PT84234A - Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines - Google Patents
Anti-histaminic compositions containing n-heterocyclyl-4-piperidinaminesInfo
- Publication number
- PT84234A PT84234A PT84234A PT8423487A PT84234A PT 84234 A PT84234 A PT 84234A PT 84234 A PT84234 A PT 84234A PT 8423487 A PT8423487 A PT 8423487A PT 84234 A PT84234 A PT 84234A
- Authority
- PT
- Portugal
- Prior art keywords
- alkyl
- substd
- alkoxy
- furanyl
- opt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82549186A | 1986-02-03 | 1986-02-03 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT84234A true PT84234A (en) | 1987-03-01 |
| PT84234B PT84234B (pt) | 1989-09-14 |
Family
ID=25244134
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT84234A PT84234B (pt) | 1986-02-03 | 1987-02-02 | Processo para a preparacao de n-heterociclil-4-piperidinaminas e de composicoes farmaceuticas anti-histaminicas que os contem |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP0232937B1 (pt) |
| JP (2) | JPH0794393B2 (pt) |
| CN (1) | CN1018614B (pt) |
| AT (1) | ATE79620T1 (pt) |
| AU (1) | AU583706B2 (pt) |
| CA (1) | CA1327579C (pt) |
| CY (1) | CY1865A (pt) |
| DE (1) | DE3781173T2 (pt) |
| DK (1) | DK173674B1 (pt) |
| EG (1) | EG17993A (pt) |
| ES (1) | ES2052544T3 (pt) |
| FI (1) | FI870448A (pt) |
| GR (1) | GR3006158T3 (pt) |
| HK (1) | HK114695A (pt) |
| HU (1) | HU201067B (pt) |
| IE (1) | IE60885B1 (pt) |
| IL (1) | IL81448A (pt) |
| MA (1) | MA20868A1 (pt) |
| NO (1) | NO870407L (pt) |
| NZ (1) | NZ219165A (pt) |
| PH (1) | PH24738A (pt) |
| PT (1) | PT84234B (pt) |
| TN (1) | TNSN87015A1 (pt) |
| ZA (1) | ZA87744B (pt) |
| ZM (1) | ZM1287A1 (pt) |
| ZW (1) | ZW2087A1 (pt) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ223654A (en) * | 1987-03-09 | 1990-03-27 | Janssen Pharmaceutica Nv | 1-alkyl-substituted-benzimidazole-4-piperidinamines and pharmaceutical compositions |
| US4897401A (en) * | 1987-06-19 | 1990-01-30 | Janssen Pharmaceutical N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases |
| US4988689A (en) * | 1987-07-01 | 1991-01-29 | Janssen Pharmaceutica N.V. | ((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines |
| CA1317939C (en) * | 1987-07-01 | 1993-05-18 | Janssen Pharmaceutica Naamloze Vennootschap | ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines |
| PH30434A (en) * | 1989-04-07 | 1997-05-09 | Janssen Pharmaceutica Nv | Hydroxyalkylfuranyl derivatives |
| IT1229231B (it) * | 1989-05-08 | 1991-07-26 | Dompe Farmaceutici Spa | Aminoimidazopiridine farmacologicamente attive |
| CA2043564A1 (en) * | 1990-07-06 | 1992-01-07 | Alfons G. M. De Knaep | 3-[(5-methyl-2-furanyl)methyl]-n-(4-piperidinyl)-3h-imidazo [4,5-b]-pyridin-2-amine 2-hydroxy-1,2,3-propanetricarboxylate |
| NZ239540A (en) * | 1990-09-24 | 1993-11-25 | Neurosearch As | 1-phenyl benzimidazole derivatives and medicaments |
| AU730229B2 (en) * | 1992-09-03 | 2001-03-01 | Sepracor, Inc. | Use of norastemizole for the treatment of allergic disorders |
| ES2210957T3 (es) * | 1992-09-03 | 2004-07-01 | Sepracor Inc. | Composiciones farmaceuticas que contienen norastemizol. |
| WO1994027973A1 (fr) * | 1993-05-20 | 1994-12-08 | Kissei Pharmaceutical Co., Ltd. | Derive 1-(2-benzimidazolyl)-1,5-diazacyclooctane |
| TW429256B (en) * | 1995-12-27 | 2001-04-11 | Janssen Pharmaceutica Nv | 1-(1,2-disubstituted piperidinyl)-4-(benzimidazolyl- and imidazopyridinyl)-piperidine derivatives |
| EP1035869A1 (en) * | 1997-03-26 | 2000-09-20 | Sepracor, Inc. | Chemically and thermally stable norastemizole formulations |
| US5817823A (en) * | 1997-04-17 | 1998-10-06 | Sepracor Inc. | Method for synthesizing 2-substituted imidazoles |
| JP2003503403A (ja) | 1999-06-28 | 2003-01-28 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 呼吸合胞体ウイルス複製阻害剤 |
| DE60013836T2 (de) | 1999-06-28 | 2006-01-19 | Janssen Pharmaceutica N.V. | Replikationsinhibitoren des respiratorischen synzytialvirus |
| TR200103806T2 (tr) * | 1999-06-28 | 2002-06-21 | Janssen Pharmaceutica N. V. | Solunum sistemi sinsitiyal virüsünün replikasyonunu inhibe edici maddeler. |
| GB0215293D0 (en) | 2002-07-03 | 2002-08-14 | Rega Foundation | Viral inhibitors |
| US20070021404A1 (en) * | 2003-06-24 | 2007-01-25 | Dan Peters | Novel aza-ring derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| ATE544765T1 (de) | 2003-12-22 | 2012-02-15 | Leuven K U Res & Dev | Imidazoä4,5-cüpyridinverbindungen und verfahren zur antiviralen behandlung |
| CA2592388C (en) | 2004-12-21 | 2013-04-02 | Steven S. Bondy | Imidazo[4,5-c]pyridine compound and method of antiviral treatment |
| US8193359B2 (en) | 2004-12-24 | 2012-06-05 | Prosidion Limited | G-protein coupled receptor agonists |
| ES2350647T3 (es) | 2005-03-08 | 2011-01-25 | Janssen Pharmaceutica Nv | Derivados de diaza-espiro-[4.4]-nonano como antagonistas de neuroquininas (nk1). |
| ES2339298T3 (es) | 2006-07-07 | 2010-05-18 | Gilead Sciences, Inc. | Compuesto de piridazina novedoso y uso del mismo. |
| UA99466C2 (en) | 2007-07-06 | 2012-08-27 | Гилиад Сайенсиз, Инк. | Crystalline pyridazine compound |
| MX2011003239A (es) * | 2008-09-26 | 2011-04-28 | Merck Sharp & Dohme | Nuevos derivados de bencimidazol ciclicos utiles como agentes anti-diabeticos. |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4219559A (en) | 1979-01-10 | 1980-08-26 | Janssen Pharmaceutica N.V. | N-Heterocyclyl-4-piperidinamines |
| CA1140119A (en) * | 1978-04-03 | 1983-01-25 | Joseph Torremans | N-heterocyclyl-4-piperidinamines |
| US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
| IN156065B (pt) * | 1982-07-12 | 1985-05-04 | Janssen Pharmaceutica Nv | |
| US4634704A (en) * | 1983-10-06 | 1987-01-06 | Janssen Pharmaceutica, N.V. | Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines |
| EP0144101B1 (en) * | 1983-11-30 | 1991-02-06 | Janssen Pharmaceutica N.V. | Bicyclic heterocyclyl containing n-(bicyclic heterocyclyl)-4-piperidinamines |
| US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
| PH23995A (en) * | 1984-01-09 | 1990-02-09 | Janssen Pharmaceutica Nv | 4((bicycle heterocyclyl)-methyl and hetero)piperidines |
| JPS60174778A (ja) * | 1984-01-09 | 1985-09-09 | ジヤンセン・フア−マシユ−チカ・ナ−ムロ−ゼ・フエンノ−トシヤツプ | Ｎ−ヘテロシクリル−４−ピペリジンアミン |
-
1987
- 1987-01-28 EG EG48/87A patent/EG17993A/xx active
- 1987-01-28 AT AT87200128T patent/ATE79620T1/de not_active IP Right Cessation
- 1987-01-28 EP EP87200128A patent/EP0232937B1/en not_active Expired - Lifetime
- 1987-01-28 CA CA000528342A patent/CA1327579C/en not_active Expired - Lifetime
- 1987-01-28 DE DE8787200128T patent/DE3781173T2/de not_active Expired - Lifetime
- 1987-01-28 ES ES87200128T patent/ES2052544T3/es not_active Expired - Lifetime
- 1987-01-30 PH PH34794A patent/PH24738A/en unknown
- 1987-02-02 ZA ZA87744A patent/ZA87744B/xx unknown
- 1987-02-02 ZM ZM12/87A patent/ZM1287A1/xx unknown
- 1987-02-02 DK DK198700541A patent/DK173674B1/da not_active IP Right Cessation
- 1987-02-02 HU HU87354A patent/HU201067B/hu unknown
- 1987-02-02 NO NO870407A patent/NO870407L/no unknown
- 1987-02-02 MA MA21102A patent/MA20868A1/fr unknown
- 1987-02-02 JP JP62020600A patent/JPH0794393B2/ja not_active Expired - Lifetime
- 1987-02-02 AU AU68218/87A patent/AU583706B2/en not_active Expired
- 1987-02-02 FI FI870448A patent/FI870448A/fi not_active Application Discontinuation
- 1987-02-02 IE IE25887A patent/IE60885B1/en not_active IP Right Cessation
- 1987-02-02 PT PT84234A patent/PT84234B/pt unknown
- 1987-02-02 IL IL81448A patent/IL81448A/xx not_active IP Right Cessation
- 1987-02-02 ZW ZW20/87A patent/ZW2087A1/xx unknown
- 1987-02-03 TN TNTNSN87015A patent/TNSN87015A1/fr unknown
- 1987-02-03 CN CN87100563A patent/CN1018614B/zh not_active Expired
- 1987-02-04 NZ NZ219165A patent/NZ219165A/en unknown
-
1992
- 1992-11-05 GR GR920402478T patent/GR3006158T3/el unknown
-
1994
- 1994-10-03 JP JP6260917A patent/JPH0819126B2/ja not_active Expired - Lifetime
-
1995
- 1995-07-13 HK HK114695A patent/HK114695A/xx not_active IP Right Cessation
-
1996
- 1996-04-05 CY CY186596A patent/CY1865A/xx unknown
Also Published As
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