PL2519512T3 - Pochodne n1-acylo-5-fluoropirymidynonu - Google Patents

Pochodne n1-acylo-5-fluoropirymidynonu

Info

Publication number
PL2519512T3
PL2519512T3 PL10807171T PL10807171T PL2519512T3 PL 2519512 T3 PL2519512 T3 PL 2519512T3 PL 10807171 T PL10807171 T PL 10807171T PL 10807171 T PL10807171 T PL 10807171T PL 2519512 T3 PL2519512 T3 PL 2519512T3
Authority
PL
Poland
Prior art keywords
acyl
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
PL10807171T
Other languages
English (en)
Polish (pl)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W. John Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2519512(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of PL2519512T3 publication Critical patent/PL2519512T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL10807171T 2009-08-07 2010-08-05 Pochodne n1-acylo-5-fluoropirymidynonu PL2519512T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
EP10807171.3A EP2519512B1 (en) 2009-08-07 2010-08-05 N1-acyl- 5-fluoropyrimidinone derivatives
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
PL2519512T3 true PL2519512T3 (pl) 2019-09-30

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
PL10807171T PL2519512T3 (pl) 2009-08-07 2010-08-05 Pochodne n1-acylo-5-fluoropirymidynonu

Country Status (33)

Country Link
US (1) US8470839B2 (enExample)
EP (1) EP2519512B1 (enExample)
JP (1) JP5748754B2 (enExample)
KR (1) KR101792285B1 (enExample)
CN (1) CN102548981B (enExample)
AU (1) AU2010279402B2 (enExample)
BR (1) BR112012002810B1 (enExample)
CA (1) CA2768510C (enExample)
CL (1) CL2012000316A1 (enExample)
CO (1) CO6491117A2 (enExample)
CR (1) CR20120030A (enExample)
CY (1) CY1122115T1 (enExample)
DK (1) DK2519512T3 (enExample)
EA (1) EA023411B1 (enExample)
EC (1) ECSP12011653A (enExample)
ES (1) ES2728966T3 (enExample)
HN (1) HN2012000269A (enExample)
HR (1) HRP20190919T1 (enExample)
HU (1) HUE045290T2 (enExample)
IL (1) IL217952A (enExample)
IN (1) IN2012DN00539A (enExample)
LT (1) LT2519512T (enExample)
MX (1) MX2012001620A (enExample)
NI (1) NI201200022A (enExample)
NZ (1) NZ597570A (enExample)
PE (1) PE20120688A1 (enExample)
PL (1) PL2519512T3 (enExample)
PT (1) PT2519512T (enExample)
SI (1) SI2519512T1 (enExample)
TR (1) TR201908180T4 (enExample)
UA (1) UA106889C2 (enExample)
WO (1) WO2011017538A1 (enExample)
ZA (1) ZA201200819B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20120691A1 (es) * 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-Substituted-5-fluoro-3,6-dihydro-6-imino-2 (1H) -pyrimidinone derivatives as fungicidal compositions for use in plant protection
CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
JP2016503816A (ja) 2012-12-31 2016-02-08 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての3−アルキル−5−フルオロ−4置換イミノ−3,4−ジヒドロピリミジン−2(1h)−オン誘導体
JP6585057B2 (ja) 2013-12-31 2019-10-02 アダマ・マクテシム・リミテッド 5−フルオロ−4−イミノ−3−(アルキル/置換アルキル)−1−(アリールスルホニル)−3,4−ジヒドロピリミジン−2(1h)−オンおよびそれらの調製方法
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
JP6734267B2 (ja) 2014-09-26 2020-08-05 ザ ケマーズ カンパニー エフシー リミテッド ライアビリティ カンパニー イソシアネート由来のオルガノシラン
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
WO2020095181A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
WO1997002262A1 (en) * 1995-07-05 1997-01-23 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
PL328777A1 (en) * 1996-03-11 1999-02-15 Novartis Ag Pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) * 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) * 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2252594B1 (en) * 2008-01-22 2015-08-19 Dow AgroSciences LLC 4-amino-5-fluoro-pyrimidine derivatives as fungicides
EP2317851B1 (en) 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
USRE46144E1 (en) 2009-01-23 2016-09-13 Purdue Pharmaceutical Products L.P. Hydroxamic acid derivatives
PE20120691A1 (es) * 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona

Also Published As

Publication number Publication date
LT2519512T (lt) 2019-07-25
JP2013501723A (ja) 2013-01-17
CY1122115T1 (el) 2020-11-25
CL2012000316A1 (es) 2014-06-27
CN102548981A (zh) 2012-07-04
PT2519512T (pt) 2019-06-04
TR201908180T4 (tr) 2019-06-21
EP2519512B1 (en) 2019-03-20
PE20120688A1 (es) 2012-06-06
IL217952A0 (en) 2012-03-29
HK1172894A1 (en) 2013-05-03
CR20120030A (es) 2012-03-28
IL217952A (en) 2017-11-30
BR112012002810A2 (pt) 2015-09-15
UA106889C2 (uk) 2014-10-27
ZA201200819B (en) 2013-05-29
BR112012002810B1 (pt) 2018-12-11
EP2519512A4 (en) 2013-01-16
US8470839B2 (en) 2013-06-25
CN102548981B (zh) 2015-05-13
KR101792285B1 (ko) 2017-10-31
WO2011017538A1 (en) 2011-02-10
CO6491117A2 (es) 2012-07-31
KR20120041786A (ko) 2012-05-02
CA2768510C (en) 2018-05-15
CA2768510A1 (en) 2011-02-10
AU2010279402A1 (en) 2012-02-02
IN2012DN00539A (enExample) 2015-06-12
HRP20190919T1 (hr) 2019-09-20
NI201200022A (es) 2012-05-22
NZ597570A (en) 2014-04-30
EA023411B1 (ru) 2016-06-30
MX2012001620A (es) 2012-04-11
AU2010279402B2 (en) 2015-04-16
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
EP2519512A1 (en) 2012-11-07
EA201270253A1 (ru) 2012-07-30
ES2728966T3 (es) 2019-10-29
SI2519512T1 (sl) 2019-09-30
DK2519512T3 (da) 2019-05-27
JP5748754B2 (ja) 2015-07-15
HN2012000269A (es) 2015-04-27
US20110034490A1 (en) 2011-02-10

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