PT89792A - Processo de preparacao de derivados da quinolina substituidos e de composicoes farmaceuticas que os contem - Google Patents

Processo de preparacao de derivados da quinolina substituidos e de composicoes farmaceuticas que os contem

Info

Publication number
PT89792A
PT89792A PT89792A PT8979289A PT89792A PT 89792 A PT89792 A PT 89792A PT 89792 A PT89792 A PT 89792A PT 8979289 A PT8979289 A PT 8979289A PT 89792 A PT89792 A PT 89792A
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
compositions containing
quinoline derivatives
substituted quinoline
preparing substituted
Prior art date
Application number
PT89792A
Other languages
English (en)
Other versions
PT89792B (pt
Inventor
Thomas Henry Brown
Robert John Ife
Colin Andrew Leach
Original Assignee
Smithkline Beckman Intercredit
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Intercredit filed Critical Smithkline Beckman Intercredit
Publication of PT89792A publication Critical patent/PT89792A/pt
Publication of PT89792B publication Critical patent/PT89792B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT89792A 1988-02-25 1989-02-22 Processo de preparacao de derivados da quinolina substituidos e de composicoes farmaceuticas que os contem PT89792B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888804447A GB8804447D0 (en) 1988-02-25 1988-02-25 Compounds

Publications (2)

Publication Number Publication Date
PT89792A true PT89792A (pt) 1989-10-04
PT89792B PT89792B (pt) 1994-05-31

Family

ID=10632379

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89792A PT89792B (pt) 1988-02-25 1989-02-22 Processo de preparacao de derivados da quinolina substituidos e de composicoes farmaceuticas que os contem

Country Status (8)

Country Link
US (1) US5006535A (pt)
EP (1) EP0336544A1 (pt)
JP (1) JPH01261388A (pt)
AU (1) AU3011589A (pt)
DK (1) DK82189A (pt)
GB (1) GB8804447D0 (pt)
PT (1) PT89792B (pt)
ZA (1) ZA891442B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2011086A1 (en) * 1989-03-17 1990-09-17 Karl-Heinz Geiss 2-alkyl-4-arylmethylaminoquinolines, the use thereof and drugs prepared therefrom
US4916135A (en) * 1989-05-08 1990-04-10 Hoechst Roussel Pharmaceuticals Inc. N-heteroaryl-4-quinolinamines
GB8918265D0 (en) * 1989-08-10 1989-09-20 Smithkline Beckman Intercredit Compounds
US5493027A (en) * 1993-01-22 1996-02-20 Board Of Regents, The University Of Texas System Anticonvulsive agents and uses thereof
IS4164A (is) * 1993-06-11 1994-12-12 Ab Astra Efnasambönd sem hindra flæði magasýru
US5556863A (en) * 1993-06-11 1996-09-17 Astra Aktiebolag Compound for gastric acid secretion inhibition
US6576644B2 (en) 2000-09-06 2003-06-10 Bristol-Myers Squibb Co. Quinoline inhibitors of cGMP phosphodiesterase
CN1304374C (zh) * 2002-04-30 2007-03-14 永进药品工业株式会社 可用做caspase-3抑制剂的喹啉衍生物及其制备方法和药用组合物
SE0400284D0 (sv) * 2004-02-10 2004-02-10 Astrazeneca Ab Novel compounds
AU2011235069B2 (en) 2010-04-02 2016-03-17 Senomyx, Inc. Sweet flavor modifier
CN103764630B (zh) 2011-08-12 2017-08-08 赛诺米克斯公司 甜味调节剂
WO2016073251A1 (en) 2014-11-07 2016-05-12 Senomyx, Inc. Substituted 4-amino-5-(cyclohexyloxy)quinoline-3-carboxylic acids as sweet flavor modifiers

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2652398A (en) * 1949-11-17 1953-09-15 Endo Products Inc N-substituted-2-amino (methyl) quinolines
US3470186A (en) * 1967-06-02 1969-09-30 American Cyanamid Co Substituted 4-anilino-3-quinolinecarboxylic acids and esters
CA942748A (en) * 1970-09-18 1974-02-26 Venkatachala L. Narayanan 1-aziridinylcarbonyl substituted-3-quinolinecarboxylic acid compounds
US3755332A (en) * 1971-07-01 1973-08-28 Ciba Geigy Corp Substituted 4 indazolaminoquinolines
US4343804A (en) * 1979-03-26 1982-08-10 A. H. Robins Company, Inc. 4-Amino-3-quinolinecarboxylic acids and esters-antisecretory anti-ulcer compounds
GB8621425D0 (en) * 1986-09-05 1986-10-15 Smith Kline French Lab Compounds

Also Published As

Publication number Publication date
JPH01261388A (ja) 1989-10-18
PT89792B (pt) 1994-05-31
ZA891442B (en) 1990-06-27
GB8804447D0 (en) 1988-03-23
US5006535A (en) 1991-04-09
DK82189D0 (da) 1989-02-22
EP0336544A1 (en) 1989-10-11
AU3011589A (en) 1989-08-31
DK82189A (da) 1989-08-26

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19931105

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19950531