NO20043239D0 - Piperidinderivater - Google Patents

Piperidinderivater

Info

Publication number
NO20043239D0
NO20043239D0 NO20043239A NO20043239A NO20043239D0 NO 20043239 D0 NO20043239 D0 NO 20043239D0 NO 20043239 A NO20043239 A NO 20043239A NO 20043239 A NO20043239 A NO 20043239A NO 20043239 D0 NO20043239 D0 NO 20043239D0
Authority
NO
Norway
Prior art keywords
piperidine
Prior art date
Application number
NO20043239A
Other languages
English (en)
Other versions
NO20043239L (no
NO329379B1 (no
Inventor
Romano Di Fabio
Giuseppe Alvaro
Maria Elvira Tranquillini
Simone Spada
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20043239D0 publication Critical patent/NO20043239D0/no
Publication of NO20043239L publication Critical patent/NO20043239L/no
Publication of NO329379B1 publication Critical patent/NO329379B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Addiction (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20043239A 2002-02-08 2004-08-02 Piperidinderivater samt anvendelse og fremstilling derav og farmasoytisk preparat NO329379B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0203020.3A GB0203020D0 (en) 2002-02-08 2002-02-08 Chemical compounds
PCT/EP2003/001308 WO2003066635A1 (en) 2002-02-08 2003-02-10 Piperidine derivatives

Publications (3)

Publication Number Publication Date
NO20043239D0 true NO20043239D0 (no) 2004-08-02
NO20043239L NO20043239L (no) 2004-08-02
NO329379B1 NO329379B1 (no) 2010-10-04

Family

ID=9930717

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20043239A NO329379B1 (no) 2002-02-08 2004-08-02 Piperidinderivater samt anvendelse og fremstilling derav og farmasoytisk preparat

Country Status (27)

Country Link
US (3) US7189713B2 (no)
EP (2) EP1666465B1 (no)
JP (1) JP4488743B2 (no)
KR (1) KR101011316B1 (no)
CN (1) CN1319973C (no)
AR (1) AR038818A1 (no)
AT (2) ATE394375T1 (no)
AU (1) AU2003205753B9 (no)
BR (1) BRPI0307123B8 (no)
CA (1) CA2475619C (no)
CO (1) CO5611152A2 (no)
DE (2) DE60320865D1 (no)
DK (1) DK1472256T3 (no)
ES (2) ES2250870T3 (no)
GB (1) GB0203020D0 (no)
HK (1) HK1072251A1 (no)
IL (2) IL162765A0 (no)
IS (1) IS2402B (no)
MX (1) MXPA04006791A (no)
MY (1) MY130411A (no)
NO (1) NO329379B1 (no)
NZ (1) NZ533785A (no)
PL (1) PL211082B1 (no)
RU (1) RU2336276C2 (no)
TW (1) TWI291466B (no)
WO (1) WO2003066635A1 (no)
ZA (1) ZA200404842B (no)

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WO2015024203A1 (en) * 2013-08-20 2015-02-26 Leo Pharma A/S Novel neurokinin 1 receptor antagonist compounds ii
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AU2016384267B2 (en) * 2016-01-08 2022-02-03 Nerre Therapeutics Limited Orvepitant for the treatment of chronic cough
IL269875B2 (en) 2017-04-10 2024-06-01 Chase Therapeutics Corp NK1 antagonist combination and a method for the treatment of synucleinopathies
CN111032158A (zh) 2017-06-30 2020-04-17 才思治疗公司 用于治疗抑郁的nk-1拮抗剂组合物和方法
EP4125875A1 (en) 2020-04-03 2023-02-08 NeRRe Therapeutics Limited An nk-1 receptor antagonist for treating a disease selecting from sepsis, septic shock,, acute respiratory distress syndrome (ards) or multiple organ dysfunction syndrome (mods)
BR112022024208A2 (pt) 2020-06-02 2022-12-20 Nerre Therapeutics Ltd Antagonistas do receptor de neurocinina (nk)-1 para uso no tratamento de condições de fibrose pulmonar promovidas por lesão mecânica aos pulmões

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GB0308968D0 (en) 2003-04-17 2003-05-28 Glaxo Group Ltd Medicaments

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EP1666465A1 (en) 2006-06-07
ES2250870T3 (es) 2006-04-16
AU2003205753B9 (en) 2010-03-04
EP1472256B1 (en) 2005-11-02
ATE394375T1 (de) 2008-05-15
TW200400192A (en) 2004-01-01
DE60302137T2 (de) 2006-07-20
IS2402B (is) 2008-09-15
JP4488743B2 (ja) 2010-06-23
CA2475619C (en) 2011-04-12
CA2475619A1 (en) 2003-08-14
IL162765A (en) 2012-04-30
NO20043239L (no) 2004-08-02
CN1628115A (zh) 2005-06-15
RU2336276C2 (ru) 2008-10-20
ATE308543T1 (de) 2005-11-15
AU2003205753B2 (en) 2010-01-07
TWI291466B (en) 2007-12-21
AU2003205753B8 (en) 2010-02-18
DE60302137D1 (de) 2005-12-08
WO2003066635A1 (en) 2003-08-14
CO5611152A2 (es) 2006-02-28
AR038818A1 (es) 2005-01-26
DK1472256T3 (da) 2006-03-20
US7652012B2 (en) 2010-01-26
US20050176715A1 (en) 2005-08-11
JP2005524637A (ja) 2005-08-18
PL373532A1 (en) 2005-09-05
RU2004126957A (ru) 2005-04-20
IS7382A (is) 2004-08-04
PL211082B1 (pl) 2012-04-30
EP1666465B1 (en) 2008-05-07
HK1072251A1 (en) 2005-08-19
US20070099914A1 (en) 2007-05-03
BRPI0307123B1 (pt) 2018-06-19
NZ533785A (en) 2007-05-31
BR0307123A (pt) 2004-12-07
MY130411A (en) 2007-06-29
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US20100152446A1 (en) 2010-06-17
US7189713B2 (en) 2007-03-13
GB0203020D0 (en) 2002-03-27
BRPI0307123B8 (pt) 2021-05-25
KR101011316B1 (ko) 2011-01-28
DE60320865D1 (de) 2008-06-19
EP1472256A1 (en) 2004-11-03
ZA200404842B (en) 2005-09-28
IL162765A0 (en) 2005-11-20
AU2003205753A1 (en) 2003-09-02
CN1319973C (zh) 2007-06-06
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MXPA04006791A (es) 2004-12-06

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