PT93241A - Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem - Google Patents

Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem

Info

Publication number
PT93241A
PT93241A PT93241A PT9324190A PT93241A PT 93241 A PT93241 A PT 93241A PT 93241 A PT93241 A PT 93241A PT 9324190 A PT9324190 A PT 9324190A PT 93241 A PT93241 A PT 93241A
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
preparation process
compositions containing
piperidine derivatives
piperidine
Prior art date
Application number
PT93241A
Other languages
English (en)
Other versions
PT93241B (pt
Inventor
Per Sauerberg
Preben H Olesen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK82589A external-priority patent/DK82589A/da
Priority claimed from DK231589A external-priority patent/DK231589D0/da
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of PT93241A publication Critical patent/PT93241A/pt
Publication of PT93241B publication Critical patent/PT93241B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PT93241A 1989-02-22 1990-02-22 Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem PT93241B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK82589A DK82589A (da) 1989-02-22 1989-02-22 Piperidinforbindelser, deres fremstilling og anvendelse
DK231589A DK231589D0 (da) 1989-05-12 1989-05-12 Piperidinforbindelser og deres fremstilling og anvendelse

Publications (2)

Publication Number Publication Date
PT93241A true PT93241A (pt) 1990-08-31
PT93241B PT93241B (pt) 1996-01-31

Family

ID=26064725

Family Applications (2)

Application Number Title Priority Date Filing Date
PT93242A PT93242A (pt) 1989-02-22 1990-02-22 Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem
PT93241A PT93241B (pt) 1989-02-22 1990-02-22 Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PT93242A PT93242A (pt) 1989-02-22 1990-02-22 Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem

Country Status (22)

Country Link
US (5) US5043345A (pt)
EP (2) EP0384285A3 (pt)
JP (2) JPH02255680A (pt)
KR (1) KR0163763B1 (pt)
CN (1) CN1028105C (pt)
AR (1) AR247565A1 (pt)
AT (1) ATE123030T1 (pt)
AU (2) AU629302B2 (pt)
CA (2) CA2010579A1 (pt)
DE (1) DE69019550T2 (pt)
DK (1) DK0384288T3 (pt)
ES (1) ES2072323T3 (pt)
FI (2) FI95704C (pt)
GR (1) GR3017062T3 (pt)
HU (2) HU221623B1 (pt)
IE (1) IE69672B1 (pt)
IL (2) IL93352A (pt)
NO (2) NO179639C (pt)
NZ (1) NZ232615A (pt)
PH (1) PH26465A (pt)
PT (2) PT93242A (pt)
RU (1) RU2042676C1 (pt)

Families Citing this family (94)

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US5264444A (en) * 1989-02-22 1993-11-23 Novo Nordisk A/S Piperidine compounds and use
US5043345A (en) * 1989-02-22 1991-08-27 Novo Nordisk A/S Piperidine compounds and their preparation and use
US5260311A (en) * 1989-02-22 1993-11-09 Novo Nordisk A/S Piperidine compounds and their use
US5328925A (en) * 1989-02-22 1994-07-12 Novo Nordisk A/S Piperidine compounds and their use
EP0459568A3 (en) * 1990-05-31 1992-09-30 Merck Sharp & Dohme Ltd. Substituted oxadiazoles and thiadiazoles for use in the treatment of glaucoma and novel compounds having such use
DK198490D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5418240A (en) * 1990-08-21 1995-05-23 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
USRE35822E (en) * 1990-08-21 1998-06-09 Novo Nordisk A/S Heterocyclic compounds
US5527813A (en) * 1990-08-21 1996-06-18 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
DK198390D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5376668A (en) * 1990-08-21 1994-12-27 Novo Nordisk A/S Heterocyclic compounds
DK198590D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
ATE164519T1 (de) * 1990-11-29 1998-04-15 Allergan Inc Verwendung von pyridine derivate zur behandlung der okulären hypertomie
EP0492903A1 (en) * 1990-12-21 1992-07-01 MERCK SHARP & DOHME LTD. Substituted pyrazines, pyrimidines and pyridazines for use in the treatment of glaucoma
IE922270A1 (en) * 1991-07-26 1993-01-27 Akzo Nv Pyrazole derivatives
US5641791A (en) * 1991-08-13 1997-06-24 Novo Nordisk A.S Heterocyclic compounds and their preparation and use
US5175166A (en) * 1991-08-27 1992-12-29 The University Of Toledo Muscarinic agonists
WO1993014089A1 (en) * 1992-01-13 1993-07-22 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
US5244906A (en) * 1992-01-23 1993-09-14 Dowelanco Insect control with substituted oxadiazole and thiadiazole compounds
DE69325662T2 (de) * 1992-10-23 2000-02-10 Merck Sharp & Dohme Ltd., Hoddesdon Dopamin rezeptor subtyp liganden
CA2164296C (en) * 1993-06-04 2007-01-23 Linda Marie Osborne Heterocyclic chemistry
KR100360575B1 (ko) * 1993-08-19 2003-03-10 노보 노르디스크 에이/에스 정신분열증및정신분열형질환치료용약제학적조성물
US5753683A (en) * 1993-08-19 1998-05-19 Novo Nordisk A/S Antipsychotic method
US5545638A (en) * 1993-12-21 1996-08-13 Novo Nordisk A/S Method of treating gastrointestinal motility disorders
IL112024A (en) * 1993-12-21 1999-07-14 Novo Nordisk As Pharmaceutical compositions comprising tetrahydropyridine derivatives substituted with oxadiazole or thiadiazole for treating gastrointestinal motility disorders
US5605908A (en) * 1994-10-24 1997-02-25 Eli Lilly And Company Heterocyclic compounds and their use
US5998404A (en) * 1994-10-24 1999-12-07 Eli Lilly And Company Heterocyclic compounds and their use
US5646289A (en) * 1994-10-24 1997-07-08 Eli Lilly And Company Heterocyclic compounds and their preparation and use
US5574028A (en) * 1994-10-31 1996-11-12 Eli Lilly And Company Method for treating anxiety
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AU4139096A (en) * 1994-10-31 1996-05-23 Eli Lilly And Company Method for treating anxiety
US5726193A (en) * 1994-10-31 1998-03-10 Eli Lilly And Company Method for treating anxiety
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US5565475A (en) * 1994-11-08 1996-10-15 Muhlhauser; Mark A. Method of treating urinary bladder dysfunctions with 3-tetrahydropyridine derivatives
US5612351A (en) * 1994-11-08 1997-03-18 Novo Nordisk A/S Method of treating urinary bladder dysfunctions
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US5605701A (en) * 1995-02-17 1997-02-25 Eli Lilly And Company Transdermal formulation
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NZ219646A (en) * 1986-03-27 1990-10-26 Merck Sharp & Dohme Oxadiazole derivatives of azacyclics for treating cns disorders
IL83275A (en) * 1986-09-08 1994-02-27 Novo Nordisk As Substituted 1, 2, 4- oxadiazolyl piperidine compounds, their preparation and pharmaceutical compositions containing them
US5017618A (en) * 1987-03-16 1991-05-21 University Of Florida Labile derivatives of ketone analogs of 3-substituted-1-alkylamino-2-propanols and their use as beta-adrenergic blockers
GB8714789D0 (en) * 1987-06-24 1987-07-29 Lundbeck & Co As H Heterocyclic compounds
NZ225999A (en) * 1987-09-10 1992-04-28 Merck Sharp & Dohme Azacyclic- or azabicyclic-substituted thiadiazole derivatives and pharmaceutical compositions
IL88156A (en) * 1987-11-13 1997-02-18 Novo Nordisk As Azacyclic compounds their preparation and pharmaceutical compositions containing them
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions
DK162892C (da) * 1988-07-04 1992-05-11 Novo Nordisk As 1,2,5,6-tetrahydropyridinforbindelser, deres fremstilling og farmaceutiske praeparater indeholdende disse
US5328925A (en) * 1989-02-22 1994-07-12 Novo Nordisk A/S Piperidine compounds and their use
US5264444A (en) * 1989-02-22 1993-11-23 Novo Nordisk A/S Piperidine compounds and use
US5260311A (en) * 1989-02-22 1993-11-09 Novo Nordisk A/S Piperidine compounds and their use
US5043345A (en) * 1989-02-22 1991-08-27 Novo Nordisk A/S Piperidine compounds and their preparation and use
DK198390D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
DK198490D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
US5175166A (en) * 1991-08-27 1992-12-29 The University Of Toledo Muscarinic agonists

Also Published As

Publication number Publication date
PH26465A (en) 1992-07-27
RU2042676C1 (ru) 1995-08-27
NO900831L (no) 1990-08-23
FI900887A0 (fi) 1990-02-22
US5284859A (en) 1994-02-08
FI900886A0 (fi) 1990-02-22
HUT58326A (en) 1992-02-28
US5043345A (en) 1991-08-27
HU900884D0 (en) 1990-05-28
JPH02255679A (ja) 1990-10-16
ATE123030T1 (de) 1995-06-15
IL93423A0 (en) 1990-11-29
DE69019550T2 (de) 1995-10-05
EP0384288A2 (en) 1990-08-29
US5041455A (en) 1991-08-20
JP2921578B2 (ja) 1999-07-19
CA2010578A1 (en) 1990-08-22
FI95704B (fi) 1995-11-30
IE900504L (en) 1990-08-22
HU211705A9 (en) 1995-12-28
KR910015569A (ko) 1991-09-30
DK0384288T3 (da) 1995-10-02
EP0384285A3 (en) 1991-04-24
KR0163763B1 (ko) 1998-12-01
JPH02255680A (ja) 1990-10-16
FI95704C (fi) 1996-03-11
AU4999690A (en) 1990-08-30
GR3017062T3 (en) 1995-11-30
CN1028105C (zh) 1995-04-05
US5712297A (en) 1998-01-27
ES2072323T3 (es) 1995-07-16
AR247565A1 (es) 1995-01-31
AU629302B2 (en) 1992-10-01
US5559138A (en) 1996-09-24
EP0384288A3 (en) 1991-04-10
NO900831D0 (no) 1990-02-21
CA2010578C (en) 2000-05-23
AU4999790A (en) 1990-08-30
PT93242A (pt) 1990-08-31
HU221623B1 (hu) 2002-12-28
DE69019550D1 (de) 1995-06-29
FI900887A7 (fi) 1990-08-23
IL93352A (en) 1994-08-26
NO900830D0 (no) 1990-02-21
EP0384285A2 (en) 1990-08-29
NZ232615A (en) 1992-06-25
NO900830L (no) 1990-08-23
IE69672B1 (en) 1996-10-02
CA2010579A1 (en) 1990-08-22
PT93241B (pt) 1996-01-31
CN1045104A (zh) 1990-09-05
IL93352A0 (en) 1990-11-29
NO179639B (no) 1996-08-12
EP0384288B1 (en) 1995-05-24
NO179639C (no) 1996-11-20

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