RU2646483C2 - Твердые фармацевтические композиции для перорального введения на основе изоксазолиновых соединений - Google Patents

Твердые фармацевтические композиции для перорального введения на основе изоксазолиновых соединений Download PDF

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RU2646483C2
RU2646483C2 RU2014144360A RU2014144360A RU2646483C2 RU 2646483 C2 RU2646483 C2 RU 2646483C2 RU 2014144360 A RU2014144360 A RU 2014144360A RU 2014144360 A RU2014144360 A RU 2014144360A RU 2646483 C2 RU2646483 C2 RU 2646483C2
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compound
isoxazoline
nhch
methyl
composition
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RU2014144360A
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English (en)
Russian (ru)
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RU2014144360A (ru
Inventor
Кейт ФРИХОФ
Ники УОЛДРОН
Юрген ЛУТЦ
Фрэнк Гуэрино
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Интервет Интернэшнл Б.В.
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    • AHUMAN NECESSITIES
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    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Physics & Mathematics (AREA)
  • Biomedical Technology (AREA)
  • Biochemistry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Mechanical Engineering (AREA)
  • Botany (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
RU2014144360A 2012-04-04 2013-04-03 Твердые фармацевтические композиции для перорального введения на основе изоксазолиновых соединений RU2646483C2 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP12163198.0 2012-04-04
EP12163198 2012-04-04
US201361782028P 2013-03-14 2013-03-14
US61/782,028 2013-03-14
PCT/EP2013/056992 WO2013150055A1 (en) 2012-04-04 2013-04-03 Solid oral pharmaceutical compositions for isoxazoline compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
RU2018104704A Division RU2772279C2 (ru) 2012-04-04 2013-04-03 Твердые фармацевтические композиции для перорального введения на основе изоксазолиновых соединений

Publications (2)

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RU2014144360A RU2014144360A (ru) 2016-05-27
RU2646483C2 true RU2646483C2 (ru) 2018-03-05

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Application Number Title Priority Date Filing Date
RU2014144360A RU2646483C2 (ru) 2012-04-04 2013-04-03 Твердые фармацевтические композиции для перорального введения на основе изоксазолиновых соединений
RU2014144001A RU2632965C2 (ru) 2012-04-04 2013-04-03 Мягкие жевательные фармацевтические продукты
RU2017133665A RU2765231C2 (ru) 2012-04-04 2013-04-03 Мягкие жевательные фармацевтические продукты

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RU2014144001A RU2632965C2 (ru) 2012-04-04 2013-04-03 Мягкие жевательные фармацевтические продукты
RU2017133665A RU2765231C2 (ru) 2012-04-04 2013-04-03 Мягкие жевательные фармацевтические продукты

Country Status (14)

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US (15) US9770440B2 (OSRAM)
EP (2) EP2833867B2 (OSRAM)
JP (2) JP6088637B2 (OSRAM)
KR (1) KR102077874B1 (OSRAM)
CN (4) CN109010296A (OSRAM)
AU (7) AU2013245011B2 (OSRAM)
BR (3) BR112014024832B1 (OSRAM)
CA (2) CA2869242C (OSRAM)
ES (1) ES2633611T5 (OSRAM)
FI (1) FI2833866T4 (OSRAM)
NZ (1) NZ631100A (OSRAM)
RU (3) RU2646483C2 (OSRAM)
WO (2) WO2013150052A1 (OSRAM)
ZA (2) ZA201406968B (OSRAM)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2847348C1 (ru) * 2024-04-27 2025-10-03 Общество С Ограниченной Ответственностью "Научно-Исследовательский Центр "Фарматол" Противопаразитарное средство для лечения и профилактики эктопаразитозов собак.

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SG11201404595TA (en) 2012-02-06 2014-09-26 Merial Ltd Parasiticidal oral veterinary compositions comprising systemically-acting active agents, methods and uses thereof
BR112014024832B1 (pt) 2012-04-04 2022-05-31 Intervet International B.V. Método para a preparação de uma composição farmacêutica veterinária mastigável macia, composição farmacêutica, e, uso da composição
US9532946B2 (en) 2012-11-20 2017-01-03 Intervet Inc. Manufacturing of semi-plastic pharmaceutical dosage units
ES2742815T3 (es) 2013-12-10 2020-02-17 Intervet Int Bv Uso antiparasitario de compuestos de isoxazolina
HUE063842T2 (hu) 2013-12-20 2024-02-28 Intervet Int Bv Izoxazolin vegyületek felhasználása baromfiban
WO2015091898A1 (en) 2013-12-20 2015-06-25 Intervet International B.V. Isoxazoline compositions and use thereof in the prevention or treatment of parasite infestations in animals
MX2017005721A (es) * 2014-11-03 2017-07-28 Zoetis Services Llc Composicion veterinaria masticable agradable al paladar.
PL3236960T3 (pl) 2014-12-22 2025-07-07 Intervet International B.V. Fluralaner do zastosowania w leczeniu demodekozy
UY36570A (es) 2015-02-26 2016-10-31 Merial Inc Formulaciones inyectables de acción prolongada que comprenden un agente activo isoxazolina, métodos y usos de las mismas
UY37137A (es) 2016-02-24 2017-09-29 Merial Inc Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos
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