RS56609B1 - 1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji bilja - Google Patents
1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji biljaInfo
- Publication number
- RS56609B1 RS56609B1 RS20171186A RSP20171186A RS56609B1 RS 56609 B1 RS56609 B1 RS 56609B1 RS 20171186 A RS20171186 A RS 20171186A RS P20171186 A RSP20171186 A RS P20171186A RS 56609 B1 RS56609 B1 RS 56609B1
- Authority
- RS
- Serbia
- Prior art keywords
- imino
- dihydro
- fluoro
- substituted
- plant protection
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161524506P | 2011-08-17 | 2011-08-17 | |
| PCT/US2012/050930 WO2013025795A1 (en) | 2011-08-17 | 2012-08-15 | 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives |
| EP12824035.5A EP2775842B1 (en) | 2011-08-17 | 2012-08-15 | 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1H)-pyrimidinone derivatives as fungicidal agents for use in plant protection |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RS56609B1 true RS56609B1 (sr) | 2018-02-28 |
Family
ID=47713076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RS20171186A RS56609B1 (sr) | 2011-08-17 | 2012-08-15 | 1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji bilja |
Country Status (31)
| Country | Link |
|---|---|
| US (1) | US8658660B2 (sr) |
| EP (1) | EP2775842B1 (sr) |
| JP (3) | JP6128658B2 (sr) |
| KR (1) | KR102012992B1 (sr) |
| CN (2) | CN103874413B (sr) |
| AR (1) | AR087549A1 (sr) |
| BR (1) | BR112014003587B1 (sr) |
| CA (1) | CA2844497C (sr) |
| CL (1) | CL2014000352A1 (sr) |
| CO (1) | CO6910204A2 (sr) |
| CR (1) | CR20140058A (sr) |
| DK (1) | DK2775842T3 (sr) |
| EC (1) | ECSP14013251A (sr) |
| ES (1) | ES2646725T3 (sr) |
| GT (1) | GT201400023A (sr) |
| HK (1) | HK1199177A1 (sr) |
| HR (1) | HRP20171776T1 (sr) |
| HU (1) | HUE035248T2 (sr) |
| IL (1) | IL230981A (sr) |
| LT (1) | LT2775842T (sr) |
| ME (1) | ME02924B (sr) |
| MX (1) | MX354021B (sr) |
| NO (1) | NO2874589T3 (sr) |
| PL (1) | PL2775842T3 (sr) |
| PT (1) | PT2775842T (sr) |
| RS (1) | RS56609B1 (sr) |
| RU (1) | RU2613451C2 (sr) |
| SI (1) | SI2775842T1 (sr) |
| UA (1) | UA113062C2 (sr) |
| WO (1) | WO2013025795A1 (sr) |
| ZA (1) | ZA201400875B (sr) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6128658B2 (ja) * | 2011-08-17 | 2017-05-17 | アダマ・マクテシム・リミテッド | ５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体 |
| AU2013370490B2 (en) | 2012-12-28 | 2018-05-10 | Adama Makhteshim Ltd. | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives |
| CN110003118A (zh) | 2012-12-28 | 2019-07-12 | 阿达玛马克西姆股份有限公司 | 制备羧酸酯衍生物的方法 |
| NZ708981A (en) | 2012-12-31 | 2020-01-31 | Adama Makhteshim Ltd | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides |
| CN103819412B (zh) * | 2013-12-11 | 2016-02-03 | 浙江先锋科技股份有限公司 | 一种5-氟胞嘧啶的制备方法 |
| BR112016015158A2 (pt) | 2013-12-31 | 2017-08-08 | Adama Makhteshim Ltd | Misturas fungicidas sinergísticas para controle de fungos em cereais |
| CN106068268A (zh) * | 2013-12-31 | 2016-11-02 | 阿达玛马克西姆股份有限公司 | 5‑氟‑4‑亚氨基‑3‑（烷基/取代烷基）‑1‑（芳基磺酰基）‑3,4‑二氢嘧啶‑2（1h）‑酮及其制备方法 |
| MA41272A (fr) * | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
| TWI774761B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
| TWI801380B (zh) * | 2017-05-02 | 2023-05-11 | 美商科迪華農業科技有限責任公司 | 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途 |
| TWI801381B (zh) * | 2017-05-02 | 2023-05-11 | 美商科迪華農業科技有限責任公司 | 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途 |
| TW201842851A (zh) * | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
| TWI774762B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途 |
| TWI774760B (zh) * | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於蔬菜中的真菌防治之協同性混合物 |
| CA3069619A1 (en) | 2017-07-17 | 2019-02-28 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| CN109053553A (zh) * | 2018-10-16 | 2018-12-21 | 山东省农药科学研究院 | 杀虫剂氟啶虫胺腈中间体3-[1-(甲硫基)乙基]-6(三氟甲基)吡啶的合成方法 |
| WO2021031431A1 (en) | 2019-08-22 | 2021-02-25 | Fujian Yongjing Technology Co., Ltd | Process for preparing fluorobenzene by direct fluorination |
| WO2021181274A1 (en) * | 2020-03-09 | 2021-09-16 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| WO2023042126A1 (en) * | 2021-09-15 | 2023-03-23 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3635977A (en) * | 1969-11-03 | 1972-01-18 | American Cyanamid Co | Certain 6-trifluoromethylcytosines and thiocytosines their synthesis and their use in the synthesis of uracisls and thiouracil |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (sr) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| EP0139613A1 (de) | 1983-08-29 | 1985-05-02 | Ciba-Geigy Ag | N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| ES2057172T3 (es) | 1988-03-09 | 1994-10-16 | Ciba Geigy Ag | Agente para la proteccion de plantas contra enfermedades. |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤 |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| AU6478396A (en) | 1995-07-05 | 1997-02-05 | E.I. Du Pont De Nemours And Company | Fungicidal pyrimidinones |
| DE69712331T2 (de) | 1996-03-11 | 2002-11-28 | Syngenta Participations Ag | Pyrimidin-4-on derivate als pestizidesmittel |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) * | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| WO2003018051A1 (en) | 2001-08-27 | 2003-03-06 | Vic Jira | Anti-fungal composition |
| EA009517B1 (ru) * | 2003-06-27 | 2008-02-28 | Байер Кропсайенс Аг | Пиразолопиримидины |
| WO2005095419A1 (ja) | 2004-04-01 | 2005-10-13 | Takeda Pharmaceutial Company Limited | チアゾロピリミジン誘導体 |
| TWI402034B (zh) | 2005-07-28 | 2013-07-21 | Dow Agrosciences Llc | 具有被層狀液晶覆膜包覆之油球之水包油乳化劑之農用組成物 |
| CA2629295A1 (en) * | 2005-11-22 | 2007-05-31 | Ishihara Sangyo Kaisha, Ltd. | Germicide composition for agricultural and gardening applications and method for controlling plant disease |
| US20080004253A1 (en) | 2006-06-30 | 2008-01-03 | Bryan James Branstetter | Thiazolopyrimidine modulators of TRPV1 |
| ES2549172T3 (es) * | 2008-01-22 | 2015-10-23 | Dow Agrosciences, Llc | Derivados de 5-fluoropirimidina como fungicidas |
| RU2536492C2 (ru) | 2008-08-01 | 2014-12-27 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Применение 5-фторцитозина в качестве фунгицида |
| EP2326327B1 (en) * | 2008-09-17 | 2016-03-23 | SRI International | Analogs of indole-3-carbinol and their use as agents against infection |
| ME02254B (me) | 2009-01-23 | 2015-12-31 | Euro Celtique Sa | Derivati hidroksamske kiseline |
| JP5784603B2 (ja) * | 2009-08-07 | 2015-09-24 | ダウ アグロサイエンシィズ エルエルシー | Ｎ１−スルホニル−５−フルオロピリミジノン誘導体 |
| UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| UA112284C2 (uk) | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| UA106246C2 (ru) * | 2009-10-07 | 2014-08-11 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Синергическая фунгицидная композиция, которая содержит 5-фторцитозин для борьбы с грибковыми болезнями зерновых культур |
| JP6128658B2 (ja) * | 2011-08-17 | 2017-05-17 | アダマ・マクテシム・リミテッド | ５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体 |
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2012
- 2012-08-15 JP JP2014526166A patent/JP6128658B2/ja active Active
- 2012-08-15 ME MEP-2017-274A patent/ME02924B/me unknown
- 2012-08-15 ES ES12824035.5T patent/ES2646725T3/es active Active
- 2012-08-15 SI SI201231158T patent/SI2775842T1/en unknown
- 2012-08-15 CN CN201280049656.1A patent/CN103874413B/zh active Active
- 2012-08-15 EP EP12824035.5A patent/EP2775842B1/en active Active
- 2012-08-15 PL PL12824035T patent/PL2775842T3/pl unknown
- 2012-08-15 WO PCT/US2012/050930 patent/WO2013025795A1/en active Application Filing
- 2012-08-15 UA UAA201402588A patent/UA113062C2/uk unknown
- 2012-08-15 RS RS20171186A patent/RS56609B1/sr unknown
- 2012-08-15 MX MX2014001885A patent/MX354021B/es active IP Right Grant
- 2012-08-15 KR KR1020147006630A patent/KR102012992B1/ko active IP Right Grant
- 2012-08-15 CA CA2844497A patent/CA2844497C/en active Active
- 2012-08-15 BR BR112014003587-3A patent/BR112014003587B1/pt active IP Right Grant
- 2012-08-15 LT LTEP12824035.5T patent/LT2775842T/lt unknown
- 2012-08-15 PT PT128240355T patent/PT2775842T/pt unknown
- 2012-08-15 CN CN201710076214.0A patent/CN106977462B/zh active Active
- 2012-08-15 DK DK12824035.5T patent/DK2775842T3/en active
- 2012-08-15 AR ARP120102991A patent/AR087549A1/es active IP Right Grant
- 2012-08-15 US US13/586,450 patent/US8658660B2/en active Active
- 2012-08-15 HU HUE12824035A patent/HUE035248T2/en unknown
- 2012-08-15 RU RU2014110049A patent/RU2613451C2/ru active
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2013
- 2013-07-19 NO NO13745256A patent/NO2874589T3/no unknown
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2014
- 2014-01-30 CR CR20140058A patent/CR20140058A/es unknown
- 2014-02-05 ZA ZA2014/00875A patent/ZA201400875B/en unknown
- 2014-02-12 CL CL2014000352A patent/CL2014000352A1/es unknown
- 2014-02-13 IL IL230981A patent/IL230981A/en active IP Right Grant
- 2014-02-14 GT GT201400023A patent/GT201400023A/es unknown
- 2014-03-14 CO CO14055677A patent/CO6910204A2/es unknown
- 2014-03-17 EC ECSP14013251 patent/ECSP14013251A/es unknown
- 2014-12-18 HK HK14112698.4A patent/HK1199177A1/xx unknown
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2017
- 2017-04-07 JP JP2017076823A patent/JP2017125060A/ja not_active Withdrawn
- 2017-11-16 HR HRP20171776TT patent/HRP20171776T1/hr unknown
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2018
- 2018-12-21 JP JP2018239307A patent/JP6901462B2/ja active Active
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