FI95704B - Menetelmä uusien terapeuttisesti käyttökelpoisten pyridiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten pyridiinijohdannaisten valmistamiseksi

Info

Publication number
FI95704B
FI95704B FI900886A FI900886A FI95704B FI 95704 B FI95704 B FI 95704B FI 900886 A FI900886 A FI 900886A FI 900886 A FI900886 A FI 900886A FI 95704 B FI95704 B FI 95704B
Authority
FI
Finland
Prior art keywords
preparation
therapeutically useful
pyridine derivatives
novel therapeutically
useful pyridine
Prior art date
Application number
FI900886A
Other languages
English (en)
Swedish (sv)
Other versions
FI900886A0 (fi
FI95704C (fi
Inventor
Per Sauerberg
Preben H Olesen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK82589A external-priority patent/DK82589A/da
Priority claimed from DK231589A external-priority patent/DK231589D0/da
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of FI900886A0 publication Critical patent/FI900886A0/fi
Application granted granted Critical
Publication of FI95704B publication Critical patent/FI95704B/fi
Publication of FI95704C publication Critical patent/FI95704C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
FI900886A 1989-02-22 1990-02-22 Menetelmä uusien terapeuttisesti käyttökelpoisten pyridiinijohdannaisten valmistamiseksi FI95704C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DK82589A DK82589A (da) 1989-02-22 1989-02-22 Piperidinforbindelser, deres fremstilling og anvendelse
DK82589 1989-02-22
DK231589A DK231589D0 (da) 1989-05-12 1989-05-12 Piperidinforbindelser og deres fremstilling og anvendelse
DK231589 1989-05-12

Publications (3)

Publication Number Publication Date
FI900886A0 FI900886A0 (fi) 1990-02-22
FI95704B true FI95704B (fi) 1995-11-30
FI95704C FI95704C (fi) 1996-03-11

Family

ID=26064725

Family Applications (2)

Application Number Title Priority Date Filing Date
FI900886A FI95704C (fi) 1989-02-22 1990-02-22 Menetelmä uusien terapeuttisesti käyttökelpoisten pyridiinijohdannaisten valmistamiseksi
FI900887A FI900887A0 (fi) 1989-02-22 1990-02-22 Piperidinfoereningar samt framstaellning och anvaendning av dessa.

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI900887A FI900887A0 (fi) 1989-02-22 1990-02-22 Piperidinfoereningar samt framstaellning och anvaendning av dessa.

Country Status (22)

Country Link
US (5) US5043345A (fi)
EP (2) EP0384285A3 (fi)
JP (2) JPH02255680A (fi)
KR (1) KR0163763B1 (fi)
CN (1) CN1028105C (fi)
AR (1) AR247565A1 (fi)
AT (1) ATE123030T1 (fi)
AU (2) AU629302B2 (fi)
CA (2) CA2010578C (fi)
DE (1) DE69019550T2 (fi)
DK (1) DK0384288T3 (fi)
ES (1) ES2072323T3 (fi)
FI (2) FI95704C (fi)
GR (1) GR3017062T3 (fi)
HU (2) HU221623B1 (fi)
IE (1) IE69672B1 (fi)
IL (2) IL93352A (fi)
NO (2) NO900831L (fi)
NZ (1) NZ232615A (fi)
PH (1) PH26465A (fi)
PT (2) PT93241B (fi)
RU (1) RU2042676C1 (fi)

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US5264444A (en) * 1989-02-22 1993-11-23 Novo Nordisk A/S Piperidine compounds and use
US5043345A (en) * 1989-02-22 1991-08-27 Novo Nordisk A/S Piperidine compounds and their preparation and use
EP0459568A3 (en) * 1990-05-31 1992-09-30 Merck Sharp & Dohme Ltd. Substituted oxadiazoles and thiadiazoles for use in the treatment of glaucoma and novel compounds having such use
DK198490D0 (da) * 1990-08-21 1990-08-21 Novo Nordisk As Heterocykliske forbindelser, deres fremstilling og anvendelse
USRE35822E (en) * 1990-08-21 1998-06-09 Novo Nordisk A/S Heterocyclic compounds
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US5376668A (en) * 1990-08-21 1994-12-27 Novo Nordisk A/S Heterocyclic compounds
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US5418240A (en) * 1990-08-21 1995-05-23 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
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IE922270A1 (en) * 1991-07-26 1993-01-27 Akzo Nv Pyrazole derivatives
US5641791A (en) * 1991-08-13 1997-06-24 Novo Nordisk A.S Heterocyclic compounds and their preparation and use
US5175166A (en) * 1991-08-27 1992-12-29 The University Of Toledo Muscarinic agonists
WO1993014089A1 (en) * 1992-01-13 1993-07-22 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
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US5545638A (en) * 1993-12-21 1996-08-13 Novo Nordisk A/S Method of treating gastrointestinal motility disorders
IL112024A (en) * 1993-12-21 1999-07-14 Novo Nordisk As Pharmaceutical compositions comprising tetrahydropyridine derivatives substituted with oxadiazole or thiadiazole for treating gastrointestinal motility disorders
US5665745A (en) * 1994-10-24 1997-09-09 Eli Lilly And Company Heterocyclic compounds and their preparation and use
US5998404A (en) * 1994-10-24 1999-12-07 Eli Lilly And Company Heterocyclic compounds and their use
US5605908A (en) * 1994-10-24 1997-02-25 Eli Lilly And Company Heterocyclic compounds and their use
US5488056A (en) * 1994-10-31 1996-01-30 Eli Lilly And Company Method for treating anxiety
EP0709094B1 (en) * 1994-10-31 2000-04-05 Eli Lilly And Company Tetrahydropyridine oxadiazole or thiadiazole compound for treating anxiety
US5484794A (en) * 1994-11-09 1996-01-16 Eli Lilly And Company Method for treating anxiety
US5574028A (en) * 1994-10-31 1996-11-12 Eli Lilly And Company Method for treating anxiety
US5726193A (en) * 1994-10-31 1998-03-10 Eli Lilly And Company Method for treating anxiety
US5565475A (en) * 1994-11-08 1996-10-15 Muhlhauser; Mark A. Method of treating urinary bladder dysfunctions with 3-tetrahydropyridine derivatives
US5612351A (en) * 1994-11-08 1997-03-18 Novo Nordisk A/S Method of treating urinary bladder dysfunctions
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US5605701A (en) * 1995-02-17 1997-02-25 Eli Lilly And Company Transdermal formulation
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WO1997020819A1 (en) * 1995-12-06 1997-06-12 Eli Lilly And Company Composition for treating pain
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GB9603755D0 (en) * 1996-02-22 1996-04-24 Pfizer Ltd Therapeutic agents
EP0912183A4 (en) * 1996-04-23 1999-08-04 Lilly Co Eli HETEROCYCLIC COMPOSITIONS
AU2991397A (en) * 1996-04-23 1997-11-12 Eli Lilly And Company Heterocyclic compounds
WO1997040045A1 (en) * 1996-04-24 1997-10-30 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
EP0821959A3 (en) * 1996-08-01 1998-09-16 Eli Lilly And Company Use of 3-(4-hexyloxy-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyridine for treating nicotine withdrawal
US6090829A (en) * 1996-08-01 2000-07-18 Eli Lilly And Company Method for treating excessive aggression
EP0821957A3 (en) * 1996-08-01 1998-04-22 Eli Lilly And Company Use of 3-(4-hexyloxy-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyridine (xanomeline) for treating substance abuse
US6043258A (en) * 1996-08-01 2000-03-28 Eli Lilly And Company Method for treating disruptive behavior disorders with xanomeline
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Also Published As

Publication number Publication date
CA2010578A1 (en) 1990-08-22
AU629302B2 (en) 1992-10-01
EP0384288B1 (en) 1995-05-24
NZ232615A (en) 1992-06-25
AU4999790A (en) 1990-08-30
CN1028105C (zh) 1995-04-05
IE900504L (en) 1990-08-22
IL93423A0 (en) 1990-11-29
NO179639C (no) 1996-11-20
NO900831L (no) 1990-08-23
FI900886A0 (fi) 1990-02-22
CA2010579A1 (en) 1990-08-22
HU221623B1 (hu) 2002-12-28
US5712297A (en) 1998-01-27
IL93352A (en) 1994-08-26
HU211705A9 (en) 1995-12-28
EP0384285A3 (en) 1991-04-24
EP0384288A3 (en) 1991-04-10
PH26465A (en) 1992-07-27
CN1045104A (zh) 1990-09-05
NO900830L (no) 1990-08-23
HU900884D0 (en) 1990-05-28
PT93241A (pt) 1990-08-31
AR247565A1 (es) 1995-01-31
PT93241B (pt) 1996-01-31
IL93352A0 (en) 1990-11-29
JP2921578B2 (ja) 1999-07-19
IE69672B1 (en) 1996-10-02
US5041455A (en) 1991-08-20
KR0163763B1 (ko) 1998-12-01
AU4999690A (en) 1990-08-30
US5284859A (en) 1994-02-08
US5559138A (en) 1996-09-24
JPH02255680A (ja) 1990-10-16
DE69019550D1 (de) 1995-06-29
DE69019550T2 (de) 1995-10-05
EP0384288A2 (en) 1990-08-29
EP0384285A2 (en) 1990-08-29
ES2072323T3 (es) 1995-07-16
FI95704C (fi) 1996-03-11
CA2010578C (en) 2000-05-23
DK0384288T3 (da) 1995-10-02
HUT58326A (en) 1992-02-28
NO900831D0 (no) 1990-02-21
FI900887A0 (fi) 1990-02-22
JPH02255679A (ja) 1990-10-16
PT93242A (pt) 1990-08-31
US5043345A (en) 1991-08-27
KR910015569A (ko) 1991-09-30
ATE123030T1 (de) 1995-06-15
GR3017062T3 (en) 1995-11-30
NO900830D0 (no) 1990-02-21
NO179639B (no) 1996-08-12
RU2042676C1 (ru) 1995-08-27

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