PL373532A1 - Pochodne piperydyny - Google Patents

Pochodne piperydyny

Info

Publication number
PL373532A1
PL373532A1 PL03373532A PL37353203A PL373532A1 PL 373532 A1 PL373532 A1 PL 373532A1 PL 03373532 A PL03373532 A PL 03373532A PL 37353203 A PL37353203 A PL 37353203A PL 373532 A1 PL373532 A1 PL 373532A1
Authority
PL
Poland
Prior art keywords
piperidine derivatives
piperidine
derivatives
Prior art date
Application number
PL03373532A
Other languages
English (en)
Other versions
PL211082B1 (pl
Inventor
Giuseppe Alvaro
Fabio Romano Di
Maria Elvira Tranquillini
Simone Spada
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of PL373532A1 publication Critical patent/PL373532A1/pl
Publication of PL211082B1 publication Critical patent/PL211082B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
PL373532A 2002-02-08 2003-02-10 Pochodne piperydyny, ich zastosowanie, zawierająca je kompozycja i sposób ich wytwarzania PL211082B1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0203020.3A GB0203020D0 (en) 2002-02-08 2002-02-08 Chemical compounds

Publications (2)

Publication Number Publication Date
PL373532A1 true PL373532A1 (pl) 2005-09-05
PL211082B1 PL211082B1 (pl) 2012-04-30

Family

ID=9930717

Family Applications (1)

Application Number Title Priority Date Filing Date
PL373532A PL211082B1 (pl) 2002-02-08 2003-02-10 Pochodne piperydyny, ich zastosowanie, zawierająca je kompozycja i sposób ich wytwarzania

Country Status (27)

Country Link
US (3) US7189713B2 (pl)
EP (2) EP1472256B1 (pl)
JP (1) JP4488743B2 (pl)
KR (1) KR101011316B1 (pl)
CN (1) CN1319973C (pl)
AR (1) AR038818A1 (pl)
AT (2) ATE308543T1 (pl)
AU (1) AU2003205753B9 (pl)
BR (1) BRPI0307123B8 (pl)
CA (1) CA2475619C (pl)
CO (1) CO5611152A2 (pl)
DE (2) DE60320865D1 (pl)
DK (1) DK1472256T3 (pl)
ES (2) ES2304660T3 (pl)
GB (1) GB0203020D0 (pl)
HK (1) HK1072251A1 (pl)
IL (2) IL162765A0 (pl)
IS (1) IS2402B (pl)
MX (1) MXPA04006791A (pl)
MY (1) MY130411A (pl)
NO (1) NO329379B1 (pl)
NZ (1) NZ533785A (pl)
PL (1) PL211082B1 (pl)
RU (1) RU2336276C2 (pl)
TW (1) TWI291466B (pl)
WO (1) WO2003066635A1 (pl)
ZA (1) ZA200404842B (pl)

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ES2750662T3 (es) * 2012-10-11 2020-03-26 Nerre Therapeutics Ltd Orvepitant para el tratamiento del prurito crónico
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SI3377064T1 (sl) * 2016-01-08 2019-11-29 Nerre Therapeutics Ltd Orvepitant za zdravljenje kroničnega kašlja
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BR112022018876A2 (pt) 2020-04-03 2022-11-22 Nerre Therapeutics Ltd Antagonista de receptor de nk-1 para tratar uma doença selecionada a partir de sepse, choque séptico, síndrome de desconforto respiratório agudo (ards) ou síndrome de disfunção múltipla dos órgãos
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Also Published As

Publication number Publication date
WO2003066635A1 (en) 2003-08-14
KR101011316B1 (ko) 2011-01-28
RU2004126957A (ru) 2005-04-20
PL211082B1 (pl) 2012-04-30
CA2475619A1 (en) 2003-08-14
MXPA04006791A (es) 2004-12-06
KR20040086354A (ko) 2004-10-08
CA2475619C (en) 2011-04-12
ZA200404842B (en) 2005-09-28
DE60302137D1 (de) 2005-12-08
IL162765A0 (en) 2005-11-20
AU2003205753B9 (en) 2010-03-04
EP1666465A1 (en) 2006-06-07
IS2402B (is) 2008-09-15
EP1666465B1 (en) 2008-05-07
RU2336276C2 (ru) 2008-10-20
US7652012B2 (en) 2010-01-26
TW200400192A (en) 2004-01-01
AU2003205753A1 (en) 2003-09-02
GB0203020D0 (en) 2002-03-27
EP1472256A1 (en) 2004-11-03
NO329379B1 (no) 2010-10-04
MY130411A (en) 2007-06-29
ES2250870T3 (es) 2006-04-16
EP1472256B1 (en) 2005-11-02
US7189713B2 (en) 2007-03-13
DE60302137T2 (de) 2006-07-20
DE60320865D1 (de) 2008-06-19
BR0307123A (pt) 2004-12-07
TWI291466B (en) 2007-12-21
NO20043239D0 (no) 2004-08-02
US20050176715A1 (en) 2005-08-11
HK1072251A1 (en) 2005-08-19
AU2003205753B8 (en) 2010-02-18
IS7382A (is) 2004-08-04
JP2005524637A (ja) 2005-08-18
ES2304660T3 (es) 2008-10-16
JP4488743B2 (ja) 2010-06-23
US20070099914A1 (en) 2007-05-03
NZ533785A (en) 2007-05-31
IL162765A (en) 2012-04-30
BRPI0307123B8 (pt) 2021-05-25
CN1628115A (zh) 2005-06-15
NO20043239L (no) 2004-08-02
AU2003205753B2 (en) 2010-01-07
ATE308543T1 (de) 2005-11-15
ATE394375T1 (de) 2008-05-15
CN1319973C (zh) 2007-06-06
DK1472256T3 (da) 2006-03-20
BRPI0307123B1 (pt) 2018-06-19
AR038818A1 (es) 2005-01-26
US20100152446A1 (en) 2010-06-17
CO5611152A2 (es) 2006-02-28

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