FI93119B - Uusien tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä - Google Patents

Uusien tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä

Info

Publication number
FI93119B
FI93119B FI902355A FI902355A FI93119B FI 93119 B FI93119 B FI 93119B FI 902355 A FI902355 A FI 902355A FI 902355 A FI902355 A FI 902355A FI 93119 B FI93119 B FI 93119B
Authority
FI
Finland
Prior art keywords
diethepines
triazolo
preparation
novel thieno
thieno
Prior art date
Application number
FI902355A
Other languages
English (en)
Swedish (sv)
Other versions
FI902355A0 (fi
FI93119C (fi
Inventor
Pierre Braquet
Andr Esanu
Jean-Pierre Laurent
Jacques Pommier
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of FI902355A0 publication Critical patent/FI902355A0/fi
Publication of FI93119B publication Critical patent/FI93119B/fi
Application granted granted Critical
Publication of FI93119C publication Critical patent/FI93119C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/22Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI902355A 1989-05-13 1990-05-11 Uusien tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä FI93119C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8911030 1989-05-13
GB898911030A GB8911030D0 (en) 1989-05-13 1989-05-13 Hetrazepine derivatives

Publications (3)

Publication Number Publication Date
FI902355A0 FI902355A0 (fi) 1990-05-11
FI93119B true FI93119B (fi) 1994-11-15
FI93119C FI93119C (fi) 1995-02-27

Family

ID=10656702

Family Applications (1)

Application Number Title Priority Date Filing Date
FI902355A FI93119C (fi) 1989-05-13 1990-05-11 Uusien tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä

Country Status (32)

Country Link
US (1) US5049559A (fi)
JP (1) JPH06104668B2 (fi)
KR (1) KR900018113A (fi)
AR (1) AR245725A1 (fi)
AT (1) AT399153B (fi)
AU (1) AU628171B2 (fi)
BE (1) BE1004122A3 (fi)
CA (1) CA2016551C (fi)
CH (1) CH681009A5 (fi)
DE (1) DE4015137C2 (fi)
DK (1) DK102990A (fi)
DZ (1) DZ1414A1 (fi)
ES (1) ES2019840A6 (fi)
FI (1) FI93119C (fi)
FR (2) FR2646774B1 (fi)
GB (2) GB8911030D0 (fi)
GR (1) GR1000295B (fi)
HK (1) HK94992A (fi)
IE (1) IE65246B1 (fi)
IN (1) IN174000B (fi)
IT (1) IT1240935B (fi)
LU (1) LU87733A1 (fi)
MA (1) MA21842A1 (fi)
NL (1) NL9001089A (fi)
NO (1) NO173607C (fi)
NZ (1) NZ233574A (fi)
OA (1) OA09209A (fi)
PT (1) PT94008B (fi)
SE (1) SE505407C2 (fi)
SG (1) SG91992G (fi)
TN (1) TNSN90061A1 (fi)
ZA (1) ZA903305B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5304553A (en) * 1988-10-31 1994-04-19 Eisai Co., Ltd. 1,4-diazepine derivative and its pharmaceutical use
US5221671A (en) * 1988-10-31 1993-06-22 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
US5382579A (en) * 1988-10-31 1995-01-17 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
US5468740A (en) * 1988-10-31 1995-11-21 Eisai Co., Ltd. 1,4-diazepine derivative and its pharmaceutical use
FI95708C (fi) * 1988-10-31 1996-03-11 Eisai Co Ltd Analogiamenetelmä 1,4-diatsepiinijohdannaisen ja sen farmaseuttisesti sopivan suolan valmistamiseksi
AT394563B (de) * 1990-05-09 1992-05-11 Scras Verfahren zur herstellung von thieno-triazolodiazepinderivaten
GB9207645D0 (en) * 1992-04-08 1992-05-27 Smithkline Beecham Corp Methods
ES2061406B1 (es) * 1993-05-07 1995-06-01 Uriach & Cia Sa J Nuevos derivados de la 2-(quinolina) con actividad farmacologica.
US6262044B1 (en) 1998-03-12 2001-07-17 Novo Nordisk A/S Modulators of protein tyrosine phosphatases (PTPASES)
US6987105B2 (en) * 2000-04-28 2006-01-17 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Synthesis and use of thienotriazolodiazepines
EA009646B1 (ru) 2003-05-30 2008-02-28 Рэнбакси Лабораториз Лтд. Замещённые производные пиррола и их применение в качестве ингибиторов hmg-coa
AU2006313430B2 (en) 2005-11-08 2012-09-06 Ranbaxy Laboratories Limited Process for (3R,5R)-7-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4- [(4-hydroxy methyl phenyl amino) carbonyl]-pyrrol-1-yl]-3, 5-dihydroxy-heptanoic acid hemi calcium salt

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3435973A1 (de) * 1984-10-01 1986-04-10 Boehringer Ingelheim KG, 6507 Ingelheim Diazepine enthaltende pharmazeutische zusammensetzungen mit paf-antagonistischer wirkung
DE3724031A1 (de) * 1986-07-22 1988-01-28 Boehringer Ingelheim Kg Neue hetrazepine und verfahren zu ihrer herstellung
PH30676A (en) * 1986-07-22 1997-09-16 Boehringer Ingelhein Kg Hetrazepine compounds which have useful pharmaceutical utility
WO1988009792A1 (en) * 1987-06-08 1988-12-15 Yoshitomi Pharmaceutical Industries, Ltd. Ester-substituted thienotriazolodiazepine compounds and their medicinal use

Also Published As

Publication number Publication date
SG91992G (en) 1992-12-04
TNSN90061A1 (fr) 1991-03-05
OA09209A (fr) 1992-06-30
CA2016551A1 (en) 1990-11-13
IT9020276A0 (it) 1990-05-11
GR1000295B (el) 1992-05-12
IN174000B (fi) 1994-08-20
SE9001670L (fi)
FI902355A0 (fi) 1990-05-11
GB9010403D0 (en) 1990-06-27
FR2646851A1 (fr) 1990-11-16
GR900100319A (en) 1991-10-10
LU87733A1 (fr) 1990-09-19
IE65246B1 (en) 1995-10-04
JPH06104668B2 (ja) 1994-12-21
AR245725A1 (es) 1994-02-28
FR2646774A1 (fr) 1990-11-16
HK94992A (en) 1992-12-04
DE4015137C2 (de) 2003-06-12
IE901583L (en) 1990-11-13
IT1240935B (it) 1993-12-27
FI93119C (fi) 1995-02-27
NZ233574A (en) 1991-07-26
DZ1414A1 (fr) 2004-09-13
ZA903305B (en) 1991-02-27
NO173607B (no) 1993-09-27
SE9001670D0 (sv) 1990-05-09
CA2016551C (en) 1997-09-09
PT94008B (pt) 1996-12-31
IT9020276A1 (it) 1991-11-11
GB8911030D0 (en) 1989-06-28
FR2646851B1 (fr) 1992-02-14
DK102990A (da) 1990-11-14
US5049559A (en) 1991-09-17
BE1004122A3 (fr) 1992-09-29
GB2231330A (en) 1990-11-14
NO901813L (no) 1990-11-14
ES2019840A6 (es) 1991-07-01
MA21842A1 (fr) 1990-12-31
NL9001089A (nl) 1990-12-03
AT399153B (de) 1995-03-27
DE4015137A1 (de) 1990-11-15
KR900018113A (ko) 1990-12-20
SE505407C2 (sv) 1997-08-25
PT94008A (pt) 1991-01-08
AU628171B2 (en) 1992-09-10
NO901813D0 (no) 1990-04-24
AU5493190A (en) 1990-11-15
NO173607C (no) 1994-01-05
FR2646774B1 (fr) 1992-02-14
DK102990D0 (da) 1990-04-26
GB2231330B (en) 1992-04-29
JPH035484A (ja) 1991-01-11
CH681009A5 (en) 1992-12-31
ATA95690A (de) 1994-08-15

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Legal Events

Date Code Title Description
BB Publication of examined application
FG Patent granted

Owner name: SOCIETE DE CONSEILS DE RECHERCHES ET D APPLICATION

MA Patent expired