 2652987C2
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ylamino
oxo
dihydropyridin
oxoethyl
oxohept
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RU2015104969A
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RU2015104969A (ru
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Кристиан БЮХОЛЬД
Уве Герлах
Мартин ХИЛС
Ральф ПАСТЕРНАК
Йоханнес ВЕБЕР
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Цедира Гмбх
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    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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RU2015104969A 2012-07-17 2013-07-12 Производные пиридинона в качестве ингибиторов трансглутаминазы тканей RU2652987C2 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP12176776.8 2012-07-17
EP12176776.8A EP2687511A1 (de) 2012-07-17 2012-07-17 Pyridinonderivate als Gewebetransglutaminaseinhibitoren
US201261741871P 2012-07-30 2012-07-30
US61/741,871 2012-07-30
PCT/EP2013/064789 WO2014012858A1 (de) 2012-07-17 2013-07-12 Pyridinonderivate als gewebetransglutaminaseinhibitoren

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RU2015104969A RU2015104969A (ru) 2016-09-10
RU2652987C2 true RU2652987C2 (ru) 2018-05-04

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WO2017021111A1 (en) 2015-08-05 2017-02-09 Ratiopharm Gmbh New crystalline form and acetic acid adducts of palbociclib
WO2019201432A1 (en) * 2018-04-17 2019-10-24 Zedira Gmbh Inhibitors of blood coagulation factor xiii
TWI825144B (zh) 2018-08-10 2023-12-11 美商思達利醫藥公司 第二型轉麩醯胺酸酶(tg2)抑制劑
CN118027041A (zh) * 2019-05-31 2024-05-14 西藏海思科制药有限公司 一种btk抑制剂环衍生物及其制备方法和药学上的应用
IL297020A (en) * 2020-04-24 2022-12-01 Dr Falk Pharma Gmbh A systemic preparation of a pyridonone derivative related to tg2
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