PT82744B - Processo para a preparacao de novos esteres de acido sulfonico - Google Patents

Processo para a preparacao de novos esteres de acido sulfonico

Info

Publication number
PT82744B
PT82744B PT82744A PT8274486A PT82744B PT 82744 B PT82744 B PT 82744B PT 82744 A PT82744 A PT 82744A PT 8274486 A PT8274486 A PT 8274486A PT 82744 B PT82744 B PT 82744B
Authority
PT
Portugal
Prior art keywords
substituted
preparation
sulfonic acid
acid esters
compounds
Prior art date
Application number
PT82744A
Other languages
English (en)
Other versions
PT82744A (en
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of PT82744A publication Critical patent/PT82744A/pt
Publication of PT82744B publication Critical patent/PT82744B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Neurology (AREA)
  • Genetics & Genomics (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Detergent Compositions (AREA)
PT82744A 1985-06-13 1986-06-11 Processo para a preparacao de novos esteres de acido sulfonico PT82744B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH250185 1985-06-13

Publications (2)

Publication Number Publication Date
PT82744A PT82744A (en) 1986-07-01
PT82744B true PT82744B (pt) 1988-12-15

Family

ID=4235223

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82744A PT82744B (pt) 1985-06-13 1986-06-11 Processo para a preparacao de novos esteres de acido sulfonico

Country Status (18)

Country Link
US (2) US4785089A (pt)
EP (1) EP0206993B1 (pt)
JP (2) JPS61289073A (pt)
KR (1) KR940007529B1 (pt)
AT (1) ATE53014T1 (pt)
CA (1) CA1338089C (pt)
CY (1) CY1710A (pt)
DD (2) DD266097A5 (pt)
DE (1) DE3671439D1 (pt)
DK (2) DK170277B1 (pt)
ES (2) ES8801197A1 (pt)
FI (1) FI86171C (pt)
HK (1) HK63293A (pt)
HU (1) HU203074B (pt)
IE (1) IE58477B1 (pt)
IL (1) IL79077A (pt)
PT (1) PT82744B (pt)
SG (1) SG32393G (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3586445T2 (de) * 1984-06-26 1993-01-14 Merck & Co Inc Kondensierte benzo-laktam-verbindungen und deren pharmazeutische zusammensetzungen.
US4785089A (en) * 1985-06-13 1988-11-15 Ciba-Geigy Corporation Novel sulfonic acid esters and their preparation
US5145864A (en) * 1987-09-15 1992-09-08 Alcoholism And Drug Addiction Research Foundation Reduction of voluntary alcohol consumption by treatment with angiotensin converting enzyme inhibitors
US5110813A (en) * 1987-09-15 1992-05-05 Alcoholism And Drug Addiction Research Foundation Reduction of voluntary alcohol consumption by treatment with angiotensin converting enzyme inhibitors
US5371014A (en) * 1988-02-12 1994-12-06 Daicel Chemical Industries, Ltd. Process for the production of optically active 2-hydroxy acid esters using microbes to reduce the 2-oxo precursor
ES2059817T3 (es) * 1988-06-06 1994-11-16 Ciba Geigy Ag Procedimiento para la preparacion de hidroxiacidos.
JP3915015B2 (ja) 1995-08-22 2007-05-16 味の素株式会社 光学活性２−ヒドロキシ−４−アリール酪酸またはそのエステルの製造方法
AU753021B2 (en) 1998-03-31 2002-10-03 Ciba Specialty Chemicals Holding Inc. Process for the preparation of HPB esters
WO2001079176A1 (en) * 2000-04-18 2001-10-25 Scinopharm Singapore Pte Ltd Process for preparation of 3-[(1'-(alkoxycarbonyl)-3'-phenylpropyl)amino]-2-oxo-[1]-benzazepine and its derivatives
WO2002076375A2 (en) * 2001-03-27 2002-10-03 Ranbaxy Laboratories Limited Process for the preparation of benazepril
EP1291336A3 (en) * 2001-09-05 2003-10-08 Solvias AG Preparation of optically active alpha-hydroxyethers
ITMI20020934A1 (it) * 2002-05-03 2003-11-03 Danimite Dipharma S P A Processo per la sintesi di benazepril cloridrato
AU2003247159A1 (en) * 2003-07-07 2005-01-21 Hetero Drugs Limited A novel process for the preparation of cilazapril
US20090082559A1 (en) * 2005-05-12 2009-03-26 Lupin Limited Process for Crystallization of Benazepril Hydrochloride
CN105061312B (zh) * 2015-07-17 2017-12-12 惠州信立泰药业有限公司 一种改进的盐酸贝那普利的制备方法及含有该盐酸贝那普利的药物组合物

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5535060A (en) * 1978-09-05 1980-03-11 Agency Of Ind Science & Technol Asymmetric hydrogenation of alpha-keto-acid ester
JPS5823861B2 (ja) * 1979-06-05 1983-05-18 工業技術院長 α−ケトエステルの不斉水素化方法
US4344949A (en) * 1980-10-03 1982-08-17 Warner-Lambert Company Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids
US4374847A (en) * 1980-10-27 1983-02-22 Ciba-Geigy Corporation 1-Carboxyalkanoylindoline-2-carboxylic acids
CY1403A (en) * 1981-08-11 1987-12-18 Ciba Geigy Ag Benzazepin-2-ones
US4410520A (en) * 1981-11-09 1983-10-18 Ciba-Geigy Corporation 3-Amino-[1]-benzazepin-2-one-1-alkanoic acids
EP0081320A3 (en) * 1981-12-07 1984-07-18 Beecham Group Plc Preparation of acetic acid derivatives
US4473575A (en) * 1982-07-19 1984-09-25 Ciba-Geigy Corporation 3-Amino-(1)-benzazepin-2-one-1-alkanoic acids
US4470988A (en) * 1983-02-10 1984-09-11 Ciba-Geigy Corporation Benzazocinone and benzazoninone derivatives, and their pharmaceutical use
DE3315464A1 (de) * 1983-04-28 1984-10-31 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von n-alkylierten dipeptiden und deren estern
DE3328986A1 (de) * 1983-08-11 1985-02-21 Degussa Ag, 6000 Frankfurt Verfahren zur praktisch stereospezifischen herstellung von optisch aktiven (alpha)-aminocarbonsaeureestern
US4785089A (en) * 1985-06-13 1988-11-15 Ciba-Geigy Corporation Novel sulfonic acid esters and their preparation

Also Published As

Publication number Publication date
DE3671439D1 (de) 1990-06-28
DK171950B1 (da) 1997-08-25
JPS61289073A (ja) 1986-12-19
PT82744A (en) 1986-07-01
DK276386A (da) 1986-12-14
FI862462A (fi) 1986-12-14
JPH0735358B2 (ja) 1995-04-19
KR940007529B1 (ko) 1994-08-19
US5066801A (en) 1991-11-19
IL79077A0 (en) 1986-09-30
KR870000291A (ko) 1987-02-17
DK276386D0 (da) 1986-06-12
DK39695A (da) 1995-04-07
FI862462A0 (fi) 1986-06-09
ATE53014T1 (de) 1990-06-15
JPH0567140B2 (pt) 1993-09-24
ES8802013A1 (es) 1988-03-16
EP0206993A1 (de) 1986-12-30
CY1710A (en) 1994-01-14
DD266097A5 (de) 1989-03-22
DK170277B1 (da) 1995-07-24
IE58477B1 (en) 1993-09-22
SG32393G (en) 1993-05-21
CA1338089C (en) 1996-02-27
JPH05310656A (ja) 1993-11-22
ES557722A0 (es) 1988-03-16
EP0206993B1 (de) 1990-05-23
DD283611A5 (de) 1990-10-17
ES555954A0 (es) 1987-12-16
ES8801197A1 (es) 1987-12-16
US4785089A (en) 1988-11-15
FI86171B (fi) 1992-04-15
FI86171C (fi) 1992-07-27
HK63293A (en) 1993-07-09
IL79077A (en) 1994-01-25
IE861571L (en) 1986-11-13
HU203074B (en) 1991-05-28

Similar Documents

Publication Publication Date Title
PT82744B (pt) Processo para a preparacao de novos esteres de acido sulfonico
ATE49195T1 (de) Herstellung von fibraten.
PT83388B (pt) Processo para a preparacao de acidos quinolonocarboxilicos substituidos com diazabicicloalquilo com ponte
AR245445A1 (es) Procedimiento para la preparacion de cis-1-aril-2-(fluormetil)oxiranos,compuestos asi obtenidos y preparacion de (treo)-1-aril-2-acilamido-3-fluor-1-propanoles utilizando dichos compuestos.
ES2000604A6 (es) Un procedimiento para preparar aril-piperidin esteres
ATE47138T1 (de) Verfahren zur herstellung von 1,2-dithiolan-3pentans|ure (thioctsaeure).
PT1246812E (pt) Metodo para a preparacao de citalopram
SE8601646D0 (sv) Intermediates for the production of epipodophyllotoxin and related compounds and processes for the preparation and use thereof
DK141786A (da) Fremgangsmaade til fremstilling af et mellemprodukt til brug ved fremstilling af 1-beta-methylcarbapenemantibiotika
ATE82291T1 (de) Clavamderivate, herstellung und zwischenprodukte.
ES2060375T3 (es) Un procedimiento para descomponer acidos peroxicarboxilicos.
DE3686049D1 (de) Verfahren zur herstellung chiraler glycinderivate.
ES497136A0 (es) Procedimiento para la sintesis de esteres de la n-(4'hidro- xifenil) acetamida con acidos 5-benzoil-1-metilpirrol-2-ace-tico
ATE8883T1 (de) Verfahren zur herstellung von nbenzylsubstituierten imiden.
FI956247A0 (fi) Uusia menetelmiä (S)-4-amino-hepta-5,6-dieenihappo ja sen välituotteiden valmistamiseksi
PT80798B (pt) Processo para a preparacao de derivados do acido apovincaminico substituidos nas posicoes 9 ou 11
DE69023246D1 (de) Verfahren zur herstellung von optisch aktiven oder racemischen cyclopropancarbonsäurechloriden.
ATE32719T1 (de) Neues nortropinderivat, verfahren zu seiner herstellung und seine verwendung.
ES8704447A1 (es) Un procedimiento para preparar el homero s de un 3-eter de 2-hidroxi -profil-amina.
ES8307254A1 (es) Un procedimiento para la preparacion de un enantiomero de beta-lactama.

Legal Events

Date Code Title Description
PC3A Transfer or assignment

Free format text: 970619 NOVARTIS AG CH