PT84794B - Processo de preparacao de derivados de benzimidazois substituido e de composicoes farmaceuticas que os contem - Google Patents

Processo de preparacao de derivados de benzimidazois substituido e de composicoes farmaceuticas que os contem

Info

Publication number
PT84794B
PT84794B PT84794A PT8479487A PT84794B PT 84794 B PT84794 B PT 84794B PT 84794 A PT84794 A PT 84794A PT 8479487 A PT8479487 A PT 8479487A PT 84794 B PT84794 B PT 84794B
Authority
PT
Portugal
Prior art keywords
benzimidazoes
substituted
pharmaceutical compositions
compositions containing
preparing derivatives
Prior art date
Application number
PT84794A
Other languages
English (en)
Other versions
PT84794A (en
Inventor
Robert John Ife
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Publication of PT84794A publication Critical patent/PT84794A/pt
Publication of PT84794B publication Critical patent/PT84794B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/73Unsubstituted amino or imino radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT84794A 1986-04-30 1987-04-29 Processo de preparacao de derivados de benzimidazois substituido e de composicoes farmaceuticas que os contem PT84794B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868610607A GB8610607D0 (en) 1986-04-30 1986-04-30 Chemical compounds

Publications (2)

Publication Number Publication Date
PT84794A PT84794A (en) 1987-05-01
PT84794B true PT84794B (pt) 1989-12-29

Family

ID=10597134

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84794A PT84794B (pt) 1986-04-30 1987-04-29 Processo de preparacao de derivados de benzimidazois substituido e de composicoes farmaceuticas que os contem

Country Status (7)

Country Link
EP (1) EP0246774A1 (pt)
JP (1) JPS62263177A (pt)
AU (1) AU7216287A (pt)
DK (1) DK210487A (pt)
GB (1) GB8610607D0 (pt)
PT (1) PT84794B (pt)
ZA (1) ZA873074B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62201884A (ja) * 1986-02-28 1987-09-05 Tokyo Tanabe Co Ltd ベンズイミダゾール誘導体及びその製造法
DE3722810A1 (de) * 1987-07-10 1989-01-19 Hoechst Ag Substituierte benzimidazole, verfahren zu deren herstellung, diese enthaltende pharmazeutische zubereitungen und deren verwendung
JP2536173B2 (ja) * 1988-08-18 1996-09-18 武田薬品工業株式会社 注射剤
SE8804628D0 (sv) * 1988-12-22 1988-12-22 Ab Haessle New compounds
AU2923595A (en) * 1994-06-23 1996-01-19 Byk Gulden Lomberg Chemische Fabrik Gmbh 4-s- and n-substituted 6-alkylpyridines for controlling helicobacter bacteria
EP0983263A1 (en) * 1997-05-30 2000-03-08 Dr. Reddy's Research Foundation Novel benzimidazole derivatives as antiulcer agents, process for their preparation and pharmaceutical compositions containing them
JP4127740B2 (ja) * 1998-04-20 2008-07-30 エーザイ・アール・アンド・ディー・マネジメント株式会社 安定化したベンズイミダゾール系化合物含有組成物
US6852739B1 (en) 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
AU2003254282A1 (en) 2002-08-01 2004-02-23 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
JP2011515369A (ja) * 2008-03-19 2011-05-19 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト 殺菌剤ヒドロキシモイル−テトラゾール誘導体

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0178438A1 (en) * 1984-09-19 1986-04-23 Beecham Group Plc Novel compounds
JO1406B1 (en) * 1984-11-02 1986-11-30 سميث كلاين اند فرينش لابوراتوريز ليمتد Chemical compounds

Also Published As

Publication number Publication date
AU7216287A (en) 1987-11-05
DK210487D0 (da) 1987-04-24
EP0246774A1 (en) 1987-11-25
JPS62263177A (ja) 1987-11-16
ZA873074B (en) 1987-11-25
PT84794A (en) 1987-05-01
GB8610607D0 (en) 1986-06-04
DK210487A (da) 1987-10-31

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