IN2012DN00539A - - Google Patents

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Publication number
IN2012DN00539A
IN2012DN00539A IN539DEN2012A IN2012DN00539A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A IN 539DEN2012 A IN539DEN2012 A IN 539DEN2012A IN 2012DN00539 A IN2012DN00539 A IN 2012DN00539A
Authority
IN
India
Prior art keywords
fluoropyrimidinones
fungicides
acyl
derivatives
compounds
Prior art date
Application number
Inventor
Boebel Timothy
Bryan Kristy
Lorsbach Beth
Martin Timothy
Owen W
Pobanz Mark
Thornburgh Scott
Webster Jeffery
Yao Chenglin
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2012DN00539(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of IN2012DN00539A publication Critical patent/IN2012DN00539A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

This present disclosure is related to filed of N1-acyl-5- fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.
IN539DEN2012 2009-08-07 2010-08-05 IN2012DN00539A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
IN2012DN00539A true IN2012DN00539A (en) 2015-06-12

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
IN539DEN2012 IN2012DN00539A (en) 2009-08-07 2010-08-05

Country Status (34)

Country Link
US (1) US8470839B2 (en)
EP (1) EP2519512B1 (en)
JP (1) JP5748754B2 (en)
KR (1) KR101792285B1 (en)
CN (1) CN102548981B (en)
AU (1) AU2010279402B2 (en)
BR (1) BR112012002810B1 (en)
CA (1) CA2768510C (en)
CL (1) CL2012000316A1 (en)
CO (1) CO6491117A2 (en)
CR (1) CR20120030A (en)
CY (1) CY1122115T1 (en)
DK (1) DK2519512T3 (en)
EA (1) EA023411B1 (en)
EC (1) ECSP12011653A (en)
ES (1) ES2728966T3 (en)
HK (1) HK1172894A1 (en)
HN (1) HN2012000269A (en)
HR (1) HRP20190919T1 (en)
HU (1) HUE045290T2 (en)
IL (1) IL217952A (en)
IN (1) IN2012DN00539A (en)
LT (1) LT2519512T (en)
MX (1) MX2012001620A (en)
NI (1) NI201200022A (en)
NZ (1) NZ597570A (en)
PE (1) PE20120688A1 (en)
PL (1) PL2519512T3 (en)
PT (1) PT2519512T (en)
SI (1) SI2519512T1 (en)
TR (1) TR201908180T4 (en)
UA (1) UA106889C2 (en)
WO (1) WO2011017538A1 (en)
ZA (1) ZA201200819B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012002830B1 (en) * 2009-08-07 2019-05-28 Adama Makhteshim Ltd. Derivatives of n1-sulfonyl-5-fluoropyrimidinone, composition for controlling a fungal pathogen, and method for controlling or preventing fungal attack in a plant
MX354021B (en) 2011-08-17 2018-02-08 Adama Makhteshim Ltd 5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1<i>H</ i>)-ONE DERIVATIVES.
AU2013370493B2 (en) 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
RU2656101C2 (en) * 2012-12-28 2018-05-31 Адама Мактешим Лтд. 1-(substituted benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
EP2945634A4 (en) 2012-12-28 2016-05-25 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxamides derivatives
CA2894553C (en) * 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CR20160345A (en) 2013-12-31 2017-02-21 Adama Makhteshim Ltd SYNERGIC FUNGICIDE MIXTURES AND COMPOSITIONS THAT INCLUDE 5-FLUORO-4-IMINO-3-METIL-1-TOSIL-3,4-DIHYDROPIRIMIDIN-2 (1H) -ONA AND INHIBITOR (S) OF THE STEROL BIOSYNTHESIS FOR PHYSICAL CONTROL
UA122200C2 (en) 2013-12-31 2020-10-12 Адама Махтешім Лтд. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
US10011617B2 (en) 2014-09-26 2018-07-03 The Chemours Company Fc, Llc Isocyanate derived organosilanes
CA3069619A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (en) * 1962-05-01 1966-10-15 Hoffmann La Roche Process for the production of a cytosine derivative
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (en) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (en) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie NOVEL DERIVATIVES OF 2,3,6,7-TETRAHYDRO 5H-THIAZOLO (3,2-A) PYRIMIDINE, THEIR PREPARATION AND THEIR USE AS HERBICIDES
EP0139613A1 (en) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives, their preparation and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (en) 1988-03-09 1994-08-15 Ciba Geigy Ag MEANS OF PROTECTING PLANTS AGAINST DISEASES.
DE3821711A1 (en) 1988-06-28 1990-02-08 Bayer Ag THIAZOLOPYRIMIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A SCHAEDLINGSBEKAEMPFUNGSMITTEL
JP3217191B2 (en) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト Heteroaromatic compounds and plant protective agents containing the same
EP0836602B1 (en) 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
DK0888359T3 (en) * 1996-03-11 2002-08-12 Syngenta Participations Ag Pyrimidin-4-one derivative as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (en) 1998-11-06 2001-04-18 NOVEDOSA PIRIMIDIN-4-ENAMINE AS A FUNGICIDE.
US7914799B2 (en) 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
US20080004253A1 (en) 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562161A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
BRPI0916930A2 (en) 2008-08-01 2015-07-28 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide.
SI2389375T1 (en) 2009-01-23 2015-11-30 Euro-Celtique S.A. Hydroxamic acid derivatives
BR112012002830B1 (en) 2009-08-07 2019-05-28 Adama Makhteshim Ltd. Derivatives of n1-sulfonyl-5-fluoropyrimidinone, composition for controlling a fungal pathogen, and method for controlling or preventing fungal attack in a plant

Also Published As

Publication number Publication date
US20110034490A1 (en) 2011-02-10
SI2519512T1 (en) 2019-09-30
CR20120030A (en) 2012-03-28
CL2012000316A1 (en) 2014-06-27
EP2519512A1 (en) 2012-11-07
EP2519512B1 (en) 2019-03-20
CA2768510C (en) 2018-05-15
NZ597570A (en) 2014-04-30
CA2768510A1 (en) 2011-02-10
HK1172894A1 (en) 2013-05-03
ECSP12011653A (en) 2012-03-30
HUE045290T2 (en) 2019-12-30
JP2013501723A (en) 2013-01-17
EA023411B1 (en) 2016-06-30
AU2010279402B2 (en) 2015-04-16
UA106889C2 (en) 2014-10-27
CN102548981B (en) 2015-05-13
ES2728966T3 (en) 2019-10-29
BR112012002810B1 (en) 2018-12-11
CO6491117A2 (en) 2012-07-31
BR112012002810A2 (en) 2015-09-15
IL217952A (en) 2017-11-30
HN2012000269A (en) 2015-04-27
EP2519512A4 (en) 2013-01-16
DK2519512T3 (en) 2019-05-27
CY1122115T1 (en) 2020-11-25
CN102548981A (en) 2012-07-04
EA201270253A1 (en) 2012-07-30
NI201200022A (en) 2012-05-22
KR101792285B1 (en) 2017-10-31
US8470839B2 (en) 2013-06-25
MX2012001620A (en) 2012-04-11
AU2010279402A1 (en) 2012-02-02
ZA201200819B (en) 2013-05-29
PL2519512T3 (en) 2019-09-30
IL217952A0 (en) 2012-03-29
KR20120041786A (en) 2012-05-02
PE20120688A1 (en) 2012-06-06
WO2011017538A1 (en) 2011-02-10
PT2519512T (en) 2019-06-04
LT2519512T (en) 2019-07-25
JP5748754B2 (en) 2015-07-15
HRP20190919T1 (en) 2019-09-20
TR201908180T4 (en) 2019-06-21

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