PH30894A - 1,5-Benzodiazepine derivative. - Google Patents
1,5-Benzodiazepine derivative.Info
- Publication number
- PH30894A PH30894A PH45583A PH45583A PH30894A PH 30894 A PH30894 A PH 30894A PH 45583 A PH45583 A PH 45583A PH 45583 A PH45583 A PH 45583A PH 30894 A PH30894 A PH 30894A
- Authority
- PH
- Philippines
- Prior art keywords
- benzodiazepine derivative
- benzodiazepine
- derivative
- Prior art date
Links
- ZVAPWJGRRUHKGP-UHFFFAOYSA-N 1h-1,5-benzodiazepine Chemical class N1C=CC=NC2=CC=CC=C12 ZVAPWJGRRUHKGP-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/12—1,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB929201180A GB9201180D0 (en) | 1992-01-21 | 1992-01-21 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH30894A true PH30894A (en) | 1997-12-23 |
Family
ID=10708914
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH45583A PH30894A (en) | 1992-01-21 | 1993-01-20 | 1,5-Benzodiazepine derivative. |
Country Status (29)
| Country | Link |
|---|---|
| US (2) | US5580895A (cs) |
| JP (1) | JP3253723B2 (cs) |
| KR (1) | KR100263625B1 (cs) |
| CN (1) | CN1049217C (cs) |
| AP (1) | AP369A (cs) |
| AU (2) | AU3450193A (cs) |
| BG (1) | BG61876B1 (cs) |
| CA (1) | CA2087672C (cs) |
| CZ (1) | CZ283950B6 (cs) |
| FI (1) | FI111632B (cs) |
| GB (1) | GB9201180D0 (cs) |
| GE (1) | GEP20001968B (cs) |
| HU (2) | HU221297B1 (cs) |
| IL (1) | IL104447A (cs) |
| IS (1) | IS3970A (cs) |
| MX (1) | MX9300261A (cs) |
| MY (1) | MY131307A (cs) |
| NO (1) | NO305952B1 (cs) |
| NZ (1) | NZ245715A (cs) |
| OA (1) | OA09964A (cs) |
| PH (1) | PH30894A (cs) |
| PL (1) | PL175340B1 (cs) |
| RO (1) | RO114128B1 (cs) |
| RU (1) | RU2124009C1 (cs) |
| SK (1) | SK280173B6 (cs) |
| TW (1) | TW226013B (cs) |
| UA (1) | UA29416C2 (cs) |
| WO (1) | WO1993014074A1 (cs) |
| ZA (1) | ZA93375B (cs) |
Families Citing this family (48)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9225492D0 (en) * | 1992-12-05 | 1993-01-27 | Glaxo Group Ltd | Amine derivatives |
| GB9307833D0 (en) * | 1993-04-15 | 1993-06-02 | Glaxo Inc | Modulators of cholecystokinin and gastrin |
| FI954852A0 (fi) * | 1993-04-15 | 1995-10-12 | Glaxo Wellcome Inc | 1,5-bentsodiatsepiinijohdannaisia, joilla on CCK- ja/tai gastriiniantagonistinen aktiivisuus |
| GB9308421D0 (en) * | 1993-04-23 | 1993-06-09 | Glaxo Spa | Chemical compounds |
| GB9308431D0 (en) * | 1993-04-23 | 1993-06-09 | Glaxo Spa | Chemical compounds |
| GB9314977D0 (en) * | 1993-07-20 | 1993-09-01 | Glaxo Spa | Chemical compounds |
| GB9315018D0 (en) * | 1993-07-20 | 1993-09-01 | Glaxo Spa | Chemical compounds |
| GB2280182A (en) * | 1993-07-20 | 1995-01-25 | Glaxo Spa | Benzodiazepine derivatives |
| GB9314981D0 (en) * | 1993-07-20 | 1993-09-01 | Glaxo Spa | Chemical compounds |
| US5739129A (en) * | 1994-04-14 | 1998-04-14 | Glaxo Wellcome Inc. | CCK or gastrin modulating 5-heterocyclic-1, 5 benzodiazepines |
| AU697349B2 (en) * | 1994-04-14 | 1998-10-01 | Glaxo Wellcome Inc. | CCK or gastrin modulating 5-heterocyclic-1,5-benzodiazepines |
| PE27497A1 (es) * | 1994-04-15 | 1997-08-07 | Glaxo Inc | Derivados de 1,5 benzodiazepina |
| US5780464A (en) * | 1994-10-14 | 1998-07-14 | Glaxo Wellcome Inc. | Enteric coated compositions of 1,5-benzodiazepine derivatives having CCK antagonistic or agonistic activity |
| GB9420748D0 (en) * | 1994-10-14 | 1994-11-30 | Glaxo Inc | 1,5 benzodiazepine derivatives |
| US5750353A (en) * | 1995-12-11 | 1998-05-12 | New England Medical Center Hospitals, Inc. | Assay for non-peptide agonists to peptide hormone receptors |
| JP4442930B2 (ja) | 1995-12-11 | 2010-03-31 | タフツ メディカル センター インコーポレイテッド | ペプチドホルモンレセプターリガンドに関するアッセイ法およびその使用 |
| WO1998025911A1 (fr) * | 1996-12-10 | 1998-06-18 | Zeria Pharmaceutical Co., Ltd. | Derives de 1,5-benzodiazepine |
| RU2321583C2 (ru) * | 2001-01-22 | 2008-04-10 | Мемори Фармасьютиклз Корпорейшн | Применение производных анилина в качестве ингибиторов фосфодиэстеразы 4 |
| WO2004064730A2 (en) * | 2003-01-14 | 2004-08-05 | Cytokinetics, Inc. | Compounds, compositions and methods |
| GB0307918D0 (en) * | 2003-04-05 | 2003-05-14 | Astrazeneca Ab | Therapeutic use |
| CA2545513C (en) * | 2003-11-18 | 2013-01-08 | Boehringer Ingelheim International Gmbh | Solid pharmaceutical preparation form |
| CA2570999C (en) | 2004-06-17 | 2014-01-07 | Cytokinetics, Inc. | Compounds, compositions and methods |
| US7538223B2 (en) | 2005-08-04 | 2009-05-26 | Cytokinetics, Inc. | Compounds, compositions and methods |
| US7825120B2 (en) | 2005-12-15 | 2010-11-02 | Cytokinetics, Inc. | Certain substituted ((piperazin-1-ylmethyl)benzyl)ureas |
| JP5301284B2 (ja) | 2005-12-15 | 2013-09-25 | サイトキネティクス・インコーポレーテッド | 特定の化学物質、組成物および方法 |
| EP1959962A2 (en) | 2005-12-16 | 2008-08-27 | Cytokinetics, Inc. | Certain chemical entities, compositions, and methods |
| US7989455B2 (en) | 2005-12-19 | 2011-08-02 | Cytokinetics, Inc. | Compounds, compositions and methods |
| CU20090172A7 (es) | 2009-10-09 | 2011-10-05 | Ct De Investigación Y Desarrollo De Medicamentos | Sistemas tricíclicos y tetracíclicos con actividad sobre el sistema nervioso central y vascular |
| US9725490B2 (en) | 2011-07-29 | 2017-08-08 | Tokushima University | ERAP1-derived peptide and use thereof |
| CN103435562B (zh) * | 2013-08-26 | 2016-02-24 | 华东理工大学 | 6-取代苯并二氮卓-2,4-二酮类化合物及其用途 |
| PT3324977T (pt) | 2015-07-22 | 2022-10-14 | Enanta Pharm Inc | Derivados de benzodiazepina como inibidores de vsr |
| EP3402799B1 (en) | 2016-01-15 | 2022-05-04 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as rsv inhibitors |
| CA3065368A1 (en) | 2017-02-16 | 2018-08-23 | Enanta Pharmaceuticals, Inc. | Processes for the preparation of benzodiazepine derivatives |
| WO2018226801A1 (en) * | 2017-06-07 | 2018-12-13 | Enanta Pharmaceuticals, Inc. | Aryldiazepine derivatives as rsv inhibitors |
| WO2019006291A1 (en) | 2017-06-30 | 2019-01-03 | Enanta Pharmaceuticals, Inc. | HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS |
| WO2019006295A1 (en) | 2017-06-30 | 2019-01-03 | Enanta Pharmaceuticals, Inc. | HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS |
| EP3687543B1 (en) | 2017-09-29 | 2024-03-20 | Enanta Pharmaceuticals, Inc. | Combinations of pharmaceutical agents as rsv inhibitors |
| US10647711B2 (en) | 2017-11-13 | 2020-05-12 | Enanta Pharmaceuticals, Inc. | Azepin-2-one derivatives as RSV inhibitors |
| US10975094B2 (en) | 2018-04-11 | 2021-04-13 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as RSV inhibitors |
| EP3889264A4 (en) | 2018-11-30 | 2022-10-12 | Tokushima University | Therapeutic agent for breast caner comprising big3-phb2 interaction-inhibiting peptide derived from phb2 |
| CN113710276B (zh) | 2019-03-18 | 2024-03-29 | 英安塔制药有限公司 | 苯二氮䓬衍生物作为rsv抑制剂 |
| US11179400B2 (en) | 2019-04-09 | 2021-11-23 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as RSV inhibitors |
| US11505558B1 (en) | 2019-10-04 | 2022-11-22 | Enanta Pharmaceuticals, Inc. | Antiviral heterocyclic compounds |
| UY39032A (es) | 2020-01-24 | 2021-07-30 | Enanta Pharm Inc | Compuestos heterocíclicos como agentes antivirales |
| US11534439B2 (en) | 2020-07-07 | 2022-12-27 | Enanta Pharmaceuticals, Inc. | Dihydroquinoxaline and dihydropyridopyrazine derivatives as RSV inhibitors |
| US11945824B2 (en) | 2020-10-19 | 2024-04-02 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as anti-viral agents |
| AR129003A1 (es) | 2022-04-07 | 2024-07-03 | Enanta Pharm Inc | Compuestos heterocíclicos antivirales |
| US12162857B2 (en) | 2022-04-27 | 2024-12-10 | Enanta Pharmaceuticals, Inc. | Antiviral compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3984398A (en) * | 1966-12-14 | 1976-10-05 | Roussel-Uclaf | 1,5-Benzodiazepine-2,4-diones |
| US4207228A (en) * | 1977-09-21 | 1980-06-10 | The B. F. Goodrich Company | UV-Light-stabilized compositions containing substituted 1,5-diazacycloalkanes, novel compounds and synthesis thereof |
| JPS60158190A (ja) * | 1984-01-30 | 1985-08-19 | Eisai Co Ltd | ヒダントイン誘導体およびその製法ならびにそれを含有する医薬 |
| US4647561A (en) * | 1985-08-05 | 1987-03-03 | E. R. Squibb & Sons, Inc. | 1,5-benzodiazepine compounds |
| FR2641280B1 (fr) * | 1988-12-29 | 1994-01-21 | Roussel Uclaf | Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments |
-
1992
- 1992-01-21 GB GB929201180A patent/GB9201180D0/en active Pending
- 1992-01-21 GE GEAP19922651A patent/GEP20001968B/en unknown
-
1993
- 1993-01-15 US US08/256,359 patent/US5580895A/en not_active Expired - Fee Related
- 1993-01-19 UA UA94005364A patent/UA29416C2/uk unknown
- 1993-01-19 CZ CZ941736A patent/CZ283950B6/cs not_active IP Right Cessation
- 1993-01-19 RO RO94-01216A patent/RO114128B1/ro unknown
- 1993-01-19 WO PCT/EP1993/000098 patent/WO1993014074A1/en active IP Right Grant
- 1993-01-19 PL PL93304684A patent/PL175340B1/pl unknown
- 1993-01-19 SK SK864-94A patent/SK280173B6/sk unknown
- 1993-01-19 KR KR1019940702491A patent/KR100263625B1/ko not_active Expired - Fee Related
- 1993-01-19 HU HU9402150A patent/HU221297B1/hu not_active IP Right Cessation
- 1993-01-19 AU AU34501/93A patent/AU3450193A/en not_active Abandoned
- 1993-01-19 RU RU94037768A patent/RU2124009C1/ru active
- 1993-01-20 NZ NZ245715A patent/NZ245715A/en unknown
- 1993-01-20 IL IL104447A patent/IL104447A/en not_active IP Right Cessation
- 1993-01-20 IS IS3970A patent/IS3970A/is unknown
- 1993-01-20 CA CA002087672A patent/CA2087672C/en not_active Expired - Fee Related
- 1993-01-20 AU AU31935/93A patent/AU661749B2/en not_active Ceased
- 1993-01-20 AP APAP/P/1993/000478A patent/AP369A/en active
- 1993-01-20 PH PH45583A patent/PH30894A/en unknown
- 1993-01-20 MY MYPI93000093A patent/MY131307A/en unknown
- 1993-01-20 MX MX9300261A patent/MX9300261A/es not_active IP Right Cessation
- 1993-01-20 ZA ZA93375A patent/ZA93375B/xx unknown
- 1993-01-20 JP JP02483193A patent/JP3253723B2/ja not_active Expired - Fee Related
- 1993-01-21 CN CN93101143A patent/CN1049217C/zh not_active Expired - Fee Related
- 1993-02-02 TW TW082100666A patent/TW226013B/zh active
-
1994
- 1994-06-27 BG BG98881A patent/BG61876B1/bg unknown
- 1994-07-18 OA OA60539A patent/OA09964A/en unknown
- 1994-07-19 FI FI943421A patent/FI111632B/fi active
- 1994-07-20 NO NO942720A patent/NO305952B1/no unknown
-
1995
- 1995-06-16 HU HU95P/P00242P patent/HU211295A9/hu unknown
-
1996
- 1996-07-01 US US08/674,259 patent/US5637697A/en not_active Expired - Fee Related
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PH30894A (en) | 1,5-Benzodiazepine derivative. | |
| DE59403259D1 (en) | Tetraaroxyperylen-3,4,9,10-tetracarbonsäurepolyimide | |
| ZA942571B (en) | 1,5 benzodiazepine derivatives | |
| EP0597463A3 (en) | Thermotherapiesonde. | |
| ZA926733B (en) | 1,2-Dihydro-2-oxopyridines. | |
| ZA934603B (en) | thiazolylvinylphenyl derivatives. | |
| EP0580285A3 (en) | Auto-reclosers. | |
| ZA94335B (en) | 2,6-Diaminopurine derivatives. | |
| PL312659A1 (en) | 1,5-benzodiazepine derivatives | |
| AP9500731A0 (en) | 1,5 benzodiazepine derivatives | |
| EP0668864A4 (en) | SUBSTITUTED BIPHENYLMETHYLIMIDAZOPYRIDINES. | |
| ZA946569B (en) | 1,5-Diphenyl-3-pyrazolylalkyl-N-hydroxydithiocarbamates | |
| EP0599191A3 (en) | Engine speed control circuit. | |
| ZA934381B (en) | Phenyl-1,2,5-oxadiazolecarboxamide-2-oxides. | |
| EP0592354A3 (de) | Vakuum-Zentrifuge. | |
| ZA933848B (en) | Pyridyl-1,2,5-oxadiazolecarboxamide-2-oxides | |
| ZA935828B (en) | New insobutyl-substituted methanesulphonyl-quinolyl-methoxyphenyl-cycloalkylacetamides. | |
| ZA972302B (en) | 1,25-Dihydroxy-16,22,23-trisdehydro-cholecalciferol derivatives. | |
| ZA935478B (en) | Lactam derivatives. | |
| EP0657435A3 (de) | 1,2-Dihydro-2-oxo-pyridine. | |
| IL110556A0 (en) | 7 alpha-amino-1, 1-dioxocephem l- valylamides | |
| HU9402902D0 (en) | 1,2-dihydro-2-oxo-3-methyl-sulfonyl-aminomethyl-pyridine derivatives | |
| GB2266530B (en) | Substituted 1,1,2-triphenylbutenes | |
| EP0683787A1 (en) | 4'-O-SULFONYL-ANTHRACYCLINE DERIVATIVES. | |
| GB9217992D0 (en) | 1,2-dioxanes |