LT2519512T - N1-acil- 5-fluorpirimidinono dariniai - Google Patents

N1-acil- 5-fluorpirimidinono dariniai

Info

Publication number
LT2519512T
LT2519512T LTEP10807171.3T LT10807171T LT2519512T LT 2519512 T LT2519512 T LT 2519512T LT 10807171 T LT10807171 T LT 10807171T LT 2519512 T LT2519512 T LT 2519512T
Authority
LT
Lithuania
Prior art keywords
acyl
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
LTEP10807171.3T
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W. Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT2519512(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of LT2519512T publication Critical patent/LT2519512T/lt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LTEP10807171.3T 2009-08-07 2010-08-05 N1-acil- 5-fluorpirimidinono dariniai LT2519512T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
LT2519512T true LT2519512T (lt) 2019-07-25

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEP10807171.3T LT2519512T (lt) 2009-08-07 2010-08-05 N1-acil- 5-fluorpirimidinono dariniai

Country Status (34)

Country Link
US (1) US8470839B2 (lt)
EP (1) EP2519512B1 (lt)
JP (1) JP5748754B2 (lt)
KR (1) KR101792285B1 (lt)
CN (1) CN102548981B (lt)
AU (1) AU2010279402B2 (lt)
BR (1) BR112012002810B1 (lt)
CA (1) CA2768510C (lt)
CL (1) CL2012000316A1 (lt)
CO (1) CO6491117A2 (lt)
CR (1) CR20120030A (lt)
CY (1) CY1122115T1 (lt)
DK (1) DK2519512T3 (lt)
EA (1) EA023411B1 (lt)
EC (1) ECSP12011653A (lt)
ES (1) ES2728966T3 (lt)
HK (1) HK1172894A1 (lt)
HN (1) HN2012000269A (lt)
HR (1) HRP20190919T1 (lt)
HU (1) HUE045290T2 (lt)
IL (1) IL217952A (lt)
IN (1) IN2012DN00539A (lt)
LT (1) LT2519512T (lt)
MX (1) MX2012001620A (lt)
NI (1) NI201200022A (lt)
NZ (1) NZ597570A (lt)
PE (1) PE20120688A1 (lt)
PL (1) PL2519512T3 (lt)
PT (1) PT2519512T (lt)
SI (1) SI2519512T1 (lt)
TR (1) TR201908180T4 (lt)
UA (1) UA106889C2 (lt)
WO (1) WO2011017538A1 (lt)
ZA (1) ZA201200819B (lt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011017547A1 (en) * 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
ES2646725T3 (es) 2011-08-17 2017-12-15 Adama Makhteshim Ltd. Derivados 1-sustituidos de 5-fluoro-3,6-dihidro-6-imino-2(1H)-pirimidinona como agentes fungicidas para uso en protección de plantas
US9622474B2 (en) 2012-12-28 2017-04-18 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylate derivatives
AU2013370490B2 (en) 2012-12-28 2018-05-10 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives
EP2945635A4 (en) * 2012-12-28 2016-05-25 Dow Agrosciences Llc 1- (BENZOYL-SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-3,4-DIHYDROPYRIMIDIN-2 (1H) -ONE DERIVATIVES
US9642368B2 (en) 2012-12-31 2017-05-09 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
NZ722438A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
US10011617B2 (en) 2014-09-26 2018-07-03 The Chemours Company Fc, Llc Isocyanate derived organosilanes
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (lt) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
PL324486A1 (en) * 1995-07-05 1998-05-25 Du Pont Fungicidal pyrimidinones
EP0888359B1 (en) * 1996-03-11 2002-05-02 Syngenta Participations AG Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) * 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINE DERIVATIVE
WO2008005303A2 (en) * 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
PL2562162T3 (pl) * 2008-01-22 2016-01-29 Dow Agrosciences Llc Pochodne N-cyjano-4-amino-5-fluoropirymidyny jako fungicydy
ES2456272T3 (es) 2008-08-01 2014-04-21 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida
CA2750413C (en) 2009-01-23 2016-06-21 Northlake Biosciences Llc Hydroxamic acid derivatives
WO2011017547A1 (en) * 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
AU2010279402B2 (en) 2015-04-16
PL2519512T3 (pl) 2019-09-30
CR20120030A (es) 2012-03-28
US8470839B2 (en) 2013-06-25
BR112012002810A2 (pt) 2015-09-15
EA201270253A1 (ru) 2012-07-30
US20110034490A1 (en) 2011-02-10
IN2012DN00539A (lt) 2015-06-12
KR20120041786A (ko) 2012-05-02
TR201908180T4 (tr) 2019-06-21
EP2519512B1 (en) 2019-03-20
WO2011017538A1 (en) 2011-02-10
MX2012001620A (es) 2012-04-11
CO6491117A2 (es) 2012-07-31
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
PE20120688A1 (es) 2012-06-06
ZA201200819B (en) 2013-05-29
KR101792285B1 (ko) 2017-10-31
CY1122115T1 (el) 2020-11-25
EP2519512A1 (en) 2012-11-07
JP2013501723A (ja) 2013-01-17
HN2012000269A (es) 2015-04-27
CA2768510A1 (en) 2011-02-10
BR112012002810B1 (pt) 2018-12-11
EA023411B1 (ru) 2016-06-30
CN102548981A (zh) 2012-07-04
IL217952A (en) 2017-11-30
NI201200022A (es) 2012-05-22
DK2519512T3 (da) 2019-05-27
CN102548981B (zh) 2015-05-13
AU2010279402A1 (en) 2012-02-02
ES2728966T3 (es) 2019-10-29
JP5748754B2 (ja) 2015-07-15
HK1172894A1 (en) 2013-05-03
NZ597570A (en) 2014-04-30
UA106889C2 (uk) 2014-10-27
SI2519512T1 (sl) 2019-09-30
EP2519512A4 (en) 2013-01-16
CL2012000316A1 (es) 2014-06-27
CA2768510C (en) 2018-05-15
HRP20190919T1 (hr) 2019-09-20
IL217952A0 (en) 2012-03-29
PT2519512T (pt) 2019-06-04

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