RU2017123878A - Пиколинамидные соединения с фунгицидной активностью - Google Patents
Пиколинамидные соединения с фунгицидной активностью Download PDFInfo
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- RU2017123878A RU2017123878A RU2017123878A RU2017123878A RU2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A RU 2017123878 A RU2017123878 A RU 2017123878A
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- Prior art keywords
- alkyl
- hydrogen
- optionally substituted
- aryl
- compound
- Prior art date
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- 230000000855 fungicidal effect Effects 0.000 title 1
- IBBMAWULFFBRKK-UHFFFAOYSA-N picolinamide Chemical class NC(=O)C1=CC=CC=N1 IBBMAWULFFBRKK-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 claims 32
- 150000001875 compounds Chemical class 0.000 claims 29
- 229910052739 hydrogen Inorganic materials 0.000 claims 29
- 239000001257 hydrogen Substances 0.000 claims 29
- 125000003118 aryl group Chemical group 0.000 claims 22
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical group [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 21
- 125000003342 alkenyl group Chemical group 0.000 claims 12
- 125000003545 alkoxy group Chemical group 0.000 claims 6
- 150000002431 hydrogen Chemical class 0.000 claims 6
- 125000002252 acyl group Chemical group 0.000 claims 3
- 229910052736 halogen Inorganic materials 0.000 claims 3
- 150000002367 halogens Chemical class 0.000 claims 3
- 125000000623 heterocyclic group Chemical group 0.000 claims 3
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- 125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 claims 1
- 125000000740 n-pentyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
- A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
- A01N37/44—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio analogue of a carboxylic group, e.g. amino-carboxylic acids
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
Claims (45)
1. Соединение формулы I
I
где X представляет собой водород или C(О)R5;
Y представляет собой водород, C(O)R5 или Q;
Q представляет собой
R1 и R11 независимо выбраны из водорода или алкила, необязательно замещенного 0, 1 или несколькими R8; альтернативно, R1 и R11 могут быть взяты вместе с образованием 3-6-членного насыщенного или частично насыщенного карбоцикла или гетероцикла, необязательно замещенного 0, 1 или несколькими R8;
R2 и R12 независимо выбраны из водорода, алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8;
R3 выбран из водорода, C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8;
R4 выбран из алкила, арила или ацила, каждый необязательно замещен 0, 1 или несколькими R8;
R5 выбран из алкокси или бензилокси, каждый необязательно замещен 0, 1 или несколькими R8;
R6 выбран из водорода, алкокси или галогена, каждый необязательно замещен 0, 1 или несколькими R8;
R7 выбран из водорода, -С(О)R9 или -CH2OC(О)R9;
R8 выбран из водорода, алкила, арила, ацила, галогена, алкенила, алкокси или гетероциклила, каждый необязательно замещен 0, 1 или несколькими R10;
R9 выбран из алкила, алкокси или арила, каждый необязательно замещен 0, 1 или несколькими R8;
R10 выбран из водорода, алкила, арила, ацила, галогена, алкенила, алкокси или гетероциклила.
2. Соединение по п.1, где Х и Y представляют собой водород.
3. Соединение по п.2, где R1 и R11 независимо выбраны из водорода или алкила.
4. Соединение по п.2, где R2 и R12 независимо выбраны из водорода или алкила.
5. Соединение по п.2, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
6. Соединение по п.2, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
7. Соединение по п.2, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
8. Соединение по п.1, где Х представляет собой C(O)R5, и Y представляет собой водород.
9. Соединение по п.8, где R1 и R11 независимо выбраны из водорода или алкила.
10. Соединение по п.8, где R2 и R12 независимо выбраны из водорода или алкила.
11. Соединение по п.8, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
12. Соединение по п.8, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
13. Соединение по п.8, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
14. Соединение по п.1, где X представляет собой водород и Y представляет собой Q.
15. Соединение по п.14, где R6 представляет собой алкокси.
16. Соединение по п.15, где R7 представляет собой водород.
17. Соединение по п.16, где R1 и R11 независимо выбраны из водорода или алкила.
18. Соединение по п.16, где R2 и R12 независимо выбраны из водорода или алкила.
19. Соединение по п.16, где R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
20. Соединение по п.16, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
21. Соединение по п.16, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
22. Соединение по п.15, где R7 выбран из -C(O)R9 или -CH2OC(O)R9.
23. Соединение по п.22, где R9 представляет собой алкил, необязательно замещенный 0, 1 или несколькими R8.
24. Соединение по п.23, где R1 и R11 независимо выбраны из водорода или алкила.
25. Соединение по п.23, где R2 и R12 независимо выбраны из водорода или алкила.
26. Соединение по п.23, где R3 выбран из алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8.
27. Соединение по п.23, где R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
28. Соединение по п.23, где R1 и R11 независимо выбраны из водорода или алкила, R2 и R12 независимо выбраны из водорода или алкила, R3 выбран из C2-C6 алкила, арила или алкенила, каждый необязательно замещен 0, 1 или несколькими R8, и R4 выбран из алкила или арила, каждый необязательно замещен 0, 1 или несколькими R8.
29. Соединение по п.28, где R9 выбран из -CH3, -CH2OCH2CH3, -CH2CH2OCH3, -CH(CH3)2, -CH2CH2CH2CH3, -циклопропила.
Applications Claiming Priority (17)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462098097P | 2014-12-30 | 2014-12-30 | |
US201462098089P | 2014-12-30 | 2014-12-30 | |
US62/098,089 | 2014-12-30 | ||
US62/098,097 | 2014-12-30 | ||
US201562255131P | 2015-11-13 | 2015-11-13 | |
US201562255125P | 2015-11-13 | 2015-11-13 | |
US201562255152P | 2015-11-13 | 2015-11-13 | |
US201562255163P | 2015-11-13 | 2015-11-13 | |
US201562255168P | 2015-11-13 | 2015-11-13 | |
US201562255144P | 2015-11-13 | 2015-11-13 | |
US62/255,144 | 2015-11-13 | ||
US62/255,125 | 2015-11-13 | ||
US62/255,168 | 2015-11-13 | ||
US62/255,152 | 2015-11-13 | ||
US62/255,163 | 2015-11-13 | ||
US62/255,131 | 2015-11-13 | ||
PCT/US2015/067113 WO2016109289A1 (en) | 2014-12-30 | 2015-12-21 | Picolinamide compounds with fungicidal activity |
Publications (3)
Publication Number | Publication Date |
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RU2017123878A true RU2017123878A (ru) | 2019-01-31 |
RU2017123878A3 RU2017123878A3 (ru) | 2019-02-20 |
RU2687160C2 RU2687160C2 (ru) | 2019-05-07 |
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Application Number | Title | Priority Date | Filing Date |
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RU2017123854A RU2704867C2 (ru) | 2014-12-30 | 2015-12-21 | Применение соединений пиколинамида с фунгицидным действием |
RU2017123878A RU2687160C2 (ru) | 2014-12-30 | 2015-12-21 | Пиколинамидные соединения с фунгицидной активностью |
Family Applications Before (1)
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RU2017123854A RU2704867C2 (ru) | 2014-12-30 | 2015-12-21 | Применение соединений пиколинамида с фунгицидным действием |
Country Status (17)
Country | Link |
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US (2) | US10433555B2 (ru) |
EP (2) | EP3240412A4 (ru) |
JP (2) | JP2018500362A (ru) |
KR (2) | KR20170100550A (ru) |
CN (2) | CN107426999B (ru) |
AU (4) | AU2015374458B2 (ru) |
BR (2) | BR112017013758B1 (ru) |
CA (2) | CA2972413A1 (ru) |
CO (2) | CO2017006852A2 (ru) |
IL (2) | IL253092A0 (ru) |
MX (2) | MX2017008408A (ru) |
NZ (2) | NZ732573A (ru) |
RU (2) | RU2704867C2 (ru) |
TW (2) | TW201625516A (ru) |
UY (2) | UY36489A (ru) |
WO (2) | WO2016109288A1 (ru) |
ZA (2) | ZA201704555B (ru) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2972034A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Picolinamides with fungicidal activity |
WO2016109288A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Use of picolinamide compounds with fungicidal activity |
BR122019026066B1 (pt) | 2014-12-30 | 2022-01-18 | Dow Agrosciences Llc | Compostos de picolinamida |
CA2972403A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Picolinamide compounds with fungicidal activity |
BR112017013608B8 (pt) * | 2014-12-30 | 2022-08-23 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
TW201811803A (zh) * | 2016-08-30 | 2018-04-01 | 美商陶氏農業科學公司 | 具有殺真菌活性之吡啶並-1,3-噁嗪-2,4-二酮化合物 |
WO2018045010A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Pyrido-1,3-oxazine-2,4-dione compounds with fungicidal activity |
WO2018044996A1 (en) * | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Picolinamides as fungicides |
US10111432B2 (en) | 2016-08-30 | 2018-10-30 | Dow Agrosciences Llc | Picolinamide N-oxide compounds with fungicidal activity |
WO2018044991A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Thiopicolinamide compounds with fungicidal activity |
BR102018000183B1 (pt) * | 2017-01-05 | 2023-04-25 | Dow Agrosciences Llc | Picolinamidas, composição para controle de um patógeno fúngico, e método para controle e prevenção de um ataque por fungos em uma planta |
JP7082110B2 (ja) | 2017-03-29 | 2022-06-07 | テルモ株式会社 | アジュバント組成物およびこれを含むワクチン組成物並びに薬剤キット |
TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
WO2018204438A1 (en) | 2017-05-02 | 2018-11-08 | Dow Agrosciences Llc | Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses |
TW201842851A (zh) | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
UY37912A (es) | 2017-10-05 | 2019-05-31 | Syngenta Participations Ag | Derivados de picolinamida fungicidas que portan grupos terminales heteroarilo o heteroariloxi |
UY37913A (es) * | 2017-10-05 | 2019-05-31 | Syngenta Participations Ag | Derivados de picolinamida fungicidas que portan un grupo terminal cuaternario |
WO2019068819A1 (en) | 2017-10-06 | 2019-04-11 | Syngenta Participations Ag | PYRROLE DERIVATIVES ACTIVE ON THE PESTICIDE PLAN |
BR112020009659A2 (pt) | 2017-11-15 | 2020-11-10 | Syngenta Participations Ag | derivados picolinamida microbiocidas |
WO2019121149A1 (en) | 2017-12-19 | 2019-06-27 | Syngenta Participations Ag | Microbiocidal picolinamide derivatives |
BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
EP3802493A1 (en) | 2018-05-25 | 2021-04-14 | Syngenta Participations Ag | Microbiocidal picolinamide derivatives |
EP3866597A4 (en) | 2018-10-15 | 2022-06-29 | Corteva Agriscience LLC | Methods for sythesis of oxypicolinamides |
US20220167615A1 (en) * | 2019-04-10 | 2022-06-02 | Syngenta Crop Protection Ag | Fungicidal compositions |
WO2020208095A1 (en) | 2019-04-10 | 2020-10-15 | Syngenta Crop Protection Ag | Microbiocidal picolinamide derivatives |
US20220264877A1 (en) * | 2019-07-05 | 2022-08-25 | Syngenta Crop Protection Ag | Microbiocidal picolinamide derivatives |
AR123501A1 (es) | 2020-09-15 | 2022-12-07 | Pi Industries Ltd | Nuevos compuestos de picolinamida para combatir hongos fitopatógenos |
AR123502A1 (es) | 2020-09-15 | 2022-12-07 | Pi Industries Ltd | Nuevos compuestos de picolinamida para combatir hongos fitopatógenos |
CN113429338B (zh) * | 2021-05-20 | 2023-05-02 | 陕西泰合利华工业有限公司 | 一种合成氟吡菌酰胺的方法 |
Family Cites Families (111)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4051173A (en) | 1974-04-02 | 1977-09-27 | Merck Patent Gesellschaft Mit Beschrankter Haftung | Phenoxyalkanol derivatives |
JPS51133423A (en) * | 1975-03-15 | 1976-11-19 | Nissan Chem Ind Ltd | Controlling agents against soil disease germs |
US4588735A (en) | 1983-02-28 | 1986-05-13 | Chevron Research Company | Fungicidal (trihalophenoxy or trihalophenthio) alkylaminoalkyl pyridines and pyrroles |
FR2649699A1 (fr) | 1989-07-13 | 1991-01-18 | Rhone Poulenc Agrochimie | 4-phenyl pyrimidine fongicides |
IL91418A (en) | 1988-09-01 | 1997-11-20 | Rhone Poulenc Agrochimie | (hetero) cyclic amide derivatives, process for their preparation and fungicidal compositions containing them |
JPH0626884A (ja) | 1992-07-07 | 1994-02-04 | San Tesuto Kk | 位置検出装置 |
ES2120523T3 (es) | 1993-02-25 | 1998-11-01 | Goldschmidt Ag Th | Organopolisiloxano-polieteres y su empleo como agentes de reticulacion estables a la hidrolisis en sistemas acuosos. |
US5466823A (en) | 1993-11-30 | 1995-11-14 | G.D. Searle & Co. | Substituted pyrazolyl benzenesulfonamides |
CA2276945C (en) | 1993-11-30 | 2006-08-01 | G.D. Searle & Co. | Tricyclic-substituted pyrazolyl benzenesulfonamides and pharmaceutical compositions thereof |
DE4434637A1 (de) | 1994-09-28 | 1996-04-04 | Hoechst Schering Agrevo Gmbh | Substituierte Pyridine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide |
JPH11510788A (ja) | 1995-05-24 | 1999-09-21 | ノバルティス アクチェンゲゼルシャフト | ピリジン殺菌剤 |
JPH09208541A (ja) * | 1995-11-29 | 1997-08-12 | Nippon Nohyaku Co Ltd | 新規フェニルアラニン誘導体、その光学活性体、その塩類又は錯化合物及びその用途並びにその使用方法 |
AU7710596A (en) | 1995-11-29 | 1997-06-19 | Nihon Nohyaku Co., Ltd. | Phenylalanine derivatives, optically active substances, salts or coordination compounds thereof, and their use as fungicides |
JP2000509047A (ja) | 1996-04-30 | 2000-07-18 | ヘキスト・アクチエンゲゼルシヤフト | 3―アルコキシピリジン―2―カルボキサミドエステル類、その製法および薬剤としてのその使用 |
JPH1045747A (ja) | 1996-08-06 | 1998-02-17 | Pola Chem Ind Inc | アンチマイシンa系化合物の混合物 |
JPH1053583A (ja) | 1996-08-09 | 1998-02-24 | Mitsubishi Chem Corp | ピラゾール化合物およびこれを有効成分とする殺菌、殺虫、殺ダニ剤 |
GB9622636D0 (en) | 1996-10-30 | 1997-01-08 | Scotia Holdings Plc | Presentation of bioactives |
ATE242962T1 (de) | 1997-03-03 | 2003-07-15 | Rohm & Haas | Pestizide zusammensetzungen |
AU8887898A (en) | 1997-08-29 | 1999-03-22 | Meiji Seika Kaisha Ltd. | Rice blast control agent and wheat scab control agent |
TW491686B (en) | 1997-12-18 | 2002-06-21 | Basf Ag | Fungicidal mixtures based on amide compounds and tetrachloroisophthalonitrile |
US7250389B1 (en) | 1998-02-06 | 2007-07-31 | Meiji Seika Kaisha, Ltd. | Antifungal compound and process for producing the same |
CA2353627C (en) | 1998-11-04 | 2010-10-26 | Keiichi Imamura | Picolinamide derivative and harmful organism control agent comprising said picolinamide derivative as active component |
WO2000076979A1 (de) | 1999-06-09 | 2000-12-21 | Bayer Aktiengesellschaft | Pyridincarboxamide und ihre verwendung als pflanzenschutzmittel |
WO2001005769A2 (en) | 1999-07-20 | 2001-01-25 | Dow Agrosciences Llc | Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
US6355660B1 (en) | 1999-07-20 | 2002-03-12 | Dow Agrosciences Llc | Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
US20020177578A1 (en) | 1999-07-20 | 2002-11-28 | Ricks Michael J. | Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
EP1204643B1 (en) * | 1999-08-20 | 2008-06-04 | Dow AgroSciences LLC | Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
JP2003507474A (ja) | 1999-08-20 | 2003-02-25 | フレッド ハッチンソン キャンサー リサーチ センター | bcl−2ファミリーメンバータンパク質を過剰発現する細胞においてアポトーシスを調節するための組成物および方法 |
US20050239873A1 (en) | 1999-08-20 | 2005-10-27 | Fred Hutchinson Cancer Research Center | 2 Methoxy antimycin a derivatives and methods of use |
FR2803592A1 (fr) * | 2000-01-06 | 2001-07-13 | Aventis Cropscience Sa | Nouveaux derives de l'acide 3-hydroxypicolinique, leur procede de preparation et compositions fongicides les contenant. |
US7241804B1 (en) | 2000-08-18 | 2007-07-10 | Fred Hutchinson Cancer Research Center | Compositions and methods for modulating apoptosis in cells over-expressing Bcl-2 family member proteins |
US20020119979A1 (en) | 2000-10-17 | 2002-08-29 | Degenhardt Charles Raymond | Acyclic compounds and methods for treating multidrug resistance |
EP1275653A1 (en) | 2001-07-10 | 2003-01-15 | Bayer CropScience S.A. | Oxazolopyridines and their use as fungicides |
FR2827286A1 (fr) | 2001-07-11 | 2003-01-17 | Aventis Cropscience Sa | Nouveaux composes fongicides |
KR20040018538A (ko) | 2001-07-31 | 2004-03-03 | 다우 아그로사이언시즈 엘엘씨 | Uk-2a의 엑소사이클릭 에스테르 또는 이의 유도체의환원성 분해 및 이로부터 형성된 생성물 |
AU2002341989A1 (en) | 2001-10-05 | 2003-04-22 | Dow Agrosciences Llc | Process to produce derivatives from uk-2a derivatives |
AR037328A1 (es) | 2001-10-23 | 2004-11-03 | Dow Agrosciences Llc | Compuesto de [7-bencil-2,6-dioxo-1,5-dioxonan-3-il]-4-metoxipiridin-2-carboxamida, composicion que lo comprende y metodo que lo utiliza |
WO2004105490A1 (de) | 2003-05-28 | 2004-12-09 | Basf Aktiengesellschaft | Fungizide mischungen zur bekämpfung von reispathogenen |
WO2005014569A1 (en) | 2003-07-17 | 2005-02-17 | Akzo Nobel N.V. | 1,2,4,-trioxepanes as precursors for lactones |
DE10347090A1 (de) | 2003-10-10 | 2005-05-04 | Bayer Cropscience Ag | Synergistische fungizide Wirkstoffkombinationen |
JP4781352B2 (ja) | 2004-06-04 | 2011-09-28 | ゼノポート,インコーポレーテッド | レボドパプロドラッグおよびその組成物ならびにその使用 |
GB0419694D0 (en) * | 2004-09-06 | 2004-10-06 | Givaudan Sa | Anti-bacterial compounds |
BRPI0607008A2 (pt) | 2005-02-04 | 2009-08-04 | Mitsui Chemicals Inc | composição para evitar as doenças de planta e método para evitar as doenças |
BRPI0622303B1 (pt) | 2005-04-18 | 2016-03-01 | Basf Se | copolímeros cp na forma de um polímero obtido por polimerização com radical de pelo menos três monômeros m diferentes monoetilenicamente insaturados |
WO2007054835A2 (en) | 2005-06-21 | 2007-05-18 | Cheminova Agro A/S | Synergistic combination of a glyphosate herbicide and a triazole fungicide |
AP2008004381A0 (en) | 2005-08-05 | 2008-04-30 | Basf Se | Fungicidal mixtures comprising substituted 1-methlpyrazol-4-ylcarboxanillides |
US8008231B2 (en) | 2005-10-13 | 2011-08-30 | Momentive Performance Materials Inc. | Extreme environment surfactant compositions comprising hydrolysis resistant organomodified disiloxane surfactants |
US7829592B2 (en) | 2006-12-21 | 2010-11-09 | Xenoport, Inc. | Catechol protected levodopa diester prodrugs, compositions, and methods of use |
WO2008105964A1 (en) | 2007-02-26 | 2008-09-04 | Stepan Company | Adjuvants for agricultural applications |
AU2008303528B2 (en) | 2007-09-26 | 2013-05-23 | Basf Se | Ternary fungicidal compositions comprising boscalid and chlorothalonil |
PE20091928A1 (es) * | 2008-05-29 | 2009-12-31 | Bristol Myers Squibb Co | Tienopirimidinas hidroxisustituidas como antagonistas de receptor-1 de hormona concentradora de melanina no basicos |
EP2296467B1 (en) | 2008-05-30 | 2015-11-04 | Dow AgroSciences LLC | Methods to control qoi-resistant fungal pathogens |
EP2346872B1 (en) * | 2008-10-08 | 2015-11-25 | Bristol-Myers Squibb Company | Azolotriazinone melanin concentrating hormone receptor-1 antagonists |
TWI504598B (zh) | 2009-03-20 | 2015-10-21 | Onyx Therapeutics Inc | 結晶性三肽環氧酮蛋白酶抑制劑 |
US8465562B2 (en) | 2009-04-14 | 2013-06-18 | Indiana University Research And Technology Corporation | Scalable biomass reactor and method |
CN101530104B (zh) | 2009-04-21 | 2013-07-31 | 上虞颖泰精细化工有限公司 | 一种含有磺酰脲类、吡啶类、氰氟草酯的除草剂组合物及其应用 |
UA112284C2 (uk) | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
US9006259B2 (en) | 2009-08-07 | 2015-04-14 | Dow Agrosciences Llc | N1-sulfonyl-5-fluoropyrimidinone derivatives |
US8470840B2 (en) | 2009-09-01 | 2013-06-25 | Dow Agrosciences, Llc. | Synergistic fungicidal compositions containing a 5-fluoropyrimidine derivative for fungal control in cereals |
WO2011037968A1 (en) | 2009-09-22 | 2011-03-31 | Valent U.S.A, Corporation | Metconazole compositions and methods of use |
UA109416C2 (xx) | 2009-10-06 | 2015-08-25 | Стабільні емульсії типу "масло в воді" | |
JP5655080B2 (ja) | 2009-10-07 | 2015-01-14 | ダウ アグロサイエンシィズ エルエルシー | 穀類において真菌を制御するための5−フルオロシトシンを含有する相乗的殺真菌組成物 |
PT3178321T (pt) | 2009-10-07 | 2019-08-01 | Dow Agrosciences Llc | Misturas fungicidas sinérgicas de epoxiconazol para o controlo de fungos em cereais |
CN101723980A (zh) * | 2009-12-04 | 2010-06-09 | 陕西合成药业有限公司 | 用于治疗的三唑衍生物 |
EA022245B1 (ru) | 2009-12-08 | 2015-11-30 | Басф Се | Пестицидные смеси |
BR112012020509B1 (pt) | 2010-02-26 | 2018-01-23 | Nippon Soda Co., Ltd. | Derivado de tetrazoliloxima e fungicida |
PL2563771T3 (pl) | 2010-04-24 | 2016-06-30 | Viamet Pharmaceuticals Nc Inc | Związki inhibitora metaloenzymu |
WO2011159067A2 (en) | 2010-06-18 | 2011-12-22 | Green Cross Corporation | Thiazole derivatives as sglt2 inhibitors and pharmaceutical composition comprising same |
UA111593C2 (uk) | 2010-07-07 | 2016-05-25 | Баєр Інтеллекчуел Проперті Гмбх | Аміди антранілової кислоти у комбінації з фунгіцидами |
US20130130898A1 (en) | 2010-08-03 | 2013-05-23 | Markus Gewehr | Fungicidal Compositions |
HUE039384T2 (hu) | 2010-08-05 | 2018-12-28 | Bayer Cropscience Ag | Protiokonazolt és fluxapiroxádot tartalmazó aktív vegyület-kombinációk kukorica-betegségek kontrollálására |
UA111167C2 (uk) | 2010-08-05 | 2016-04-11 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Пестицидні композиції мезорозмірних частинок з підсиленою дією |
JP2012036143A (ja) | 2010-08-10 | 2012-02-23 | Sumitomo Chemical Co Ltd | 植物病害防除組成物およびその用途 |
JP2014503504A (ja) | 2010-11-24 | 2014-02-13 | ステマージ バイオテクノロジー エスエー | ミトコンドリアの電子伝達系の複合体iiiの活性の阻害剤、及び疾患を治療するためのその使用 |
JP6013032B2 (ja) | 2011-07-08 | 2016-10-25 | 石原産業株式会社 | 殺菌剤組成物及び植物病害の防除方法 |
EA201491386A1 (ru) | 2012-01-20 | 2014-11-28 | Вайамет Фармасьютикалс, Инк. | Соединения, ингибирующие металлоферменты |
TWI568721B (zh) | 2012-02-01 | 2017-02-01 | 杜邦股份有限公司 | 殺真菌之吡唑混合物 |
AU2013259790B2 (en) | 2012-05-07 | 2016-09-08 | Corteva Agriscience Llc | Use of pro-fungicides of UK-2A for control of Black Sigatoka |
RU2014149194A (ru) | 2012-05-07 | 2016-06-27 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Макроциклические пиколинамиды в качестве фунгицидов |
JP6129300B2 (ja) | 2012-05-07 | 2017-05-17 | ダウ アグロサイエンシィズ エルエルシー | 殺真菌剤としての大環状ピコリンアミド |
WO2013169662A2 (en) | 2012-05-07 | 2013-11-14 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
WO2013169658A1 (en) | 2012-05-07 | 2013-11-14 | Dow Agrosciences Llc | Use of pro-fungicides of uk-2a for control of soybean rust |
US8900625B2 (en) | 2012-12-15 | 2014-12-02 | Nexmed Holdings, Inc. | Antimicrobial compounds and methods of use |
CL2015001862A1 (es) | 2012-12-28 | 2015-10-02 | Dow Agrosciences Llc | Derivados de n-(sustitutos)-5-fluoro-4-imino-3-metil-2-oxo-3, 4-dihidropirimidon-1 (2h)-carboxilato |
CN110003118A (zh) | 2012-12-28 | 2019-07-12 | 阿达玛马克西姆股份有限公司 | 制备羧酸酯衍生物的方法 |
EP2945634A4 (en) | 2012-12-28 | 2016-05-25 | Dow Agrosciences Llc | N- (SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDIN-1 (2H) -CARBOXAMIDE DERIVATIVES |
EP3689142A1 (en) | 2012-12-28 | 2020-08-05 | Adama Makhteshim Ltd. | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives |
ES2666144T3 (es) | 2012-12-28 | 2018-05-03 | Dow Agrosciences Llc | Mezclas fungicidas sinérgicas para control fúngico en cereales |
US9482661B2 (en) | 2012-12-31 | 2016-11-01 | Dow Agrosciences Llc | Synthesis and use of isotopically labeled macrocyclic compounds |
WO2014105817A1 (en) | 2012-12-31 | 2014-07-03 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
US9750248B2 (en) | 2012-12-31 | 2017-09-05 | Dow Agrosciences Llc | Synergistic fungicidal compositions |
TW201542089A (zh) | 2013-07-10 | 2015-11-16 | Meiji Seika Pharma Co Ltd | 含有吡啶羧酸衍生物而成之協同作用植物病害防治用組成物 |
UA117375C2 (uk) * | 2013-09-04 | 2018-07-25 | Медівір Аб | Інгібітори полімерази hcv |
EP3052490A4 (en) | 2013-10-01 | 2017-06-07 | Dow AgroSciences LLC | Macrocyclic picolinamide compounds with fungicidal activity |
CN105745205A (zh) | 2013-10-01 | 2016-07-06 | 美国陶氏益农公司 | 具有杀真菌活性的大环吡啶酰胺化合物 |
WO2015100184A1 (en) | 2013-12-26 | 2015-07-02 | Dow Agrosciences Llc | Use of macrocyclic picolinamides as fungicides |
US9549555B2 (en) | 2013-12-26 | 2017-01-24 | Dow Agrosciences Llc | Macrocyclic picolinamide compounds with fungicidal activity |
EP3089587B1 (en) | 2013-12-31 | 2019-07-24 | Dow AgroSciences LLC | Synergistic fungicidal mixtures for fungal control in cereals |
US20150322051A1 (en) | 2014-05-06 | 2015-11-12 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
BR112017000169A2 (pt) | 2014-07-08 | 2017-10-31 | Dow Agrosciences Llc | picolinamidas macrocíclicas como fungicidas |
WO2016007525A1 (en) | 2014-07-08 | 2016-01-14 | Dow Agrosciences Llc | Macrocyclic picolinamides as a seed treatment |
WO2016007531A1 (en) | 2014-07-08 | 2016-01-14 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
US20160037774A1 (en) | 2014-08-08 | 2016-02-11 | Dow Agrosciences Llc | Synergistic fungicidal mixtures for fungal control in cereals |
CA2972034A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Picolinamides with fungicidal activity |
BR122019026066B1 (pt) | 2014-12-30 | 2022-01-18 | Dow Agrosciences Llc | Compostos de picolinamida |
HUE060055T2 (hu) | 2014-12-30 | 2023-01-28 | Corteva Agriscience Llc | Gombaölõ készítmények |
CN107105661A (zh) | 2014-12-30 | 2017-08-29 | 美国陶氏益农公司 | 具有杀真菌活性的大环吡啶酰胺化合物 |
WO2016109291A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Use of macrocyclic picolinamides as fungicides |
BR112017013608B8 (pt) | 2014-12-30 | 2022-08-23 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
WO2016109288A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Use of picolinamide compounds with fungicidal activity |
CA2972403A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Picolinamide compounds with fungicidal activity |
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