RU2003128311A - Способ лечения резистентных опухолей с применением аналогов эпотилона - Google Patents

Способ лечения резистентных опухолей с применением аналогов эпотилона Download PDF

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Publication number
RU2003128311A
RU2003128311A RU2003128311/14A RU2003128311A RU2003128311A RU 2003128311 A RU2003128311 A RU 2003128311A RU 2003128311/14 A RU2003128311/14 A RU 2003128311/14A RU 2003128311 A RU2003128311 A RU 2003128311A RU 2003128311 A RU2003128311 A RU 2003128311A
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RU
Russia
Prior art keywords
methyl
dihydroxy
thiazolyl
ethenyl
dione
Prior art date
Application number
RU2003128311/14A
Other languages
English (en)
Russian (ru)
Inventor
Фрэнсис И.Ф. ЛИ (US)
Фрэнсис И.Ф. ЛИ
Original Assignee
Бристол-Маерс Сквибб Компани (Us)
Бристол-Маерс Сквибб Компани
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23028846&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2003128311(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бристол-Маерс Сквибб Компани (Us), Бристол-Маерс Сквибб Компани filed Critical Бристол-Маерс Сквибб Компани (Us)
Publication of RU2003128311A publication Critical patent/RU2003128311A/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
RU2003128311/14A 2001-02-20 2002-02-06 Способ лечения резистентных опухолей с применением аналогов эпотилона RU2003128311A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26983601P 2001-02-20 2001-02-20
US60/269,836 2001-02-20

Publications (1)

Publication Number Publication Date
RU2003128311A true RU2003128311A (ru) 2005-03-10

Family

ID=23028846

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2003128311/14A RU2003128311A (ru) 2001-02-20 2002-02-06 Способ лечения резистентных опухолей с применением аналогов эпотилона

Country Status (18)

Country Link
US (2) US6686380B2 (enExample)
EP (1) EP1385529A4 (enExample)
JP (1) JP2004522774A (enExample)
KR (1) KR20040025895A (enExample)
CN (1) CN1774253A (enExample)
BG (1) BG108075A (enExample)
BR (1) BR0207487A (enExample)
CA (1) CA2438610A1 (enExample)
EE (1) EE200300396A (enExample)
HU (1) HUP0303175A2 (enExample)
IL (1) IL156988A0 (enExample)
IS (1) IS6918A (enExample)
MX (1) MXPA03007394A (enExample)
NO (1) NO20033684L (enExample)
PL (1) PL363362A1 (enExample)
RU (1) RU2003128311A (enExample)
WO (1) WO2002066038A1 (enExample)
ZA (1) ZA200306173B (enExample)

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RU2003126171A (ru) * 2001-01-25 2005-02-27 Бристол-Маерс Сквибб Компани (Us) Парентеральный состав, содержащий аналоги эпотилона
WO2002072085A1 (en) * 2001-03-14 2002-09-19 Bristol-Myers Squibb Company Combination of epothilone analogs and chemotherapeutic agents for the treatment of proliferative diseases
TW200403994A (en) * 2002-04-04 2004-03-16 Bristol Myers Squibb Co Oral administration of EPOTHILONES
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US7649006B2 (en) 2002-08-23 2010-01-19 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US6921769B2 (en) 2002-08-23 2005-07-26 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
WO2004018478A2 (en) * 2002-08-23 2004-03-04 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto, analogues and uses thereof
JP2006504743A (ja) 2002-10-09 2006-02-09 コーザン バイオサイエンシス インコーポレイテッド 治療製剤
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US20050171167A1 (en) * 2003-11-04 2005-08-04 Haby Thomas A. Process and formulation containing epothilones and analogs thereof
US20090004277A1 (en) * 2004-05-18 2009-01-01 Franchini Miriam K Nanoparticle dispersion containing lactam compound
WO2006017761A2 (en) * 2004-08-05 2006-02-16 Emory University Epothilone analogues as therapeutic agents
EP1824458A1 (en) * 2004-11-18 2007-08-29 Bristol-Myers Squibb Company Enteric coated bead comprising epothilone or an epothilone analog, and preparation and administration thereof
BRPI0518286A2 (pt) * 2004-11-18 2008-11-11 Bristol Myers Squibb Co microesfera com revestimento entÉrico contendo ixabepilona e sua preparaÇço
EP1856255A4 (en) 2005-02-11 2010-01-27 Univ Southern California PROCESS FOR EXPRESSING PROTEINS VIA DISULPHIDE BRIDGES
EP2029156A4 (en) * 2006-05-01 2010-07-21 Univ Southern California COMBINATION THERAPY FOR CANCER TREATMENT
US8463852B2 (en) * 2006-10-06 2013-06-11 Oracle International Corporation Groupware portlets for integrating a portal with groupware systems
US8802394B2 (en) 2008-11-13 2014-08-12 Radu O. Minea Method of expressing proteins with disulfide bridges with enhanced yields and activity
CA2799202C (en) 2010-05-18 2016-07-05 Cerulean Pharma Inc. Compositions and methods for treatment of autoimmune and other diseases
BR112022013685A2 (pt) 2020-01-10 2022-09-06 R Pharm Us Operating Llc Composições de ixabepilona

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Also Published As

Publication number Publication date
WO2002066038A1 (en) 2002-08-29
BR0207487A (pt) 2004-08-10
KR20040025895A (ko) 2004-03-26
US20020165258A1 (en) 2002-11-07
USRE41393E1 (en) 2010-06-22
EP1385529A4 (en) 2007-05-09
BG108075A (bg) 2005-04-30
ZA200306173B (en) 2004-11-23
PL363362A1 (en) 2004-11-15
CA2438610A1 (en) 2002-08-29
US6686380B2 (en) 2004-02-03
NO20033684L (no) 2003-10-13
JP2004522774A (ja) 2004-07-29
MXPA03007394A (es) 2003-12-04
EE200300396A (et) 2003-12-15
HUP0303175A2 (hu) 2003-12-29
IL156988A0 (en) 2004-02-08
CN1774253A (zh) 2006-05-17
EP1385529A1 (en) 2004-02-04
NO20033684D0 (no) 2003-08-19
IS6918A (is) 2003-08-18

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Effective date: 20060110