HRP20171776T1 - 1-supstituirani-5-fluoro-3,6-dihidro-6-imino-2(1h)-pirimidinonski derivati kao fungicidni agensi za uporabu u zaštiti bilja - Google Patents

1-supstituirani-5-fluoro-3,6-dihidro-6-imino-2(1h)-pirimidinonski derivati kao fungicidni agensi za uporabu u zaštiti bilja Download PDF

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HRP20171776T1
HRP20171776T1 HRP20171776TT HRP20171776T HRP20171776T1 HR P20171776 T1 HRP20171776 T1 HR P20171776T1 HR P20171776T T HRP20171776T T HR P20171776TT HR P20171776 T HRP20171776 T HR P20171776T HR P20171776 T1 HRP20171776 T1 HR P20171776T1
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methyl
ring system
compound
substituted
sodium
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Timothy A. Boebel
Beth Lorsbach
W. John Owen
Michael T. Sullenberger
Jeffery D. Webster
Chenglin Yao
Chris V. Galliford
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Adama Makhteshim Ltd.
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Publication of HRP20171776T1 publication Critical patent/HRP20171776T1/hr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
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  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
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  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Claims (15)

1. Spoj naznačen time, da ima formulu I: [image] u čemu R1 jest: C1-C6 alkil po izboru supstituiran s 1-3 R3; C1-C6 alkenil po izboru supstituiran s 1-3 R3; C3-C6 alkinil po izboru supstituiran s 1-3 R3; fenil ili benzil u čemu svaki od fenila ili benzila može po izboru biti supstituiran s 1-3 R4 ili s 5- ili 6-članim zasićenim ili nezasićenim prstenastim sistemom, ili s 5-6 kondenziranim prstenastim sistemom, ili s 6-6 kondenziranim prstenastim sistemom, od kojih svaki sadrži 1-3 heteroatoma i u čemu svaki prsten može po izboru biti supstituiran s 1-3 R4, -(CHR5)mOR6; -C(=O)R7; -C(=S)R7; -C(=O)OR7; -C(=S)OR7; -S(O)2R7; -(CHR5)mN(R8)R9; -C(=O)N(R8)R9; ili -C(=S)N(R8)R9; u čemu m jest cijeli broj 1-3; R2 jest: H; ili C1-C6 alkil po izboru supstituiran s R3; R3 je nezavisno halogen, C1-C6 alkil, C1-C4 haloalkil, C1-C4 alkoksi, C1-C4 haloalkoksi, C1-C4 alkiltio, C1-C4 haloalkiltio, amino, halotio, C1-C3 alkilamino, C2-C6 alkoksikarbonil, C2-C6 alkilkarbonil, C2-C6 alkilaminokarbonil, hidroksil, C3-C6 trialkilsilil, ili s 5- ili 6-članim zasićenim ili nezasićenim prstenastim sistemom ili s 5-6 kondenziranim prstenastim sistemom ili s 6-6 kondenziranim prstenastim sistemom, od kojih svaki sadrži 1-3 heteroatoma i u čemu svaki prsten može po izboru biti supstituiran s 1-3 R; R4 je nezavisno halogen, C1-C6 alkil, C1-C6 haloalkil, C1-C6 alkoksi, C1-C6 haloalkoksi, C1-C6 alkiltio, C1-C6 haloalkiltio, halotio, amino, C1-C6 alkilamino, C2-C6 dialkilamino, C2-C6 alkoksikarbonil, C1-C6 alkilsulfonil, ili C2-C6 alkilkarbonil, nitro, hidroksil ili cijano; R5 je H, C1-C6 alkil, C1-C6 alkoksi, fenil ili benzil, u čemu svaki od benzila ili fenila može po izboru biti supstituiran s 1-3 R4; R6 je H, C1-C6 alkil, C2-C6 alkenil, C3-C6 alkinil, C1-C6 haloalkil, C1-C6 alkoksialkil, C2-C6 alkilkarbonil, fenil ili benzil, gdje svaki od fenila ili benzila može po izboru biti supstituiran s 1-3 R4, ili s 5- ili 6-članim zasićenim ili nezasićenim prstenastim sistemom ili s 5-6 kondenziranim prstenastim sistemom, ili s 6-6 kondenziranim prstenastim sistemom, od kojih svaki sadrži 1-3 heteroatoma, u čemu svaki prsten može po izboru biti supstituiran s 1-3 R4, bifenil ili naftil po izboru supstituirani s 1-3 R4; R7 je H, C1-C6 alkil, C2-C6 alkenil, C3-C6 alkinil, C1-C6 haloalkil, C1-C6 alkoksialkil, fenil ili benzil, u čemu svaki od fenila ili benzila može po izboru biti supstituiran s 1-3 R4, ili s 5- ili 6-članim zasićenim ili nezasićenim prstenastim sistemom ili s 5-6 kondenziranim prstenastim sistemom ili s 6-6 kondenziranim prstenastim sistemom od kojih svaki sadrži 1-3 heteroatoma, u čemu svaki prsten može po izboru biti supstituiran s 1-3 R4, bifenil ili naftil po izboru supstituirani s 1-3 R4; R8 je H, C1-C6 alkil, C1-C6 halogenalkil, C1-C6 alkoksialkil, C2-C6 alkilkarbonil, fenil ili benzil, u čemu svaki od fenila ili benzila može po izboru biti supstituiran s 1-3 R4, ili s 5- ili 6-članim zasićenim ili nezasićenim prstenastim sistemom ili s 5-6 kondenziranim prstenastim sistemom, ili s-6-6 kondenziranim prstenastim sistemom, od kojih svaki sadrži 1-3 heteroatoma, u čemu svaki prsten može po izboru biti supstituiran s 1-3 R4; bifenil ili naftil po izboru supstituirani s 1-3 R4 ; i R9 je H, C1-C6 alkil, C1-C6 haloalkil, C1-C6 alkoksialkil, C2-C6 alkilkarbonil, ili benzil, u čemu benzil može po izboru biti supstituiran s 1-3 R4; alternativno R8 i R9 mogu se uzeti zajedno da oblikuju 5- ili 6-člani zasićeni ili nezasićeni prsten koji sadrži 1-3 heteroatoma, u čemu svaki prsten može po izboru biti supstituiran s 1-3 R4.
2. Sastav za suzbijanje gljivičnog patogena, naznačen time, da uključuje spoj iz patentnog zahtjeva 1 i fitološki prihvatljivu tvar nosioca.
3. Sastav prema patentnom zahtjevu 2, naznačen time, da gljivični patogen jest barem jedan od: krastavost jabuke (Venturia inaequalis), smeđa pjegavost lista pšenice (Septoria tritici), pjegavost lista šećerne repe (Cercospora beticola), pjegavost lista kikirikija (Cercospora arachidicola i Cercosporidium personatum) i crna sigatoka banane (Mycosphaerella fijiensis).
4. Postupak za suzbijanje i sprječavanje gljivičnog napada na biljku, naznačen time, da postupak uključuje stupnjeve: Nanošenje fungicidno učinkovite količine barem jednog od spojeva iz patentnog zahtjeva 1 na barem jednu biljku, na područje u blizini biljke, na tlo prilagođeno da pospješuje rast biljke, na korijen biljke, krošnju biljke i sjeme prilagođeno za proizvodnju biljke.
5. Pesticidna formulacija, naznačena time, da sadrži spoj prema patentnom zahtjevu 1 i drugi pesticidni spoj odabran iz skupine koja se sastoji od fungicida, insekticida, herbicida, nematocida, miticida, artropodicida, baktericida ili njihove kombinacije.
6. Pesticidna formulacija prema patentnom zahtjevu 5, naznačena time, da je težinski omjer spoja prema patentnom zahtjevu 1 u odnosu na drugi pesticidni spoj od 1:100 do 100:1.
7. Pesticidna formulacija prema patentnom zahtjevu 5, naznačena time, da drugi pesticidni spoj jest fungicidni spoj odabran iz skupine koja sadrži: 2-(tiocijanatometiltio)-benzotiazol, 2-fenilfenol, 8-hydroksikinolin sulfate, ametoktradin, amisulbrom, antimicin, Ampelomyces quisqualis, azakonazol, azoksistrobin, Bacillus subtilis, benalaksil, benomil, bentiavalikarb-izopropil, benzilaminobenzen-sulfonat (BABS) sol, bikarbonati, bifenil, bismertiazol, bitertanol, biksafen, blasticidin-S, boraks, Bordeaux smjesa, boskalid, bromukonazol, bupirimat, kalcijev polisulfid, kaptafol, kaptan, karbendazim, karboksin, karpropamid, karvon, kloroneb, klortalonil, klozolinat, Coniothyrium minitans, bakrov hidroksid, bakrov oktanoate, bakrov oksiklorid, bakrov sulfat, bakrov sulfat (tribazični), bakar (I) oksid, ciazofamid, ciflufenamid, cimoksanil, ciprokonazol, ciprodinil, dazomet, debakarb, diamonijev etilenbis-(ditiokarbamat ), diklofluanid, diklorfen, diklocimet, diklomezin, dikloran, dietofenkarb, difenokonazol, difenzokvat ion, diflumetorim, dimetomorf, dimoksistrobin, dinikonazol, dinikonazol-M, dinobuton, dinokap, difenilamin, ditianon, dodemorf, dodemorf acetat, dodin, dodin(slobodna baza), edifenfos, enestrobin, epoksikonazol, etaboksam, etoxikvin, etridiazol, famoksadon, fenamidon, fenarimol, fenbukonazol, fenfuram, fenheksamid, fenoksanil, fenpiklonil, fenpropidin, fenpropimorf,fenpirazamine,fentin, fentin acetat, fentin hidroksid, ferbam, ferimzon, fluazinam, fludioksonil, flumorf, fluopikolid, fluopiram, fluorimid, fluoksastrobin, flukvinkonazol, flusilazol, flusulfamid, flutianil, flutolanil, flutriafol, fluksapiroksad, folpet, formaldehid, fosetil, fosetil-aluminij, fuberidazol, furalaksil, furametpir, gvazatin, gvazatin acetat, GY-81, heksaklorbenzen, heksakonazol, himeksazol, imazalil, imazalil sulfat, imibenkonazol, iminoktadin, iminoktadin triacetat, iminoktadin tris(albesilat), jodokarb, ipkonazol, ipfenpirazolon, iprobenfos, iprodion, iprovalikarb, izoprotiolan, izopirazam, izotianil, laminarin, kasugamicin, kasugamicin hidroklorid hidrat, krezoksim-metil, mancopper, mankozeb, mandipropamid, maneb, meferioksam, mepanipirim, mepronil, meptildinokap, živa (II) klorid, živa (II) oksid, živa (I) klorid, metalaksil-, metalaksil-M, metam, metam-amonij, metam-kalij, metam-natrij, metkonazol, metasulfokarb, metil jodid, metil izotiocijanat, metiram, metam-inostrobin, metrafenon, mildiomicin, miclobutanil, nabam, nitrotal-izopropil, nuarimol, octilinon, ofurak, oleinska kiselina (masne kiseline), orisastrobin, oksadiksil, oksin-bakar, okspokonazol fumarat, oksikarboksin, pefurazoat, penconazol, pencycuron, penflufen, pentaklorfenol, pentaklorfenillaurat, pentiopirad, fenilživa (II) acetat, fosfonska kiselina, ftalid, pikoksistrobin, polioksin B, polioksine, polioksorim, kalijev bikarbonat, kalijevhidroksikinolinsulfat, probenazol, prokloraz, procimidon, propamokarb, propamokarb hidroklorid, propikonazol, propineb, prokvinazid, protiokonazol, piraklostrobin, pirametostrobin, piraoksistrobin, pirazofos, piribenkarb, piributikarb, pirifenoks, pirimetanil, piriofenon, pirokvilon, kvinoklamin kvinoksifen,kvintozen, Reynoutria sachalinensis ekstrakt, sedaksan, siltiofam, simekonazol, natrij 2-phenilfenoksid, natrijev bikarbonat, natrijev pentaklorfenoksid, spiroksamin, sulfur, SYP-Z071, SYP-Z048, katranska ulja, tebukonazol, tebuflokvin, teknazen, tetrakonazol, tiabendazol, tifluzamid, tiofanat-metil, tiram, tiadinil, tolklofos-metil, tolilfluanid, triadimefon, triadimenol, triazoksid, triciklazol, tridemorf, trifloksistrobin, triflumizol, triforin, tritikonazol, validamicin, valifenalat, valifenal, vinklozolin, zineb, ziram, zoksamide, Candida oleophila, Fusarium oxysporum, Gliocladium spp., Phlebiopsis gigantea, Streptomyces griseoviridis, Trichoderma spp., (RS)--N-(3,5-diklorfenil)-2-(metoksimetil)-sukcinimid, 1,2-diklorpropan, 1,3-diklor-1,1,3,3-tetrafluoraceton hidrat, 1-klor-2,4-dinitronaftalen, 1-klor-2-nitropropan, 2-(2-heptadecil-2-imidazolin-1-il)etanol, 2,3-dihidro-5-fenil-1,4-ditiin 1,1,4,4-tetraoksid, 2-metoksietilživa (II) acetat, 2-metoksietilživa(II) klorid,2-metoksietilživa (II) silikat, 3-(4-klorfenil)-5-metilrodanin, 4-(2-nitroprop-1-enil)fenil tiocianatem, ampropilfos, anilazin, azitiram, barijev polisulfid, Bayer 32394, benodanil, benkvinoks, bentaluron,benzamakril; benzamakril-izobutil, benzamorf, binapakril, bis(metilživa (II) sulfate, bis(tributiltin) oksid, butiobat, kadmij-kalcij-bakar-cinkkromatsulfat, karbamorf, CECA, klobentiazon, kloraniformetan,klorfenazol, klorkvinoks, klimbazol, ciklafuramid, cipendazol, ciprofuram, dekafentin, diklon, diklozolin,diklobutrazol, dimetirimol, dinokton, dinosulfon, dinoterbon, dipirition, ditalimfos, dodicin, drazoksolon, EBP,ESBP, etakonazol, etem, etirim, fenaminosulf, fenapanil, fenitropan, fluotrimazol, furkarbanil, furkonazol, furkonazol-cis, furmecikloks, furofanat, gliodin, griseofulvin, halakrinat, Hercules 3944, heksiltiofos, lClA0858,izopamfos, izovaledion, mebenil, mekarbinzid, metazoksolon, metfuroksam, metilživadicijandiamid, metsulfovaks, milneb, mukoklorni anhidrid, miklozolin, N-3,5-diklorfenil-sukcinimid, N-3-nitrofenilitakonimid, natamicin, N-etilživa-4-toluensulfonanilid, nikalj bis(dimetilditiokarbamat), OCH, fenilživadimetilditiokarbamat, fenilživanitrat, fosdifen, pikolinamid UK-2A i derivati od toga, protiokarb; protiokarb hidroklorid, pirakarbolid, piridinitril, piroksiklor, piroksifur, kvinacetol, kvinacetol sulfat,kvinazamid, kvinkonazol, rabenzazol, salicilanilid, SSF-109, sultropen, tekoram, tiadifluor, ticiofen, tioklorfenfim, tiofanat, tiokvinoks, tioksimid, triamifos, triarimol, triazbutil, triklamid, urbacid i zarilamid, te svaka kombinacija istih.
8. Pesticidna formulacija prema patentnom zahtjevu 5, naznačena time, da drugi pesticidni spoj jest pesticidni spoj odabran iz skupine koja sadrži: 1,2-diklorpropan, abamektin, acefat, acetamiprid, acetion, acetoprol, akrinatrin, akrilonitril, alanikarb, aldikarb, aldoksikarb, aldrin, aletrin, alosamidin, aliksikarb, alfa-cipermetrin, alfa-ekdison, alfa-endosulfan, amidition, aminokarb, amiton, amiton oksalat, amitraz, anabasin, atidation, azadirahtin, azametifos, azinfos-etil, azinfos-metil, azotoat, barijev heksafluorsilikat, bartrin, bendiokarb, benfurakarb, bensultap, beta-ciflutrin, beta-cipermetrin, bifentrin, bioaletrin, bioetanometrin, biopermetrin, bistrifluoron, boraks, borna kiselina, bromfenvinfos, bromociklen, bromo-DDT, bromofos, bromofos-etil, bufenkarb, buprofezin, butakarb, butatiofos, butokarboksim, butonat, butoksikarboksim, kadusafos, kalcijev arsenat, kalcijev polisulfid, kamfeklor, karbanolat, karbaril, karbofuran, ugljikov disulfid, uljikov tetraklorid, karbofenotion, karbosulfan, kartap, kartap hidroklorid, klorantraniliprol, klorbiciklen, klordan, klordekon, klordimeform, klordimeform hidroklorid, kloretoksifos, klorfenapir, klorfenvinfos, klorfluazuron, klormefos, kloroform, kloropikrin, klorfoksim, klorprazofos, klorpirifos, klorpirifos-metil, klortiofos, kromafenozid, cinerin I, cinerin ll, cinerini, cismetrin, kloetokarb, klosantel, klotianidin, bakar acetoarsenit, bakar arsenat, bakar naftenat, bakar oleat, kumafos, kumitoat, krotamiton, krotoksifos, krufomat, kriolit, cijanofenfos, cijanofos, cijantoat, ciantraniliprol, cikletrin, cikloprotrin, ciflutrin, cihalotrin, cipermetrin, cifenotrin, ciromazin, citioat, DDT, dekarbofuran, deltametrin, demefion, demefion-O, demefion-S, demeton, demeton-metil, demeton-0, demeton-O-metil, demeton-S, demeton-S-metil, demeton-S-metilsulfon, diafentiuron, dialifos, dijatomejska zemlja, diazinon, dikapton, diklofention, diklorvos, dikresil, dikrotofos, diciklanil, dieldrin, diflubenzuron, dilor, dimeflutrin, dimefoks,dimetan, dimetoat, dimetrin, dimetilvinfos, dimetilan, dineks, dineks-dikleksin, dinoprop, dinosam, dinotefuran, diofenolan, dioksabenzofos, dioksakarb, dioksation, disulfoton, ditikrofos, d-limonen, DNOC, DNOC-amonij, DNOC-kalij, DNOC-natrij, doramektin, ekdisteron, emamektin, emamektin benzoat, EMPC, empentrin, endosulfan, endotion, endrin, EPN, epofenonan, eprinomektin, esdepaletrin, esfenvalerat, etafos, etiofen-karb, etion, etiprol, etoat-metil, etoprofos, etil format, etil-DDD, etilendibromid, etilendiklorid, etilenoksid, etofenproks, etrimfos, EXD, famfur, fenamifos, fenazaflor, fenklorfos, fenetakarb, fen-flutrin, fenitrotion, fenobukarb, fenoksakrim, fenoksikarb, fenpiritrin, fenpropatrin, fensulfotion, fention, fention-etil, fenvalerat, fipronil, flonikamid, flubendiamid, flukofuron, flucikloksuron, flucitrinat, flufenerim, flufenoksuron, flufenproks, flufiprol, fluvalinat, fonofos, formetanat, formetanathidroklorid, formotion, formparanat, formparanathidroklorid, fosmetilan, fospirat, fostietan, furatiokarb, furetrin, gama-cihalotrin, gamma-HCH, halfenproks, halofenozid, HCH, HEOD, heptaklor, heptenofos, heterofos, heksaflumuron, HHDN, hidrametinon, cijanovodik , hidropren, hikvinkarb, imidakloprid, irniprotrin, indoksakarb, jodometan, IPSP, izazofos, izobenzan, izokarbofos, izodrin, izofenfos, izofenfos-metil, izoprokarb, izoprotiolan, izotioat, izoksation, ivermektin, jasmolin l, jasmolin il, jodfenfos, juvenilni hormon I, juvenilni hormon ll, juvenilni hormone lll, kelevan, kinopren, lambda-cihalotrin, olovni arsenate, lepimektin, leptofos, lindan, lirimfos, lufenuron, litidation, malation, malonoben, mazidoks, mekarbam, mekarfon, menazon, meperflutrin, mefosfolan, živa(I) klorid, mesulfenfos, metaflumizon, metakrifos, metamidofos, metidation, metiokarb, metokrotofos, metomil, metopren, metoksiklor, metoksifenozid, metilbromid, metilizotiocijanat, metilkloroform, metilenklorid, metoflutrin, metolkarb, metoksadiazon, mevinfos, meksakarbat, milbemektin, milbemicinoksim, mipafoks, mireks, molosultap, monokrotofos, monomehipo, monosultap, morfotion, moksidektin, naftalofos, naled, naftalen, nikotin, nifluridid, nitenpiram, nitiazin, nitrilakarb, novaluron, noviflumuron, ometoat, oksamil, oksidemeton-metil, oksideprofos, oksidisulfoton, para-diklorbenzen, paration, paration-metil, penfluoron, pentaklorfenol, permetrin, fenkapton, fenotrin, fentoat, forat, fosalon, fosfolan, fosmet, fosniklor, fosfamidon, fosfin, phoxim, foksim-metil, pirimetafos, pirimikarb, pirimifos-etil, pirimifos-metil, kalijev arsenit, kalijev tiocijanat, pp’-DDT, pralletrin, prekocen l, prekocen ll, prekocen Ill, primidofos, profenofos, profluralin, promacil, promekarb, propafos, propetamfos, propoksur, protidation, protiofos, protoate, protrifenbut, piraklofos, pirafluprol, pirazofos, piresmetrin, piretrin l, piretrin ll, piretrini, piridaben, piridalil, piridafention, piriflukvinazon, pirimidifen, pirimitat, piriprol, piriproksifen, kvasija, kvinalfos, kvinalfos-metil, kvinotion, rafoksanid, resmetrin, rotenon, riania, sabadila, schradan, selamektin, silafluofen, silika gel, natrijev arsenit, natrijev fluorid, natijev heksafluorsilikat, natrijev tiocijanat, sofamid, spinetoram, spinosad, spiromesifen, spirotetramat, sulkofuron, sulkofuron-natrij, sulfluramid, sulfotep, sulfoksaflor, sulfuril fluorid, sulprofos, tau-fluvalinat, tazimkarb, TDE, tebufenozid, tebufenpirad, tebupirimfos, teflubenzuron, teflutrin, temefos, TEPP, teraletrin, terbufos, tetrakloretan, tetraklorvinfos, tetrametrin, tetrametilflutrin, teta-cipermetrin, tiakloprid, tiametoksam, tikrofos, tiokarboksim, tiociklam, tiociklamoksalat, tiodikarb, tiofanoks, tiometon, tiosultap, tiosultap-dinatrij, tiosultap-mononatrij, turingiensin, tolfenpirad, tralometrin, transflutrin, transpermetrin, triaratene, triazamat, triazofos, triklorfon, triklormetafos-3, trikloronat, trifenofos, triflumuron, trimetakarb, tripren, vamidotion, vaniliprol, XMC, ksililkarb, zeta-cipermetrin, zolaprofos i bilo koja njihova kombinacija.
9. Pesticidna formulacija prema patentnom zahtjevu 5, naznačena time, da drugi pesticidni spoj jest herbicidni spoj odabran iz skupine koja sadrži: 4-CPA; 4-CPB; 4-CPP; 2,4-D; 3,4-DA; 2,4-DB; 3,4-DB; 2,4-DEB; 2,4-DEP; 3,4-DP; 2,3,6-TBA; 2,4,5-T; 2,4,5-TB; acetoklor, acifluorfen, aklonifen, akrolein, alaklor, alidoklor, aloksiklim, alil alkohol, alorak, ametridion, ametrin, amibuzin, amikarbazon, amidosulfuron, aminociklopiraklor, aminopiralid, amiprofos-metil, amitrol, amonijev sulfamat, anilofos, anisuron, asulam, atraton, atrazin, azafenidin, azimsulfuron, aziprotrin, barban, BCPC, beflubutamid, benazolin, benkarbazon, benfluralin, benfuresat, bensulfuron, bensulid, bentazon, benzadoks, benzfendizon, benzipram, benzobiciklon, benzofenap, benzofluor, benzoilprop,.benztiazuron, biciklopiron, bifenoks, bilanafos, bispiribak, boraks, bromacil, bromobonil, bromobutid, bromofenoksim, bromoksinil, brompirazon, butaklor, butafenacil, butamifos, butenaklor, butidazol, butiuron, butralin, butroksidim, buturon, butilat, kakodilna kiselina, kafenstrol, kalcijev klorat, kalcijev cijanamid, kambendiklor, karbasulam, karbetamid, karboksazol, klorprokarb, karfentrazon, CDEA, CEPC, klometoksifen, kloramben, kloranokril, klorazifop, klorazin, klorbromuron, klorbufam, kloreturon, klorfenak, klorfenprop, klorflurazol, klorflurenol, kloridazon, klorimuron, klornitrofen, kloropon, klorotoluron, kloroksuron, kloroksinil, klorprofam, klorsulfuron, klortal, klortiamid, cinidon-etil, cinmetilin, cinoslfuron, cisanilid, kletodim, kliodinat, klodinafop, klofop, klomazon, klomeprop, kloprop, kloproksidim, klopiralid, kloransulam, CMA, bakrov sulfat, CPMF, CPPC, kredazin, krezol, kumiluron, cianatrin, cianazin, cikloat, ciklosulfamuron, cikloksidim, cikluron, cihalofop, cyperquat, ciprazin, ciprazol, cipromid, daimuron, dalapon, dazomet, delaklor, desmedifam, desmetrin, dialat, dicamba, diklobenil, dikloralurea, diklomat, diklorprop, diklorprop-P, diklofop, diklosulam, diethamquat, dietatil, difenopenten, difenoksuron, difenzoquat, diflufenikan, diflufenzopir,dimefuron, dimepiperat, dimetaklor, dimetametrin, dimetenamid, dimetenamid-P, dimeksano, dimidazon, dinitramin, dinofenat, dinoprop, dinosam, dinoseb, dinoterb, difenamid, dipropetrin, dikvat, disul, ditiopir, diuron, DMPA, DNOC, DSMA, EBEP, eglinazin, endotal, epronaz, EPTC, erbon, esprokarb, etalfluralin, etamet-sulfuron, etidimuron, etiolat, etofumesat, etoksifen, etoksisulfuron, etinofen, etnipromid, etobenzanid, EXD, fenasulam, fenoprop, fenoksaprop, fenoksaprop-P, fenoksasulfon, fenterakol, fentiaprop, fentrazamid, fenuron, željezo(II) sulfat, flamprop, flamprop-M, flazasulfuron, florasulam, fluazifop, fluazifop-P, fluazolat, flukarbazon, flucetosulfuron, flukloralin, flufenacet. flufenikan, flufenpir, flumetsulam, flumezin, flumiklorak, flumioksazin, flumipropin, fluomeluron, fluordifen, fluorglikofen, fluoromidin, fluornitrofen, fluotiuron, flupoksam, flupropacil, flupropanat, flupirsulfuron, fluridon, fluorokloridon, fluoroksipir, flurtamon, flutiacet, fomesafen, foramsulfuron, fosamin, furioksifen, glufosinat, glufosinat-P, glifosat, halosafen, halosulfuron, haloksidin, haloksifop, haloksifop-P, heksakloraceton, heksaflurat, heksazinon, imazametabenz, imazamoks, imazapik, imazapir, imazakvin, imazetapir, imazosulfuron, indanofan, inklaziflam, jodobonil, jodomelhan, jodosulfuron, joksinil, ipazin,.ipfenkarbazon, iprimidam, izokarbamid, izocil, izometiozin, izonoruron, izopolinat, izopropalin, izoproturon, izouron, izoksaben, izoksaklortol, izoksaflutol, izoksapirifop, karbutilat, ketospiradoks, laktofen, lenacil, linuron, MAA, MAMA, MCPA, MCPA-tioetil, MCPB, mekoprop, mekoprop-P, medinoterb, mefenacet, mefluidid, mesoprazin, mesosulfuron, mesotrion, metam, metamifop, melamitron. metazaklor, metazosulfuron, metflurazon, metabenztiazuron, metapropalin, metazol, metiobenkarb, metiozolin, metiuron, metometon, metoprotrin, metil bromid, metilizotiocijanat, metildimron, metobenzuron, metobromuron, metolaklor, metosulam, metoksuron, metribuzin, metsulfuron, molinat, monalid, monisouron, monokloroctena kiselina, monolinuron, monuron, morfamkvat, MSMA, naproanilid, napropamid, naptalam, neburon, nikosulfuron, nipiraklofen, nitralin, nitrofen, nitrofluorfen, norflurazon, noruron, OCH, orbenkarb, orto diklorbenzen, ortosulfamuron, orizalin, oksadiargil, oksadiazon, oksapirazon, oksasulfuron, oksaziciklomefon, oksifluorfen, parafluoron, parakvat, pebulat, pelargonska kiselina, pendimetalin, penoksulam, pentaklorofenol, pentanoklor, pentoksazon, perfluidon, petoksamid,fenizofam, fenmedifam, fenmedifam-etil, fenobenzuron, fenilživa acetat, pikloram, pikolinafen, pinoksaden, piperofos, kalijev arsenit, kalijev azid, kalijev cijanat, pretilaklor, primisulfuron, prociazin, prodiamin, profluazol, profluralin, profoksidim, proglinazin, prometon, prometrin, propaklor, propanil, propakvizafop, propazin, profam, propizoklor, propoksikarbazon, propirisulfuron, propizamid, prosulfalin, prosulfokarb, prosulfuron, proksan, prinaklor, pidanon, piraklonil, piraflufen, pirasulfotol, pirazolinat, pirazosulfuron, pirazoksifen, piribenzoksim, piributikarb, pyriclor, piridafol, piridat, piriftalid, piriminobak, pirimisulfan, piritiobak, piroksasulfon, pirokssulam, quinclorac, quinmerac, quinoclamin, quinonamid, quizalofop, quizalofop-P, rodetanil, rimsulfuron, saflufenacil, S-metolaklor, sebutilazin, sekbumeton, setoksidim, siduron, simazin, simeton, simetrin, SMA, natrijev arsenit, natrijev azid, natrijev klorat, sulkotrion, sulfalat, sulfentrazon, sulfometuron, sulfosulfuron, sulfatna kiselina, sulglikapin, swep, TCA, tebutam, tebutiuron, tefuriltrion, tembotrion,tepraloksidim, terbacil, terbukarb, terbuklor, terbumeton, terbutilazin, terbutrin, tetrafluoron, tenilklor, tiazafluoron, tiazopir, tidiazimin, tidiazuron, tienkarbazon-metil, tifensulfuron, tiobenkarb, tiokarbazil, tioclorim, topramezon, tralkoksidim, triafamon, trialat, triasulfuron, triaziflam, tribenuron, trikamba, triklopir, tridifan, trietazin, trifloksisulfuron, trifluralin, triflusulfuron, trifop, trifopsim, trihidroksitriazin, trimeturon, tripropindan, tritac, tritosulfuron, vernolat i xylachlor.
10. Sastav prema patentnom zahtjevu 2, naznačen time, da koncentracija spoja jest od 0,1 do 1000 ppm.
11. Sastav prema patentnom zahtjevu 2, naznačen time, da koncentracija spoja jest od 1 do 500 ppm.
12. Postupak prema patentnom zahtjevu 4, naznačen time, da fungicidno učinkovita količina jest od 0,01 do 0,45 grama po kvadratnom metru.
13. Spoj prema patentnom zahtjevu 1, naznačen time, da spoj formule I jest 5-flor-4-imino-3-metil-3,4-dihidropirimidin-2(1H)-on.
14. Spoj prema patentnom zahtjevu 1, naznačen time, da spoj formule I jest 5-flor-4-imino-3-(tiofen-2-ilmetil)-3,4-dihidropirimidin-2(1H)-on
15. Spoj prema patentnom zahtjevu 1, naznačen time, da spoj formule I jest 5-flor-4-imino-3-(trideuteriometil)-1H-pirimidin-2-on.
HRP20171776TT 2011-08-17 2017-11-16 1-supstituirani-5-fluoro-3,6-dihidro-6-imino-2(1h)-pirimidinonski derivati kao fungicidni agensi za uporabu u zaštiti bilja HRP20171776T1 (hr)

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