RS53079B - Jedinjenja triazolopiridina koja se koriste kao inhibitori pim kinaze - Google Patents

Jedinjenja triazolopiridina koja se koriste kao inhibitori pim kinaze

Info

Publication number
RS53079B
RS53079B RS20130557A RSP20130557A RS53079B RS 53079 B RS53079 B RS 53079B RS 20130557 A RS20130557 A RS 20130557A RS P20130557 A RSP20130557 A RS P20130557A RS 53079 B RS53079 B RS 53079B
Authority
RS
Serbia
Prior art keywords
pyridin
triazolo
alkyl
yloxy
quinoline
Prior art date
Application number
RS20130557A
Other languages
English (en)
Serbian (sr)
Inventor
Shelley Allen
Laura L. Celeste
Gregg T. Davis
Robert Kirk Delisle
Julie Marie Greschuk
Stefan D. Gross
Erik James Hicken
Leila J. Jackson
Joseph P. Lyssikatos
Nicholas C. Kallan
Fredrik P. Marmsater
Mark C. Munson
Jed Pheneger
Bryson Rast
John E. Robinson
Stephen T. Schlachter
George T. Topalov
Dale A. Wright
Qian Zhao
Original Assignee
Array Biopharma Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc. filed Critical Array Biopharma Inc.
Publication of RS53079B publication Critical patent/RS53079B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Transplantation (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
RS20130557A 2008-08-19 2009-08-18 Jedinjenja triazolopiridina koja se koriste kao inhibitori pim kinaze RS53079B (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8995208P 2008-08-19 2008-08-19
US17527709P 2009-05-04 2009-05-04
PCT/US2009/054193 WO2010022076A1 (en) 2008-08-19 2009-08-18 Triazolopyridine compounds as pim kinase inhibitors

Publications (1)

Publication Number Publication Date
RS53079B true RS53079B (sr) 2014-06-30

Family

ID=41227138

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20130557A RS53079B (sr) 2008-08-19 2009-08-18 Jedinjenja triazolopiridina koja se koriste kao inhibitori pim kinaze

Country Status (17)

Country Link
US (1) US8575145B2 (enExample)
EP (1) EP2334677B1 (enExample)
JP (2) JP5518072B2 (enExample)
CN (1) CN102186851B (enExample)
AR (1) AR073079A1 (enExample)
CA (1) CA2734831C (enExample)
DK (1) DK2334677T3 (enExample)
ES (1) ES2439501T3 (enExample)
HR (1) HRP20131140T1 (enExample)
PL (1) PL2334677T3 (enExample)
PT (1) PT2334677E (enExample)
RS (1) RS53079B (enExample)
SI (1) SI2334677T1 (enExample)
SM (1) SMT201400154B (enExample)
TW (1) TWI496779B (enExample)
UY (1) UY32057A (enExample)
WO (1) WO2010022076A1 (enExample)

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Publication number Publication date
CN102186851A (zh) 2011-09-14
PL2334677T3 (pl) 2014-03-31
SMT201400154B (it) 2015-01-15
US8575145B2 (en) 2013-11-05
EP2334677B1 (en) 2013-10-09
DK2334677T3 (da) 2013-11-18
US20110144085A1 (en) 2011-06-16
HRP20131140T1 (hr) 2014-01-03
ES2439501T3 (es) 2014-01-23
UY32057A (es) 2011-01-31
SI2334677T1 (sl) 2013-12-31
EP2334677A1 (en) 2011-06-22
AR073079A1 (es) 2010-10-13
TWI496779B (zh) 2015-08-21
PT2334677E (pt) 2013-11-26
JP2014129409A (ja) 2014-07-10
CA2734831C (en) 2017-04-18
CA2734831A1 (en) 2010-02-25
TW201008940A (en) 2010-03-01
CN102186851B (zh) 2013-06-12
WO2010022076A1 (en) 2010-02-25
JP2012500277A (ja) 2012-01-05
JP5518072B2 (ja) 2014-06-11

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