PL377661A1 - Pochodne pirydyno [2,3-d] pirymidyny jako selektywne inhibitory kinaz KDR i FGFR - Google Patents

Pochodne pirydyno [2,3-d] pirymidyny jako selektywne inhibitory kinaz KDR i FGFR

Info

Publication number
PL377661A1
PL377661A1 PL377661A PL37766103A PL377661A1 PL 377661 A1 PL377661 A1 PL 377661A1 PL 377661 A PL377661 A PL 377661A PL 37766103 A PL37766103 A PL 37766103A PL 377661 A1 PL377661 A1 PL 377661A1
Authority
PL
Poland
Prior art keywords
selectiive
pyridino
kdr
pyrimidine derivatives
fgfr inhibitors
Prior art date
Application number
PL377661A
Other languages
English (en)
Polish (pl)
Inventor
Jin-Jun Liu
Kin-Chun Luk
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of PL377661A1 publication Critical patent/PL377661A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL377661A 2002-12-20 2003-12-11 Pochodne pirydyno [2,3-d] pirymidyny jako selektywne inhibitory kinaz KDR i FGFR PL377661A1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43496902P 2002-12-20 2002-12-20
US51361503P 2003-10-23 2003-10-23

Publications (1)

Publication Number Publication Date
PL377661A1 true PL377661A1 (pl) 2006-02-06

Family

ID=32685355

Family Applications (1)

Application Number Title Priority Date Filing Date
PL377661A PL377661A1 (pl) 2002-12-20 2003-12-11 Pochodne pirydyno [2,3-d] pirymidyny jako selektywne inhibitory kinaz KDR i FGFR

Country Status (15)

Country Link
US (1) US7098332B2 (enExample)
EP (1) EP1581531B1 (enExample)
JP (1) JP2006511563A (enExample)
KR (1) KR100763298B1 (enExample)
AR (1) AR042532A1 (enExample)
AT (1) ATE387445T1 (enExample)
AU (1) AU2003294830B2 (enExample)
BR (1) BR0317480A (enExample)
CA (1) CA2508951A1 (enExample)
DE (1) DE60319430T2 (enExample)
ES (1) ES2300639T3 (enExample)
MX (1) MXPA05006437A (enExample)
PL (1) PL377661A1 (enExample)
RU (1) RU2345077C2 (enExample)
WO (1) WO2004056822A1 (enExample)

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Also Published As

Publication number Publication date
EP1581531A1 (en) 2005-10-05
WO2004056822A1 (en) 2004-07-08
JP2006511563A (ja) 2006-04-06
EP1581531B1 (en) 2008-02-27
DE60319430D1 (de) 2008-04-10
ATE387445T1 (de) 2008-03-15
US7098332B2 (en) 2006-08-29
RU2345077C2 (ru) 2009-01-27
AU2003294830B2 (en) 2009-06-11
RU2005122901A (ru) 2006-02-27
BR0317480A (pt) 2005-11-16
DE60319430T2 (de) 2009-02-26
KR100763298B1 (ko) 2007-10-04
ES2300639T3 (es) 2008-06-16
AU2003294830A1 (en) 2004-07-14
MXPA05006437A (es) 2005-08-19
CA2508951A1 (en) 2004-07-08
KR20050088202A (ko) 2005-09-02
US20040122029A1 (en) 2004-06-24
AR042532A1 (es) 2005-06-22

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