PT3265084T - Formulações farmacêuticas de inibidor de tirosina cinase de bruton - Google Patents

Formulações farmacêuticas de inibidor de tirosina cinase de bruton

Info

Publication number
PT3265084T
PT3265084T PT167594175T PT16759417T PT3265084T PT 3265084 T PT3265084 T PT 3265084T PT 167594175 T PT167594175 T PT 167594175T PT 16759417 T PT16759417 T PT 16759417T PT 3265084 T PT3265084 T PT 3265084T
Authority
PT
Portugal
Prior art keywords
bruton
tyrosine kinase
pharmaceutical formulations
inhibtor
kinase inhibtor
Prior art date
Application number
PT167594175T
Other languages
English (en)
Portuguese (pt)
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56848552&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT3265084(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of PT3265084T publication Critical patent/PT3265084T/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PT167594175T 2015-03-03 2016-03-02 Formulações farmacêuticas de inibidor de tirosina cinase de bruton PT3265084T (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562127717P 2015-03-03 2015-03-03
US201562193518P 2015-07-16 2015-07-16

Publications (1)

Publication Number Publication Date
PT3265084T true PT3265084T (pt) 2024-02-13

Family

ID=56848552

Family Applications (1)

Application Number Title Priority Date Filing Date
PT167594175T PT3265084T (pt) 2015-03-03 2016-03-02 Formulações farmacêuticas de inibidor de tirosina cinase de bruton

Country Status (28)

Country Link
US (9) US9655857B2 (enExample)
EP (2) EP4338738A3 (enExample)
JP (3) JP7149076B2 (enExample)
KR (2) KR20170122220A (enExample)
CN (4) CN121910678A (enExample)
AU (4) AU2016226279B2 (enExample)
BR (2) BR112017018931A2 (enExample)
CA (3) CA2976695C (enExample)
DK (1) DK3265084T3 (enExample)
ES (1) ES2971597T3 (enExample)
FI (1) FI3265084T3 (enExample)
HR (1) HRP20240231T1 (enExample)
HU (1) HUE065703T2 (enExample)
IL (3) IL315294A (enExample)
LT (1) LT3265084T (enExample)
MD (1) MD3265084T2 (enExample)
MX (5) MX394784B (enExample)
NZ (1) NZ734446A (enExample)
PL (1) PL3265084T3 (enExample)
PT (1) PT3265084T (enExample)
RS (1) RS65234B1 (enExample)
RU (1) RU2017133990A (enExample)
SG (2) SG11201707122QA (enExample)
SI (1) SI3265084T1 (enExample)
SM (1) SMT202400074T1 (enExample)
TW (6) TWI810588B (enExample)
WO (1) WO2016141068A1 (enExample)
ZA (1) ZA201907661B (enExample)

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NZ772688A (en) 2010-06-03 2022-09-30 Pharmacyclics Llc The use of inhibitors of bruton’s tyrosine kinase (btk)
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AU2013293087B2 (en) 2012-07-24 2017-08-31 Pharmacyclics Llc Mutations associated with resistance to inhibitors of Bruton's tyrosine kinase (BTK)
CN111265531B (zh) * 2013-10-25 2023-11-10 药品循环有限责任公司 治疗和预防移植物抗宿主病的方法
KR20230104754A9 (ko) * 2013-12-02 2024-11-15 파마싸이클릭스 엘엘씨 동종항체 유도 만성 이식편대숙주병의 치료 및 예방 방법
US9545407B2 (en) * 2014-08-07 2017-01-17 Pharmacyclics Llc Formulations of a bruton's tyrosine kinase inhibitor
IL315294A (en) * 2015-03-03 2024-10-01 Pharmacyclics Llc Pharmaceutical formulations of bruton's tyrosine kinase inhibitor
HK1249014A1 (zh) 2015-03-20 2018-10-26 The Trustees Of The University Of Pennsylvania 具有作为佐剂的cd40配体的疫苗
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CN108472259A (zh) * 2016-01-19 2018-08-31 詹森药业有限公司 包含btk抑制剂的配制品/组合物
JP7590810B2 (ja) 2016-10-06 2024-11-27 ヤンセン ファーマシューティカ エヌ．ベー． Ｂｔｋ阻害剤を調製するための方法および中間体
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US10688050B1 (en) 2018-12-21 2020-06-23 Synthon B.V. Pharmaceutical composition comprising ibrutinib
SG11202109102PA (en) * 2019-02-22 2021-09-29 Janssen Pharmaceutica Nv Pharmaceutical formulations
ES3061133T3 (en) * 2019-08-26 2026-03-31 Arvinas Operations Inc Methods of treating breast cancer with tetrahydronaphthalene derivatives as estrogen receptor degraders
US20210228479A1 (en) * 2020-01-29 2021-07-29 Farmakeio Nutraceuticals Llc Steroidal compositions and method of making and use
SI4243782T1 (sl) * 2020-11-13 2025-11-28 Ptc Therapeutics, Inc. Tableta za uporabo v zdravljenju huntingtonove bolezni in postopek njene izdelave
WO2022260667A1 (en) * 2021-06-10 2022-12-15 Hikma Pharmaceuticals Usa Inc. Oral dosage forms of ibrutinib
US11433072B1 (en) 2021-06-10 2022-09-06 Hikma Pharmaceuticals USA, Inc. Oral dosage forms of ibrutinib
US20250302954A1 (en) 2022-05-11 2025-10-02 Celgene Corporation Methods to overcome drug resistance by re-sensitizing cancer cells to treatment with a prior therapy via treatment with a t cell therapy
KR20260035260A (ko) * 2023-07-07 2026-03-12 아크로테크 바이오파마 인코포레이티드. 말초 t 세포 림프종이 있는 환자의 치료를 위한 프랄라트렉세이트 및 cop 조합물

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