PE20120688A1 - Derivados de n1-acil-5-fluoropirimidinona - Google Patents

Derivados de n1-acil-5-fluoropirimidinona

Info

Publication number
PE20120688A1
PE20120688A1 PE2012000169A PE2012000169A PE20120688A1 PE 20120688 A1 PE20120688 A1 PE 20120688A1 PE 2012000169 A PE2012000169 A PE 2012000169A PE 2012000169 A PE2012000169 A PE 2012000169A PE 20120688 A1 PE20120688 A1 PE 20120688A1
Authority
PE
Peru
Prior art keywords
fluoro
alkyl
optionally substituted
fluoropyrimidinone
acil
Prior art date
Application number
PE2012000169A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20120688(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PE20120688A1 publication Critical patent/PE20120688A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS DE N1-ACIL-5-FLUOROPIRIMIDINONA DE FORMULA (I) DONDE R1 ES H, ALQUILO(C1-C6) OPCIONALMENTE SUSTITUIDO CON R4, ALQUINILO(C3-C6) OPCIONALMENTE SUSTITUIDO CON R4, FENILO, ENTRE OTROS; R2 ES H, ALQUILO(C1-C6) OPCIONALMENTE SUSTITUIDO CON R4, ENTRE OTROS, EN DONDE R4 ES HALOGENO, ALQUILO(C1-C6), ALCOXI(C1-C4), ALQUILTIO(C1-C4), ENTRE OTROS; R3 ES -C(=O)R8 O -C(=S)R8, EN DONDE R8 ES H, ALQUENILO(C2-C6), HALOALQUILO(C1-C6), FENILO, ENTRE OTROS. SON COMPUESTOS PREFERIDOS: N'-(1-ACETIL-5-FLUORO-2-OXO-1,2-DIHIDROPIRIMIDIN-4-IL)-N,N-DIMETILFORMAMIDINA; N'-[1-(2,6-DICLOROBENZOIL)-5-FLUORO-2-OXO-1,2-DIHIDRO-PIRIMIDIN-4-IL]-N,N-DIMETILFORMAMIDINA; 4-AMINO-1-(3,5-DIFLUOROBENZOIL)-5-FLUORO-1H-PIRIMIDIN-2-ONA; ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION. DICHOS COMPUESTOS SON FUNGICIDAS SIENDO UTILES PARA EL CONTROL Y PREVENCION DEL ATAQUE FUNGICO EN PLANTAS
PE2012000169A 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona PE20120688A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
PE20120688A1 true PE20120688A1 (es) 2012-06-06

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2012000169A PE20120688A1 (es) 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona

Country Status (34)

Country Link
US (1) US8470839B2 (es)
EP (1) EP2519512B1 (es)
JP (1) JP5748754B2 (es)
KR (1) KR101792285B1 (es)
CN (1) CN102548981B (es)
AU (1) AU2010279402B2 (es)
BR (1) BR112012002810B1 (es)
CA (1) CA2768510C (es)
CL (1) CL2012000316A1 (es)
CO (1) CO6491117A2 (es)
CR (1) CR20120030A (es)
CY (1) CY1122115T1 (es)
DK (1) DK2519512T3 (es)
EA (1) EA023411B1 (es)
EC (1) ECSP12011653A (es)
ES (1) ES2728966T3 (es)
HK (1) HK1172894A1 (es)
HN (1) HN2012000269A (es)
HR (1) HRP20190919T1 (es)
HU (1) HUE045290T2 (es)
IL (1) IL217952A (es)
IN (1) IN2012DN00539A (es)
LT (1) LT2519512T (es)
MX (1) MX2012001620A (es)
NI (1) NI201200022A (es)
NZ (1) NZ597570A (es)
PE (1) PE20120688A1 (es)
PL (1) PL2519512T3 (es)
PT (1) PT2519512T (es)
SI (1) SI2519512T1 (es)
TR (1) TR201908180T4 (es)
UA (1) UA106889C2 (es)
WO (1) WO2011017538A1 (es)
ZA (1) ZA201200819B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS53395B (en) * 2009-08-07 2014-10-31 Dow Agrosciences Llc DERIVATIVES N1-SULFONIL-5-FLUORPIRIMIDINONA
WO2013025795A1 (en) * 2011-08-17 2013-02-21 Dow Agrosciences Llc 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives
US9271497B2 (en) * 2012-12-28 2016-03-01 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
KR20150103096A (ko) 2012-12-28 2015-09-09 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체
RU2644014C2 (ru) 2012-12-31 2018-02-07 Адама Мактешим Лтд. Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов
EA201691353A1 (ru) 2013-12-31 2016-12-30 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
EP3096619A4 (en) 2013-12-31 2017-09-06 Adama Makhteshim Ltd Synergistic fungicidal mixtures for fungal control in cereals
US10011617B2 (en) 2014-09-26 2018-07-03 The Chemours Company Fc, Llc Isocyanate derived organosilanes
JP2020527563A (ja) 2017-07-17 2020-09-10 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−メチル−１−トシル−３，４−ジヒドロピリミジン−２−オンの多形体

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CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
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US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (es) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
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DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
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JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
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RS53395B (en) 2009-08-07 2014-10-31 Dow Agrosciences Llc DERIVATIVES N1-SULFONIL-5-FLUORPIRIMIDINONA

Also Published As

Publication number Publication date
UA106889C2 (uk) 2014-10-27
IN2012DN00539A (es) 2015-06-12
MX2012001620A (es) 2012-04-11
PL2519512T3 (pl) 2019-09-30
ZA201200819B (en) 2013-05-29
AU2010279402A1 (en) 2012-02-02
HK1172894A1 (en) 2013-05-03
EP2519512B1 (en) 2019-03-20
CY1122115T1 (el) 2020-11-25
KR101792285B1 (ko) 2017-10-31
EP2519512A4 (en) 2013-01-16
WO2011017538A1 (en) 2011-02-10
EA023411B1 (ru) 2016-06-30
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
CL2012000316A1 (es) 2014-06-27
HN2012000269A (es) 2015-04-27
LT2519512T (lt) 2019-07-25
CN102548981A (zh) 2012-07-04
PT2519512T (pt) 2019-06-04
JP5748754B2 (ja) 2015-07-15
US8470839B2 (en) 2013-06-25
IL217952A0 (en) 2012-03-29
BR112012002810A2 (pt) 2015-09-15
NI201200022A (es) 2012-05-22
SI2519512T1 (sl) 2019-09-30
CR20120030A (es) 2012-03-28
AU2010279402B2 (en) 2015-04-16
EA201270253A1 (ru) 2012-07-30
US20110034490A1 (en) 2011-02-10
CO6491117A2 (es) 2012-07-31
CA2768510A1 (en) 2011-02-10
JP2013501723A (ja) 2013-01-17
CA2768510C (en) 2018-05-15
NZ597570A (en) 2014-04-30
TR201908180T4 (tr) 2019-06-21
KR20120041786A (ko) 2012-05-02
IL217952A (en) 2017-11-30
BR112012002810B1 (pt) 2018-12-11
CN102548981B (zh) 2015-05-13
DK2519512T3 (da) 2019-05-27
HRP20190919T1 (hr) 2019-09-20
ES2728966T3 (es) 2019-10-29
EP2519512A1 (en) 2012-11-07

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