CO6491117A2 - Derivados de n1-acil-5-fluoropirimidinona - Google Patents

Derivados de n1-acil-5-fluoropirimidinona

Info

Publication number
CO6491117A2
CO6491117A2 CO12019954A CO12019954A CO6491117A2 CO 6491117 A2 CO6491117 A2 CO 6491117A2 CO 12019954 A CO12019954 A CO 12019954A CO 12019954 A CO12019954 A CO 12019954A CO 6491117 A2 CO6491117 A2 CO 6491117A2
Authority
CO
Colombia
Prior art keywords
compounds
formulations
formula
present description
fluoropirimidinona
Prior art date
Application number
CO12019954A
Other languages
English (en)
Spanish (es)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6491117(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of CO6491117A2 publication Critical patent/CO6491117A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CO12019954A 2009-08-07 2012-02-06 Derivados de n1-acil-5-fluoropirimidinona CO6491117A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
CO6491117A2 true CO6491117A2 (es) 2012-07-31

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
CO12019954A CO6491117A2 (es) 2009-08-07 2012-02-06 Derivados de n1-acil-5-fluoropirimidinona

Country Status (33)

Country Link
US (1) US8470839B2 (enExample)
EP (1) EP2519512B1 (enExample)
JP (1) JP5748754B2 (enExample)
KR (1) KR101792285B1 (enExample)
CN (1) CN102548981B (enExample)
AU (1) AU2010279402B2 (enExample)
BR (1) BR112012002810B1 (enExample)
CA (1) CA2768510C (enExample)
CL (1) CL2012000316A1 (enExample)
CO (1) CO6491117A2 (enExample)
CR (1) CR20120030A (enExample)
CY (1) CY1122115T1 (enExample)
DK (1) DK2519512T3 (enExample)
EA (1) EA023411B1 (enExample)
EC (1) ECSP12011653A (enExample)
ES (1) ES2728966T3 (enExample)
HN (1) HN2012000269A (enExample)
HR (1) HRP20190919T1 (enExample)
HU (1) HUE045290T2 (enExample)
IL (1) IL217952A (enExample)
IN (1) IN2012DN00539A (enExample)
LT (1) LT2519512T (enExample)
MX (1) MX2012001620A (enExample)
NI (1) NI201200022A (enExample)
NZ (1) NZ597570A (enExample)
PE (1) PE20120688A1 (enExample)
PL (1) PL2519512T3 (enExample)
PT (1) PT2519512T (enExample)
SI (1) SI2519512T1 (enExample)
TR (1) TR201908180T4 (enExample)
UA (1) UA106889C2 (enExample)
WO (1) WO2011017538A1 (enExample)
ZA (1) ZA201200819B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
RS56609B1 (sr) 2011-08-17 2018-02-28 Adama Makhteshim Ltd 1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji bilja
CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体
WO2014105821A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound

Family Cites Families (22)

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Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
EP0836602B1 (en) * 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
DE69712331T2 (de) * 1996-03-11 2002-11-28 Syngenta Participations Ag, Basel Pyrimidin-4-on derivate als pestizidesmittel
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562166B1 (en) * 2008-01-22 2015-08-19 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
EP2317851B1 (en) 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
PL2389375T3 (pl) 2009-01-23 2015-11-30 Euro Celtique Sa Pochodne kwasu hydroksamowego
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体

Also Published As

Publication number Publication date
LT2519512T (lt) 2019-07-25
BR112012002810A2 (pt) 2015-09-15
MX2012001620A (es) 2012-04-11
CL2012000316A1 (es) 2014-06-27
CA2768510A1 (en) 2011-02-10
NI201200022A (es) 2012-05-22
JP2013501723A (ja) 2013-01-17
BR112012002810B1 (pt) 2018-12-11
CR20120030A (es) 2012-03-28
AU2010279402B2 (en) 2015-04-16
TR201908180T4 (tr) 2019-06-21
ES2728966T3 (es) 2019-10-29
DK2519512T3 (da) 2019-05-27
IL217952A0 (en) 2012-03-29
EA023411B1 (ru) 2016-06-30
HRP20190919T1 (hr) 2019-09-20
JP5748754B2 (ja) 2015-07-15
NZ597570A (en) 2014-04-30
WO2011017538A1 (en) 2011-02-10
IN2012DN00539A (enExample) 2015-06-12
EP2519512B1 (en) 2019-03-20
EP2519512A4 (en) 2013-01-16
PL2519512T3 (pl) 2019-09-30
CY1122115T1 (el) 2020-11-25
KR20120041786A (ko) 2012-05-02
UA106889C2 (uk) 2014-10-27
EA201270253A1 (ru) 2012-07-30
AU2010279402A1 (en) 2012-02-02
PE20120688A1 (es) 2012-06-06
US8470839B2 (en) 2013-06-25
CN102548981B (zh) 2015-05-13
SI2519512T1 (sl) 2019-09-30
HN2012000269A (es) 2015-04-27
IL217952A (en) 2017-11-30
ZA201200819B (en) 2013-05-29
KR101792285B1 (ko) 2017-10-31
EP2519512A1 (en) 2012-11-07
PT2519512T (pt) 2019-06-04
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
CN102548981A (zh) 2012-07-04
US20110034490A1 (en) 2011-02-10
HK1172894A1 (en) 2013-05-03
CA2768510C (en) 2018-05-15

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