KR101792285B1 - Ｎ1-아실-5-플루오로피리미디논 유도체 - Google Patents

Ｎ1-아실-5-플루오로피리미디논 유도체 Download PDF

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Publication number
KR101792285B1
KR101792285B1 KR1020127005927A KR20127005927A KR101792285B1 KR 101792285 B1 KR101792285 B1 KR 101792285B1 KR 1020127005927 A KR1020127005927 A KR 1020127005927A KR 20127005927 A KR20127005927 A KR 20127005927A KR 101792285 B1 KR101792285 B1 KR 101792285B1
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KR
South Korea
Prior art keywords
compound
compounds
herbicides
insecticides
plant
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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KR1020127005927A
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English (en)
Korean (ko)
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KR20120041786A (ko
Inventor
티모시 뵈벨
크리스티 브라이언
베스 로스바흐
티모시 마틴
더블유 오웬
마크 포반즈
스콧 쏜버그
제프리 웹스터
쳉린 야오
Original Assignee
아다마 마켓심 리미티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101792285(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 아다마 마켓심 리미티드 filed Critical 아다마 마켓심 리미티드
Publication of KR20120041786A publication Critical patent/KR20120041786A/ko
Application granted granted Critical
Publication of KR101792285B1 publication Critical patent/KR101792285B1/ko
Expired - Fee Related legal-status Critical Current
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020127005927A 2009-08-07 2010-08-05 Ｎ1-아실-5-플루오로피리미디논 유도체 Expired - Fee Related KR101792285B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
US61/232,223 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (2)

Publication Number Publication Date
KR20120041786A KR20120041786A (ko) 2012-05-02
KR101792285B1 true KR101792285B1 (ko) 2017-10-31

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020127005927A Expired - Fee Related KR101792285B1 (ko) 2009-08-07 2010-08-05 Ｎ1-아실-5-플루오로피리미디논 유도체

Country Status (33)

Country Link
US (1) US8470839B2 (enExample)
EP (1) EP2519512B1 (enExample)
JP (1) JP5748754B2 (enExample)
KR (1) KR101792285B1 (enExample)
CN (1) CN102548981B (enExample)
AU (1) AU2010279402B2 (enExample)
BR (1) BR112012002810B1 (enExample)
CA (1) CA2768510C (enExample)
CL (1) CL2012000316A1 (enExample)
CO (1) CO6491117A2 (enExample)
CR (1) CR20120030A (enExample)
CY (1) CY1122115T1 (enExample)
DK (1) DK2519512T3 (enExample)
EA (1) EA023411B1 (enExample)
EC (1) ECSP12011653A (enExample)
ES (1) ES2728966T3 (enExample)
HN (1) HN2012000269A (enExample)
HR (1) HRP20190919T1 (enExample)
HU (1) HUE045290T2 (enExample)
IL (1) IL217952A (enExample)
IN (1) IN2012DN00539A (enExample)
LT (1) LT2519512T (enExample)
MX (1) MX2012001620A (enExample)
NI (1) NI201200022A (enExample)
NZ (1) NZ597570A (enExample)
PE (1) PE20120688A1 (enExample)
PL (1) PL2519512T3 (enExample)
PT (1) PT2519512T (enExample)
SI (1) SI2519512T1 (enExample)
TR (1) TR201908180T4 (enExample)
UA (1) UA106889C2 (enExample)
WO (1) WO2011017538A1 (enExample)
ZA (1) ZA201200819B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
RS56609B1 (sr) 2011-08-17 2018-02-28 Adama Makhteshim Ltd 1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji bilja
CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体
WO2014105821A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997033890A1 (en) 1996-03-11 1997-09-18 Novartis Ag Pyrimidin-4-one derivatives as pesticide

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
EP0836602B1 (en) * 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562166B1 (en) * 2008-01-22 2015-08-19 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
EP2317851B1 (en) 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
PL2389375T3 (pl) 2009-01-23 2015-11-30 Euro Celtique Sa Pochodne kwasu hydroksamowego
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997033890A1 (en) 1996-03-11 1997-09-18 Novartis Ag Pyrimidin-4-one derivatives as pesticide

Also Published As

Publication number Publication date
LT2519512T (lt) 2019-07-25
BR112012002810A2 (pt) 2015-09-15
MX2012001620A (es) 2012-04-11
CL2012000316A1 (es) 2014-06-27
CA2768510A1 (en) 2011-02-10
NI201200022A (es) 2012-05-22
JP2013501723A (ja) 2013-01-17
BR112012002810B1 (pt) 2018-12-11
CR20120030A (es) 2012-03-28
AU2010279402B2 (en) 2015-04-16
TR201908180T4 (tr) 2019-06-21
ES2728966T3 (es) 2019-10-29
DK2519512T3 (da) 2019-05-27
IL217952A0 (en) 2012-03-29
EA023411B1 (ru) 2016-06-30
HRP20190919T1 (hr) 2019-09-20
JP5748754B2 (ja) 2015-07-15
NZ597570A (en) 2014-04-30
WO2011017538A1 (en) 2011-02-10
IN2012DN00539A (enExample) 2015-06-12
EP2519512B1 (en) 2019-03-20
EP2519512A4 (en) 2013-01-16
PL2519512T3 (pl) 2019-09-30
CO6491117A2 (es) 2012-07-31
CY1122115T1 (el) 2020-11-25
KR20120041786A (ko) 2012-05-02
UA106889C2 (uk) 2014-10-27
EA201270253A1 (ru) 2012-07-30
AU2010279402A1 (en) 2012-02-02
PE20120688A1 (es) 2012-06-06
US8470839B2 (en) 2013-06-25
CN102548981B (zh) 2015-05-13
SI2519512T1 (sl) 2019-09-30
HN2012000269A (es) 2015-04-27
IL217952A (en) 2017-11-30
ZA201200819B (en) 2013-05-29
EP2519512A1 (en) 2012-11-07
PT2519512T (pt) 2019-06-04
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
CN102548981A (zh) 2012-07-04
US20110034490A1 (en) 2011-02-10
HK1172894A1 (en) 2013-05-03
CA2768510C (en) 2018-05-15

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