DK2334677T3 - Triazolpyridinforbindelser som PIM-kinasehæmmere - Google Patents

Triazolpyridinforbindelser som PIM-kinasehæmmere

Info

Publication number
DK2334677T3
DK2334677T3 DK09791625.8T DK09791625T DK2334677T3 DK 2334677 T3 DK2334677 T3 DK 2334677T3 DK 09791625 T DK09791625 T DK 09791625T DK 2334677 T3 DK2334677 T3 DK 2334677T3
Authority
DK
Denmark
Prior art keywords
kinase inhibitors
pyridine compounds
pim kinase
triazole pyridine
triazole
Prior art date
Application number
DK09791625.8T
Other languages
Danish (da)
English (en)
Inventor
Shelley Allen
Laura L Celeste
Gregg T Davis
Robert Kirk Delisle
Julie Marie Greschuk
Stefan D Gross
Erik James Hicken
Leila J Jackson
Joseph P Lyssikatos
Nicholas C Kallan
Fredrik P Marmsater
Mark C Munson
Jed Pheneger
Bryson Rast
John E Robinson
Stephen T Schlachter
George T Topalov
Dale A Wright
Qian Zhao
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Application granted granted Critical
Publication of DK2334677T3 publication Critical patent/DK2334677T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK09791625.8T 2008-08-19 2009-08-18 Triazolpyridinforbindelser som PIM-kinasehæmmere DK2334677T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8995208P 2008-08-19 2008-08-19
US17527709P 2009-05-04 2009-05-04
PCT/US2009/054193 WO2010022076A1 (en) 2008-08-19 2009-08-18 Triazolopyridine compounds as pim kinase inhibitors

Publications (1)

Publication Number Publication Date
DK2334677T3 true DK2334677T3 (da) 2013-11-18

Family

ID=41227138

Family Applications (1)

Application Number Title Priority Date Filing Date
DK09791625.8T DK2334677T3 (da) 2008-08-19 2009-08-18 Triazolpyridinforbindelser som PIM-kinasehæmmere

Country Status (17)

Country Link
US (1) US8575145B2 (enExample)
EP (1) EP2334677B1 (enExample)
JP (2) JP5518072B2 (enExample)
CN (1) CN102186851B (enExample)
AR (1) AR073079A1 (enExample)
CA (1) CA2734831C (enExample)
DK (1) DK2334677T3 (enExample)
ES (1) ES2439501T3 (enExample)
HR (1) HRP20131140T1 (enExample)
PL (1) PL2334677T3 (enExample)
PT (1) PT2334677E (enExample)
RS (1) RS53079B (enExample)
SI (1) SI2334677T1 (enExample)
SM (1) SMT201400154B (enExample)
TW (1) TWI496779B (enExample)
UY (1) UY32057A (enExample)
WO (1) WO2010022076A1 (enExample)

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Publication number Publication date
EP2334677B1 (en) 2013-10-09
WO2010022076A1 (en) 2010-02-25
CN102186851B (zh) 2013-06-12
TW201008940A (en) 2010-03-01
US20110144085A1 (en) 2011-06-16
JP2012500277A (ja) 2012-01-05
PL2334677T3 (pl) 2014-03-31
SI2334677T1 (sl) 2013-12-31
EP2334677A1 (en) 2011-06-22
CN102186851A (zh) 2011-09-14
HRP20131140T1 (hr) 2014-01-03
CA2734831A1 (en) 2010-02-25
ES2439501T3 (es) 2014-01-23
PT2334677E (pt) 2013-11-26
JP2014129409A (ja) 2014-07-10
SMT201400154B (it) 2015-01-15
TWI496779B (zh) 2015-08-21
JP5518072B2 (ja) 2014-06-11
CA2734831C (en) 2017-04-18
RS53079B (sr) 2014-06-30
AR073079A1 (es) 2010-10-13
US8575145B2 (en) 2013-11-05
UY32057A (es) 2011-01-31

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