MX2012001620A - Derivados de n1-acil-5-fluoropirimidinona. - Google Patents

Derivados de n1-acil-5-fluoropirimidinona.

Info

Publication number
MX2012001620A
MX2012001620A MX2012001620A MX2012001620A MX2012001620A MX 2012001620 A MX2012001620 A MX 2012001620A MX 2012001620 A MX2012001620 A MX 2012001620A MX 2012001620 A MX2012001620 A MX 2012001620A MX 2012001620 A MX2012001620 A MX 2012001620A
Authority
MX
Mexico
Prior art keywords
acyl
derivatives
fluoropyrimidinone
fluoropyrimidinone derivatives
fluoropyrimidinones
Prior art date
Application number
MX2012001620A
Other languages
English (en)
Spanish (es)
Inventor
Timothy Martin
Timothy Boebel
Kristy Bryan
Beth Lorsbach
W Owen
Mark Pobanz
Jeffery Webster
Chenglin Yao
Scott Thornburgh
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2012001620(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of MX2012001620A publication Critical patent/MX2012001620A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2012001620A 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona. MX2012001620A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
MX2012001620A true MX2012001620A (es) 2012-04-11

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012001620A MX2012001620A (es) 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona.

Country Status (33)

Country Link
US (1) US8470839B2 (enExample)
EP (1) EP2519512B1 (enExample)
JP (1) JP5748754B2 (enExample)
KR (1) KR101792285B1 (enExample)
CN (1) CN102548981B (enExample)
AU (1) AU2010279402B2 (enExample)
BR (1) BR112012002810B1 (enExample)
CA (1) CA2768510C (enExample)
CL (1) CL2012000316A1 (enExample)
CO (1) CO6491117A2 (enExample)
CR (1) CR20120030A (enExample)
CY (1) CY1122115T1 (enExample)
DK (1) DK2519512T3 (enExample)
EA (1) EA023411B1 (enExample)
EC (1) ECSP12011653A (enExample)
ES (1) ES2728966T3 (enExample)
HN (1) HN2012000269A (enExample)
HR (1) HRP20190919T1 (enExample)
HU (1) HUE045290T2 (enExample)
IL (1) IL217952A (enExample)
IN (1) IN2012DN00539A (enExample)
LT (1) LT2519512T (enExample)
MX (1) MX2012001620A (enExample)
NI (1) NI201200022A (enExample)
NZ (1) NZ597570A (enExample)
PE (1) PE20120688A1 (enExample)
PL (1) PL2519512T3 (enExample)
PT (1) PT2519512T (enExample)
SI (1) SI2519512T1 (enExample)
TR (1) TR201908180T4 (enExample)
UA (1) UA106889C2 (enExample)
WO (1) WO2011017538A1 (enExample)
ZA (1) ZA201200819B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона
ES2646725T3 (es) * 2011-08-17 2017-12-15 Adama Makhteshim Ltd. Derivados 1-sustituidos de 5-fluoro-3,6-dihidro-6-imino-2(1H)-pirimidinona como agentes fungicidas para uso en protección de plantas
AU2013370490B2 (en) 2012-12-28 2018-05-10 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives
CN110003118A (zh) 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 制备羧酸酯衍生物的方法
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
KR102309245B1 (ko) 2012-12-31 2021-10-06 아다마 마켓심 리미티드 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체
JP6585057B2 (ja) 2013-12-31 2019-10-02 アダマ・マクテシム・リミテッド 5−フルオロ−4−イミノ−3−(アルキル/置換アルキル)−1−(アリールスルホニル)−3,4−ジヒドロピリミジン−2(1h)−オンおよびそれらの調製方法
EA030056B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
KR102430183B1 (ko) 2014-09-26 2022-08-08 더 케무어스 컴퍼니 에프씨, 엘엘씨 아이소시아네이트 유도된 유기실란
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
IL282939B2 (en) 2018-11-05 2024-10-01 Adama Makhteshim Ltd Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and methods of use thereof
BR112022005464A2 (pt) 2019-09-23 2022-08-16 Adama Makhteshim Ltd Processo para a preparação de 5-(flúor-4-imino-3-metil)-1-tosil-3,4-diidropirimidina-(1h)-ona

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
PL324486A1 (en) * 1995-07-05 1998-05-25 Du Pont Fungicidal pyrimidinones
DK0888359T3 (da) * 1996-03-11 2002-08-12 Syngenta Participations Ag Pyrimidin-4-on-derivat som pesticid
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
EP2044086A2 (en) * 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
DK2562166T3 (en) * 2008-01-22 2015-11-23 Dow Agrosciences Llc 5-fluoro-pyrimidine derivatives as fungicides
KR20110042204A (ko) 2008-08-01 2011-04-25 다우 아그로사이언시즈 엘엘씨 살진균제로서의 5-플루오로시토신의 용도
HUE025349T2 (en) 2009-01-23 2016-02-29 Euro Celtique Sa Hydroxamic acid derivatives
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона

Also Published As

Publication number Publication date
SI2519512T1 (sl) 2019-09-30
AU2010279402A1 (en) 2012-02-02
UA106889C2 (uk) 2014-10-27
CA2768510C (en) 2018-05-15
HN2012000269A (es) 2015-04-27
TR201908180T4 (tr) 2019-06-21
NI201200022A (es) 2012-05-22
BR112012002810A2 (pt) 2015-09-15
ZA201200819B (en) 2013-05-29
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
DK2519512T3 (da) 2019-05-27
PT2519512T (pt) 2019-06-04
US8470839B2 (en) 2013-06-25
JP2013501723A (ja) 2013-01-17
US20110034490A1 (en) 2011-02-10
EP2519512A4 (en) 2013-01-16
HK1172894A1 (en) 2013-05-03
KR101792285B1 (ko) 2017-10-31
CY1122115T1 (el) 2020-11-25
IL217952A0 (en) 2012-03-29
WO2011017538A1 (en) 2011-02-10
PE20120688A1 (es) 2012-06-06
BR112012002810B1 (pt) 2018-12-11
CO6491117A2 (es) 2012-07-31
CN102548981B (zh) 2015-05-13
CA2768510A1 (en) 2011-02-10
CN102548981A (zh) 2012-07-04
IN2012DN00539A (enExample) 2015-06-12
EP2519512B1 (en) 2019-03-20
PL2519512T3 (pl) 2019-09-30
EP2519512A1 (en) 2012-11-07
IL217952A (en) 2017-11-30
KR20120041786A (ko) 2012-05-02
HRP20190919T1 (hr) 2019-09-20
EA023411B1 (ru) 2016-06-30
LT2519512T (lt) 2019-07-25
NZ597570A (en) 2014-04-30
AU2010279402B2 (en) 2015-04-16
CL2012000316A1 (es) 2014-06-27
JP5748754B2 (ja) 2015-07-15
ES2728966T3 (es) 2019-10-29
EA201270253A1 (ru) 2012-07-30
CR20120030A (es) 2012-03-28

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