PT88370A - Processo para a preparacao de derivados da pirimidina fundidos triciclicos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados da pirimidina fundidos triciclicos e de composicoes farmaceuticas que os contem

Info

Publication number
PT88370A
PT88370A PT88370A PT8837088A PT88370A PT 88370 A PT88370 A PT 88370A PT 88370 A PT88370 A PT 88370A PT 8837088 A PT8837088 A PT 8837088A PT 88370 A PT88370 A PT 88370A
Authority
PT
Portugal
Prior art keywords
tricylic
tricycle
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT88370A
Other languages
English (en)
Inventor
Takehiko Nara
Taketoshi Saijo
Hiroshi Satoh
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of PT88370A publication Critical patent/PT88370A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT88370A 1987-08-31 1988-08-30 Processo para a preparacao de derivados da pirimidina fundidos triciclicos e de composicoes farmaceuticas que os contem PT88370A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP21896487 1987-08-31
JP13096988 1988-05-27

Publications (1)

Publication Number Publication Date
PT88370A true PT88370A (pt) 1989-06-30

Family

ID=26465940

Family Applications (1)

Application Number Title Priority Date Filing Date
PT88370A PT88370A (pt) 1987-08-31 1988-08-30 Processo para a preparacao de derivados da pirimidina fundidos triciclicos e de composicoes farmaceuticas que os contem

Country Status (10)

Country Link
US (1) US4912104A (pt)
EP (1) EP0306185A1 (pt)
JP (1) JP2750869B2 (pt)
KR (1) KR890003766A (pt)
CN (1) CN1031843A (pt)
DK (1) DK480588A (pt)
FI (1) FI883986A (pt)
HU (1) HUT50477A (pt)
NO (1) NO167028C (pt)
PT (1) PT88370A (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3116230B2 (ja) * 1989-02-15 2000-12-11 武田薬品工業株式会社 三環式縮合ピリミジン誘導体
US5543147A (en) * 1993-01-20 1996-08-06 Nikolai B. Leonidov Crystalline modification of 2,4-dioxo-6-methyl-1,2,3,4-tetrahydropyrimidine, a method for the preparation thereof and a medicinal preparation based on it
US9255099B2 (en) 2006-06-06 2016-02-09 Intra-Cellular Therapies, Inc. Pyrazolo[3,4-D]pyrimidine-4,6(5H,7H)-diones as phosphodiesterase 1 inhibitors
EP2240028B1 (en) 2007-12-06 2016-07-20 Intra-Cellular Therapies, Inc. Pyrazolopyrimidine-4,6-dione derivatives and their use as pharmaceutical
EA201170773A1 (ru) 2008-12-06 2012-01-30 Интра-Селлулар Терапиз, Инк. Органические соединения
SG171777A1 (en) * 2008-12-06 2011-07-28 Intra Cellular Therapies Inc Organic compounds
AU2009322899A1 (en) 2008-12-06 2010-06-10 Intra-Cellular Therapies, Inc. Organic compounds
JP5894148B2 (ja) 2010-05-31 2016-03-23 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 有機化合物
US9434730B2 (en) 2010-05-31 2016-09-06 Intra-Cellular Therapies, Inc. PDE1 inhibitor compounds
US9546175B2 (en) 2014-08-07 2017-01-17 Intra-Cellular Therapies, Inc. Organic compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1086707B (de) * 1959-02-04 1960-08-11 Chemische Werke Radebeul Veb Verfahren zur Herstellung von basischen Theophyllinderivaten und ihren quaternaeren Salzen
US3637684A (en) * 1968-01-05 1972-01-25 Pfizer Preparation of heterocycloimidazoles
DE2058501A1 (de) * 1970-11-27 1972-05-31 Bayer Ag Verfahren zur Herstellung von neuen N-verbrueckten bicyclischen Heteroaromaten
FR2303551A1 (fr) * 1975-03-12 1976-10-08 Brun Lab Sa Le Derives de la 8-amino theophylline, leur procede de preparation et leurs applications
JPS6032638B2 (ja) * 1976-09-01 1985-07-29 武田薬品工業株式会社 3−アミノピラゾロ〔3,4−d〕ピリミジン誘導体
DE2843195A1 (de) * 1978-10-04 1980-04-17 Chinoin Gyogyszer Es Vegyeszet Verfahren zur herstellung neuer kondensierter purinderivate
DE3370961D1 (en) * 1982-10-25 1987-05-21 Schering Corp Substituted 9h-8-oxo-pyrimido(2,1-f)purine-2,4-diones, process for their production and pharmaceutical compositions containing them
US4603203A (en) * 1983-12-14 1986-07-29 Takeda Chemical Industries, Ltd. 3-aminopyrazolo[3,4-d]pyrimidine derivatives and production thereof

Also Published As

Publication number Publication date
FI883986A0 (fi) 1988-08-30
FI883986A (fi) 1989-03-01
DK480588A (da) 1989-03-01
DK480588D0 (da) 1988-08-29
EP0306185A1 (en) 1989-03-08
NO167028C (no) 1991-09-25
US4912104A (en) 1990-03-27
NO883860L (no) 1989-03-01
CN1031843A (zh) 1989-03-22
JP2750869B2 (ja) 1998-05-13
NO167028B (no) 1991-06-17
KR890003766A (ko) 1989-04-18
HUT50477A (en) 1990-02-28
JPH0249784A (ja) 1990-02-20
NO883860D0 (no) 1988-08-30

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