CO6910204A2 - Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona - Google Patents

Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona

Info

Publication number
CO6910204A2
CO6910204A2 CO14055677A CO14055677A CO6910204A2 CO 6910204 A2 CO6910204 A2 CO 6910204A2 CO 14055677 A CO14055677 A CO 14055677A CO 14055677 A CO14055677 A CO 14055677A CO 6910204 A2 CO6910204 A2 CO 6910204A2
Authority
CO
Colombia
Prior art keywords
dihydropyrimidin
imino
fluoro
derivatives
substituted
Prior art date
Application number
CO14055677A
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
W John Owen
Michael Sullenberger
Jeffery D Webster
Chenglin Yao
Chris Galliford
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47713076&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6910204(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of CO6910204A2 publication Critical patent/CO6910204A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
CO14055677A 2011-08-17 2014-03-14 Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona CO6910204A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161524506P 2011-08-17 2011-08-17

Publications (1)

Publication Number Publication Date
CO6910204A2 true CO6910204A2 (es) 2014-03-31

Family

ID=47713076

Family Applications (1)

Application Number Title Priority Date Filing Date
CO14055677A CO6910204A2 (es) 2011-08-17 2014-03-14 Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona

Country Status (31)

Country Link
US (1) US8658660B2 (es)
EP (1) EP2775842B1 (es)
JP (3) JP6128658B2 (es)
KR (1) KR102012992B1 (es)
CN (2) CN103874413B (es)
AR (1) AR087549A1 (es)
BR (1) BR112014003587B1 (es)
CA (1) CA2844497C (es)
CL (1) CL2014000352A1 (es)
CO (1) CO6910204A2 (es)
CR (1) CR20140058A (es)
DK (1) DK2775842T3 (es)
EC (1) ECSP14013251A (es)
ES (1) ES2646725T3 (es)
GT (1) GT201400023A (es)
HK (1) HK1199177A1 (es)
HR (1) HRP20171776T1 (es)
HU (1) HUE035248T2 (es)
IL (1) IL230981A (es)
LT (1) LT2775842T (es)
ME (1) ME02924B (es)
MX (1) MX354021B (es)
NO (1) NO2874589T3 (es)
PL (1) PL2775842T3 (es)
PT (1) PT2775842T (es)
RS (1) RS56609B1 (es)
RU (1) RU2613451C2 (es)
SI (1) SI2775842T1 (es)
UA (1) UA113062C2 (es)
WO (1) WO2013025795A1 (es)
ZA (1) ZA201400875B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-Substituted-5-fluoro-3,6-dihydro-6-imino-2 (1H) -pyrimidinone derivatives as fungicidal compositions for use in plant protection
MX2015008444A (es) 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
WO2014105844A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
CN103819412B (zh) * 2013-12-11 2016-02-03 浙江先锋科技股份有限公司 一种5-氟胞嘧啶的制备方法
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
MX2016008758A (es) 2013-12-31 2017-05-09 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4 -dihidropirimidin-2(1h)-ona y los procesos para su preparacion.
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
TWI774762B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途
TWI774761B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) * 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
TWI801381B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途
TWI774760B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於蔬菜中的真菌防治之協同性混合物
TWI801380B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途
IL309708A (en) 2017-07-17 2024-02-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
CN109053553A (zh) * 2018-10-16 2018-12-21 山东省农药科学研究院 杀虫剂氟啶虫胺腈中间体3-[1-(甲硫基)乙基]-6(三氟甲基)吡啶的合成方法
JP7353012B2 (ja) 2019-08-22 2023-09-29 フジアン ヨンジン テクノロジー カンパニー リミテッド 直接フッ素化によるフルオロベンゼンの製造プロセス
IL296178A (en) * 2020-03-09 2022-11-01 Adama Makhteshim Ltd Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-4,3-dihydro-1h-pyrimidin-2-one
WO2023042126A1 (en) * 2021-09-15 2023-03-23 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one

Family Cites Families (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3635977A (en) * 1969-11-03 1972-01-18 American Cyanamid Co Certain 6-trifluoromethylcytosines and thiocytosines their synthesis and their use in the synthesis of uracisls and thiouracil
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (es) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
DE69618959T2 (de) 1995-07-05 2002-08-29 Du Pont Pyrimidone und ihre verwendug als fungizide
US6262058B1 (en) 1996-03-11 2001-07-17 Syngenta Crop Protection, Inc. Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
EA009517B1 (ru) * 2003-06-27 2008-02-28 Байер Кропсайенс Аг Пиразолопиримидины
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
TWI402034B (zh) 2005-07-28 2013-07-21 Dow Agrosciences Llc 具有被層狀液晶覆膜包覆之油球之水包油乳化劑之農用組成物
EP2617287A1 (en) * 2005-11-22 2013-07-24 Ishihara Sangyo Kaisha, Ltd. Germicide composition for agricultural and gardening applications and method for controlling plant disease
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
ES2549379T3 (es) 2008-01-22 2015-10-27 Dow Agrosciences Llc Derivados de 4-amino5-fluoropirimidina como fungicidas
UA107651C2 (en) 2008-08-01 2015-02-10 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
US8278341B2 (en) * 2008-09-17 2012-10-02 Sri International Analogs of indole-3-carbinol and their use as agents against infection
RS54192B1 (en) 2009-01-23 2015-12-31 Euro-Celtique S.A. DERIVATIVES OF HYDROXAMIC ACIDS
BR112012002830B1 (pt) * 2009-08-07 2019-05-28 Adama Makhteshim Ltd. Derivados de n1-sulfonil-5-fluoropiri-midinona, composição para controle de um patógeno fúngico, e método para controle ou prevenção de ataque de fungos em uma planta
UA106889C2 (uk) * 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-ацил-5-фторпіримідинону
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
UA106246C2 (ru) * 2009-10-07 2014-08-11 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Синергическая фунгицидная композиция, которая содержит 5-фторцитозин для борьбы с грибковыми болезнями зерновых культур
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-Substituted-5-fluoro-3,6-dihydro-6-imino-2 (1H) -pyrimidinone derivatives as fungicidal compositions for use in plant protection

Also Published As

Publication number Publication date
GT201400023A (es) 2015-02-27
ECSP14013251A (es) 2014-04-30
US8658660B2 (en) 2014-02-25
MX354021B (es) 2018-02-08
IL230981A0 (en) 2014-03-31
JP2014524440A (ja) 2014-09-22
CA2844497C (en) 2021-03-02
UA113062C2 (xx) 2016-12-12
DK2775842T3 (en) 2017-12-18
CR20140058A (es) 2014-03-20
RU2014110049A (ru) 2015-09-27
AU2012296629B2 (en) 2016-02-11
CN106977462A (zh) 2017-07-25
BR112014003587A8 (pt) 2017-07-11
BR112014003587A2 (pt) 2017-03-14
JP2017125060A (ja) 2017-07-20
RU2613451C2 (ru) 2017-03-16
ES2646725T3 (es) 2017-12-15
JP6128658B2 (ja) 2017-05-17
AU2012296629A8 (en) 2016-06-16
NO2874589T3 (es) 2018-02-03
KR20140057605A (ko) 2014-05-13
HK1199177A1 (en) 2015-06-26
BR112014003587B1 (pt) 2021-04-13
CN103874413B (zh) 2017-03-08
ME02924B (me) 2018-04-20
JP2019088283A (ja) 2019-06-13
AU2012296629A1 (en) 2014-02-20
SI2775842T1 (en) 2018-01-31
CL2014000352A1 (es) 2014-07-25
JP6901462B2 (ja) 2021-07-14
EP2775842A4 (en) 2015-04-15
WO2013025795A1 (en) 2013-02-21
LT2775842T (lt) 2017-12-11
NZ620537A (en) 2016-11-25
EP2775842A1 (en) 2014-09-17
ZA201400875B (en) 2015-04-29
HUE035248T2 (en) 2018-05-02
AR087549A1 (es) 2014-04-03
PL2775842T3 (pl) 2018-02-28
PT2775842T (pt) 2017-11-15
EP2775842B1 (en) 2017-10-04
US20130045984A1 (en) 2013-02-21
CA2844497A1 (en) 2013-02-21
CN106977462B (zh) 2020-04-28
HRP20171776T1 (hr) 2018-01-26
KR102012992B1 (ko) 2019-08-21
MX2014001885A (es) 2014-05-30
RS56609B1 (sr) 2018-02-28
CN103874413A (zh) 2014-06-18
IL230981A (en) 2017-10-31

Similar Documents

Publication Publication Date Title
CO6910204A2 (es) Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona
FR22C1047I2 (fr) Derives de benzimidazole-proline
CO6900145A2 (es) Compuesto de ciclopropanoamina
CO6890099A2 (es) Nuevos derivados dihidroquinolina-2-ona
CR20140147A (es) Inhibidores de aplicación viral
BR112013023048A2 (pt) composto de guanidina
CO7061068A2 (es) Derivados de polimixina
BR112013024378A2 (pt) novos derivados de pirimidina
CO7020919A2 (es) Derivados de tetrahidro-quinazolinona
DK2938194T3 (da) N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
CO6811866A2 (es) Derivados de benzamida sustituida
CO6960557A2 (es) Derivados de 2-yodo-imidazol
CL2014000325A1 (es) Compuestos derivados de piranos sustituidos, implicados en la señalizacion de nematodos
CO6920301A2 (es) Derivados insecticidas de 2-metoxibenzamida
BR112013030897A2 (pt) composição.
CO7020920A2 (es) Derivado de fenilazol sustituido
FR2978994B1 (fr) .
BR112013022508A2 (pt) novos compostos de azaespirodecanona
CO6852074A2 (es) Novedosos derivados de ftalazinona-pirrolopirimidinacarboxamida
BR112013023316A2 (pt) derivados de difenila substituídos
BR112015003217A2 (pt) novos derivados de piridina.
ES2397885B1 (es) Derivados de colismicina.
BR112013019806A2 (pt) derivado de tetrahidroisoquinolina.
FR2973145B1 (fr) Atlas visuo-tactile.
DE112012002210A5 (de) Drucksystem