MX354021B - Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona. - Google Patents

Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona.

Info

Publication number
MX354021B
MX354021B MX2014001885A MX2014001885A MX354021B MX 354021 B MX354021 B MX 354021B MX 2014001885 A MX2014001885 A MX 2014001885A MX 2014001885 A MX2014001885 A MX 2014001885A MX 354021 B MX354021 B MX 354021B
Authority
MX
Mexico
Prior art keywords
dihydropyrimidin
imino
fluoro
derivatives
substituted
Prior art date
Application number
MX2014001885A
Other languages
English (en)
Other versions
MX2014001885A (es
Inventor
A Boebel Timothy
Lorsbach Beth
W Owen John
T Sullenberger Michael
D Webster Jeffery
Yao Chenglin
V Galliford Chris
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47713076&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX354021(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of MX2014001885A publication Critical patent/MX2014001885A/es
Publication of MX354021B publication Critical patent/MX354021B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Abstract

La presente descripción se refiere al campo de las 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidina-2(1H)onas y sus derivados y al uso de estos compuestos como fungicidas.
MX2014001885A 2011-08-17 2012-08-15 Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona. MX354021B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161524506P 2011-08-17 2011-08-17
PCT/US2012/050930 WO2013025795A1 (en) 2011-08-17 2012-08-15 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives

Publications (2)

Publication Number Publication Date
MX2014001885A MX2014001885A (es) 2014-05-30
MX354021B true MX354021B (es) 2018-02-08

Family

ID=47713076

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014001885A MX354021B (es) 2011-08-17 2012-08-15 Derivados de 5-fluor-4-imino-3- (sustituido) -3,4-dihidropirimidin -2 (1h) ona.

Country Status (31)

Country Link
US (1) US8658660B2 (es)
EP (1) EP2775842B1 (es)
JP (3) JP6128658B2 (es)
KR (1) KR102012992B1 (es)
CN (2) CN106977462B (es)
AR (1) AR087549A1 (es)
BR (1) BR112014003587B1 (es)
CA (1) CA2844497C (es)
CL (1) CL2014000352A1 (es)
CO (1) CO6910204A2 (es)
CR (1) CR20140058A (es)
DK (1) DK2775842T3 (es)
EC (1) ECSP14013251A (es)
ES (1) ES2646725T3 (es)
GT (1) GT201400023A (es)
HK (1) HK1199177A1 (es)
HR (1) HRP20171776T1 (es)
HU (1) HUE035248T2 (es)
IL (1) IL230981A (es)
LT (1) LT2775842T (es)
ME (1) ME02924B (es)
MX (1) MX354021B (es)
NO (1) NO2874589T3 (es)
PL (1) PL2775842T3 (es)
PT (1) PT2775842T (es)
RS (1) RS56609B1 (es)
RU (1) RU2613451C2 (es)
SI (1) SI2775842T1 (es)
UA (1) UA113062C2 (es)
WO (1) WO2013025795A1 (es)
ZA (1) ZA201400875B (es)

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LT2775842T (lt) * 2011-08-17 2017-12-11 Adama Makhteshim Ltd. 1-pakeisti-5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinono dariniai, kaip fungicidiniai agentai, skirti panaudoti augalų apsaugai
RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
UA117743C2 (uk) 2012-12-28 2018-09-25 Адама Махтешім Лтд. N-(заміщені)-5-фтор-4-іміно-3-метил-2-оксо-3,4-дигідропіримідин-1(2h)-карбоксамідні похідні
RU2644014C2 (ru) 2012-12-31 2018-02-07 Адама Мактешим Лтд. Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов
CN103819412B (zh) * 2013-12-11 2016-02-03 浙江先锋科技股份有限公司 一种5-氟胞嘧啶的制备方法
CR20210172A (es) * 2013-12-31 2021-05-11 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2 (1h)-ona y los procesos para su preparación
BR112016015155A2 (pt) 2013-12-31 2017-08-08 Adama Makhteshim Ltd Misturas fungicidas sinergísticas para controle fúngico em cereais
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
TWI774761B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TWI774760B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於蔬菜中的真菌防治之協同性混合物
TWI774762B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途
TW201842851A (zh) * 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
TWI801380B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途
TWI801381B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CN109053553A (zh) * 2018-10-16 2018-12-21 山东省农药科学研究院 杀虫剂氟啶虫胺腈中间体3-[1-(甲硫基)乙基]-6(三氟甲基)吡啶的合成方法
WO2021031431A1 (en) 2019-08-22 2021-02-25 Fujian Yongjing Technology Co., Ltd Process for preparing fluorobenzene by direct fluorination
US20230104954A1 (en) * 2020-03-09 2023-04-06 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
AR127068A1 (es) * 2021-09-15 2023-12-13 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1(tolueno-4-sulfonil)-3,4-dihidro-1h-pirimidin-2-ona

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Also Published As

Publication number Publication date
CN106977462B (zh) 2020-04-28
KR20140057605A (ko) 2014-05-13
BR112014003587A8 (pt) 2017-07-11
DK2775842T3 (en) 2017-12-18
MX2014001885A (es) 2014-05-30
US20130045984A1 (en) 2013-02-21
BR112014003587B1 (pt) 2021-04-13
ECSP14013251A (es) 2014-04-30
RU2014110049A (ru) 2015-09-27
JP2014524440A (ja) 2014-09-22
AU2012296629A1 (en) 2014-02-20
JP2017125060A (ja) 2017-07-20
RU2613451C2 (ru) 2017-03-16
RS56609B1 (sr) 2018-02-28
CA2844497A1 (en) 2013-02-21
HK1199177A1 (en) 2015-06-26
CN106977462A (zh) 2017-07-25
AU2012296629B2 (en) 2016-02-11
SI2775842T1 (en) 2018-01-31
CO6910204A2 (es) 2014-03-31
AR087549A1 (es) 2014-04-03
WO2013025795A1 (en) 2013-02-21
JP6901462B2 (ja) 2021-07-14
GT201400023A (es) 2015-02-27
AU2012296629A8 (en) 2016-06-16
CN103874413A (zh) 2014-06-18
EP2775842A1 (en) 2014-09-17
IL230981A (en) 2017-10-31
CN103874413B (zh) 2017-03-08
UA113062C2 (xx) 2016-12-12
EP2775842A4 (en) 2015-04-15
CA2844497C (en) 2021-03-02
HRP20171776T1 (hr) 2018-01-26
ZA201400875B (en) 2015-04-29
JP6128658B2 (ja) 2017-05-17
NZ620537A (en) 2016-11-25
EP2775842B1 (en) 2017-10-04
NO2874589T3 (es) 2018-02-03
CR20140058A (es) 2014-03-20
PL2775842T3 (pl) 2018-02-28
HUE035248T2 (en) 2018-05-02
IL230981A0 (en) 2014-03-31
LT2775842T (lt) 2017-12-11
ES2646725T3 (es) 2017-12-15
JP2019088283A (ja) 2019-06-13
US8658660B2 (en) 2014-02-25
KR102012992B1 (ko) 2019-08-21
ME02924B (me) 2018-04-20
BR112014003587A2 (pt) 2017-03-14
CL2014000352A1 (es) 2014-07-25
PT2775842T (pt) 2017-11-15

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