BR112014003587A8 - Derivados de 5-flúor-4-imino-3-(substituído)-3,4-dihidropirimidin-2(1h)ona, composição e método para controle ou prevenção de um patógeno fúngico - Google Patents
Derivados de 5-flúor-4-imino-3-(substituído)-3,4-dihidropirimidin-2(1h)ona, composição e método para controle ou prevenção de um patógeno fúngicoInfo
- Publication number
- BR112014003587A8 BR112014003587A8 BR112014003587A BR112014003587A BR112014003587A8 BR 112014003587 A8 BR112014003587 A8 BR 112014003587A8 BR 112014003587 A BR112014003587 A BR 112014003587A BR 112014003587 A BR112014003587 A BR 112014003587A BR 112014003587 A8 BR112014003587 A8 BR 112014003587A8
- Authority
- BR
- Brazil
- Prior art keywords
- dihydropyrimidin
- imino
- derivatives
- fluorine
- replaced
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
Abstract
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161524506P | 2011-08-17 | 2011-08-17 | |
US61/524,506 | 2011-08-17 | ||
PCT/US2012/050930 WO2013025795A1 (en) | 2011-08-17 | 2012-08-15 | 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives |
Publications (3)
Publication Number | Publication Date |
---|---|
BR112014003587A2 BR112014003587A2 (pt) | 2017-03-14 |
BR112014003587A8 true BR112014003587A8 (pt) | 2017-07-11 |
BR112014003587B1 BR112014003587B1 (pt) | 2021-04-13 |
Family
ID=47713076
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014003587-3A BR112014003587B1 (pt) | 2011-08-17 | 2012-08-15 | Derivados de 5-flúor-4-imino-3-(substituído)-3,4-dihidropirimidin-2(1h)ona, composição e método para controle ou prevenção de um patógeno fúngico |
Country Status (31)
Country | Link |
---|---|
US (1) | US8658660B2 (pt) |
EP (1) | EP2775842B1 (pt) |
JP (3) | JP6128658B2 (pt) |
KR (1) | KR102012992B1 (pt) |
CN (2) | CN103874413B (pt) |
AR (1) | AR087549A1 (pt) |
BR (1) | BR112014003587B1 (pt) |
CA (1) | CA2844497C (pt) |
CL (1) | CL2014000352A1 (pt) |
CO (1) | CO6910204A2 (pt) |
CR (1) | CR20140058A (pt) |
DK (1) | DK2775842T3 (pt) |
EC (1) | ECSP14013251A (pt) |
ES (1) | ES2646725T3 (pt) |
GT (1) | GT201400023A (pt) |
HK (1) | HK1199177A1 (pt) |
HR (1) | HRP20171776T1 (pt) |
HU (1) | HUE035248T2 (pt) |
IL (1) | IL230981A (pt) |
LT (1) | LT2775842T (pt) |
ME (1) | ME02924B (pt) |
MX (1) | MX354021B (pt) |
NO (1) | NO2874589T3 (pt) |
PL (1) | PL2775842T3 (pt) |
PT (1) | PT2775842T (pt) |
RS (1) | RS56609B1 (pt) |
RU (1) | RU2613451C2 (pt) |
SI (1) | SI2775842T1 (pt) |
UA (1) | UA113062C2 (pt) |
WO (1) | WO2013025795A1 (pt) |
ZA (1) | ZA201400875B (pt) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013025795A1 (en) * | 2011-08-17 | 2013-02-21 | Dow Agrosciences Llc | 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives |
CN104884062B (zh) | 2012-12-28 | 2018-11-06 | 阿达玛马克西姆股份有限公司 | N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物 |
KR20150103096A (ko) | 2012-12-28 | 2015-09-09 | 다우 아그로사이언시즈 엘엘씨 | N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체 |
RU2644014C2 (ru) | 2012-12-31 | 2018-02-07 | Адама Мактешим Лтд. | Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов |
CN103819412B (zh) * | 2013-12-11 | 2016-02-03 | 浙江先锋科技股份有限公司 | 一种5-氟胞嘧啶的制备方法 |
EP3096619A4 (en) | 2013-12-31 | 2017-09-06 | Adama Makhteshim Ltd | Synergistic fungicidal mixtures for fungal control in cereals |
EA201691353A1 (ru) * | 2013-12-31 | 2016-12-30 | Адама Мактешим Лтд. | 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения |
MA41272A (fr) * | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
TWI801380B (zh) * | 2017-05-02 | 2023-05-11 | 美商科迪華農業科技有限責任公司 | 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途 |
TWI774762B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途 |
TW201842851A (zh) * | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
TWI801381B (zh) * | 2017-05-02 | 2023-05-11 | 美商科迪華農業科技有限責任公司 | 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途 |
TWI774761B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
TWI774760B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於蔬菜中的真菌防治之協同性混合物 |
JP2020527563A (ja) | 2017-07-17 | 2020-09-10 | アダマ・マクテシム・リミテッド | 5−フルオロ−4−イミノ−3−メチル−1−トシル−3,4−ジヒドロピリミジン−2−オンの多形体 |
CN109053553A (zh) * | 2018-10-16 | 2018-12-21 | 山东省农药科学研究院 | 杀虫剂氟啶虫胺腈中间体3-[1-(甲硫基)乙基]-6(三氟甲基)吡啶的合成方法 |
JP7353012B2 (ja) | 2019-08-22 | 2023-09-29 | フジアン ヨンジン テクノロジー カンパニー リミテッド | 直接フッ素化によるフルオロベンゼンの製造プロセス |
US20230104954A1 (en) * | 2020-03-09 | 2023-04-06 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
WO2023042126A1 (en) * | 2021-09-15 | 2023-03-23 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
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RS53395B (en) | 2009-08-07 | 2014-10-31 | Dow Agrosciences Llc | DERIVATIVES N1-SULFONIL-5-FLUORPIRIMIDINONA |
UA112284C2 (uk) | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
WO2011043876A1 (en) * | 2009-10-07 | 2011-04-14 | Dow Agrosciences Llc | Synergistic fungicidal composition containing 5-fluorocytosine for fungal control in cereals |
WO2013025795A1 (en) * | 2011-08-17 | 2013-02-21 | Dow Agrosciences Llc | 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives |
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2012
- 2012-08-15 WO PCT/US2012/050930 patent/WO2013025795A1/en active Application Filing
- 2012-08-15 CN CN201280049656.1A patent/CN103874413B/zh active Active
- 2012-08-15 AR ARP120102991A patent/AR087549A1/es active IP Right Grant
- 2012-08-15 CA CA2844497A patent/CA2844497C/en active Active
- 2012-08-15 HU HUE12824035A patent/HUE035248T2/en unknown
- 2012-08-15 DK DK12824035.5T patent/DK2775842T3/en active
- 2012-08-15 BR BR112014003587-3A patent/BR112014003587B1/pt active IP Right Grant
- 2012-08-15 JP JP2014526166A patent/JP6128658B2/ja active Active
- 2012-08-15 CN CN201710076214.0A patent/CN106977462B/zh active Active
- 2012-08-15 ES ES12824035.5T patent/ES2646725T3/es active Active
- 2012-08-15 PL PL12824035T patent/PL2775842T3/pl unknown
- 2012-08-15 MX MX2014001885A patent/MX354021B/es active IP Right Grant
- 2012-08-15 US US13/586,450 patent/US8658660B2/en active Active
- 2012-08-15 RU RU2014110049A patent/RU2613451C2/ru active
- 2012-08-15 UA UAA201402588A patent/UA113062C2/uk unknown
- 2012-08-15 LT LTEP12824035.5T patent/LT2775842T/lt unknown
- 2012-08-15 SI SI201231158T patent/SI2775842T1/en unknown
- 2012-08-15 EP EP12824035.5A patent/EP2775842B1/en active Active
- 2012-08-15 RS RS20171186A patent/RS56609B1/sr unknown
- 2012-08-15 ME MEP-2017-274A patent/ME02924B/me unknown
- 2012-08-15 PT PT128240355T patent/PT2775842T/pt unknown
- 2012-08-15 KR KR1020147006630A patent/KR102012992B1/ko active IP Right Grant
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2013
- 2013-07-19 NO NO13745256A patent/NO2874589T3/no unknown
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2014
- 2014-01-30 CR CR20140058A patent/CR20140058A/es unknown
- 2014-02-05 ZA ZA2014/00875A patent/ZA201400875B/en unknown
- 2014-02-12 CL CL2014000352A patent/CL2014000352A1/es unknown
- 2014-02-13 IL IL230981A patent/IL230981A/en active IP Right Grant
- 2014-02-14 GT GT201400023A patent/GT201400023A/es unknown
- 2014-03-14 CO CO14055677A patent/CO6910204A2/es unknown
- 2014-03-17 EC ECSP14013251 patent/ECSP14013251A/es unknown
- 2014-12-18 HK HK14112698.4A patent/HK1199177A1/xx unknown
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2017
- 2017-04-07 JP JP2017076823A patent/JP2017125060A/ja not_active Withdrawn
- 2017-11-16 HR HRP20171776TT patent/HRP20171776T1/hr unknown
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2018
- 2018-12-21 JP JP2018239307A patent/JP6901462B2/ja active Active
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Date | Code | Title | Description |
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B25A | Requested transfer of rights approved |
Owner name: ADAMA MAKHTESHIM LTD. (IL) |
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B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B07B | Technical examination (opinion): publication cancelled [chapter 7.2 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A01N 43/54 , A61K 31/505 Ipc: A01N 43/54 (1980.01), C07D 239/47 (1980.01), C07D |
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B15K | Others concerning applications: alteration of classification |
Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A01N 43/54 , C07D 239/47 , C07D 409/06 Ipc: A01N 43/54 (1980.01), C07D 239/47 (1980.01), C07D |
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Owner name: ADAMA MAKHTESHIM LTD. (IL) |
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