PL354261A1 - Amphiphilic prodrugs - Google Patents

Amphiphilic prodrugs

Info

Publication number
PL354261A1
PL354261A1 PL00354261A PL35426100A PL354261A1 PL 354261 A1 PL354261 A1 PL 354261A1 PL 00354261 A PL00354261 A PL 00354261A PL 35426100 A PL35426100 A PL 35426100A PL 354261 A1 PL354261 A1 PL 354261A1
Authority
PL
Poland
Prior art keywords
amphiphilic prodrugs
amphiphilic
prodrugs
Prior art date
Application number
PL00354261A
Other languages
English (en)
Polish (pl)
Inventor
Nnochiri N.Ekwuribe Nnochiri N. Ekwuribe
Tatyana A.Dyakonov Tatyana A. Dyakonov
Christopher H.Price Christopher H. Price
Original Assignee
Nobex Corporationnobex Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nobex Corporationnobex Corporation filed Critical Nobex Corporationnobex Corporation
Publication of PL354261A1 publication Critical patent/PL354261A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
PL00354261A 1999-09-13 2000-09-07 Amphiphilic prodrugs PL354261A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15364999P 1999-09-13 1999-09-13
US09/474,915 US6713454B1 (en) 1999-09-13 1999-12-31 Prodrugs of etoposide and etoposide analogs

Publications (1)

Publication Number Publication Date
PL354261A1 true PL354261A1 (en) 2003-12-29

Family

ID=26850733

Family Applications (1)

Application Number Title Priority Date Filing Date
PL00354261A PL354261A1 (en) 1999-09-13 2000-09-07 Amphiphilic prodrugs

Country Status (17)

Country Link
US (3) US6713454B1 (US06713454-20040330-C00025.png)
EP (1) EP1212099A2 (US06713454-20040330-C00025.png)
JP (1) JP2003509385A (US06713454-20040330-C00025.png)
KR (1) KR20020059398A (US06713454-20040330-C00025.png)
CN (1) CN1390143A (US06713454-20040330-C00025.png)
AU (1) AU7575600A (US06713454-20040330-C00025.png)
BR (1) BR0013948A (US06713454-20040330-C00025.png)
CA (1) CA2384645A1 (US06713454-20040330-C00025.png)
CZ (1) CZ2002928A3 (US06713454-20040330-C00025.png)
HU (1) HUP0204110A3 (US06713454-20040330-C00025.png)
IL (1) IL148558A0 (US06713454-20040330-C00025.png)
MX (1) MXPA02002712A (US06713454-20040330-C00025.png)
NO (1) NO20021213L (US06713454-20040330-C00025.png)
NZ (1) NZ517681A (US06713454-20040330-C00025.png)
PL (1) PL354261A1 (US06713454-20040330-C00025.png)
RU (1) RU2002109595A (US06713454-20040330-C00025.png)
WO (1) WO2001019406A2 (US06713454-20040330-C00025.png)

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Also Published As

Publication number Publication date
US20040253206A1 (en) 2004-12-16
CA2384645A1 (en) 2001-03-22
MXPA02002712A (es) 2003-10-14
NO20021213L (no) 2002-05-13
NO20021213D0 (no) 2002-03-12
RU2002109595A (ru) 2003-11-27
AU7575600A (en) 2001-04-17
BR0013948A (pt) 2002-05-14
CN1390143A (zh) 2003-01-08
NZ517681A (en) 2004-01-30
EP1212099A2 (en) 2002-06-12
HUP0204110A2 (hu) 2003-04-28
HUP0204110A3 (en) 2003-08-28
CZ2002928A3 (cs) 2002-09-11
KR20020059398A (ko) 2002-07-12
US20040180840A1 (en) 2004-09-16
WO2001019406A2 (en) 2001-03-22
IL148558A0 (en) 2002-09-12
US7119074B2 (en) 2006-10-10
JP2003509385A (ja) 2003-03-11
US6713454B1 (en) 2004-03-30
WO2001019406A3 (en) 2002-01-17

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