PH12015500983A1 - Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections - Google Patents

Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections

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Publication number
PH12015500983A1
PH12015500983A1 PH12015500983A PH12015500983A PH12015500983A1 PH 12015500983 A1 PH12015500983 A1 PH 12015500983A1 PH 12015500983 A PH12015500983 A PH 12015500983A PH 12015500983 A PH12015500983 A PH 12015500983A PH 12015500983 A1 PH12015500983 A1 PH 12015500983A1
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PH
Philippines
Prior art keywords
amino
viral infections
treatment
quinazoline derivatives
heterocyclic substituted
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PH12015500983A
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English (en)
Other versions
PH12015500983B1 (en
Inventor
Last Stefaan Julien
Mc Gowan David Craig
Embrechts Werner
Pieters Serge Maria Aloysius
Onckers Tim Hugo Maria
Raboisson Pierre Jean-Marie Bernard
Original Assignee
Janssen Sciences Ireland Uc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47189782&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH12015500983(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of PH12015500983A1 publication Critical patent/PH12015500983A1/en
Publication of PH12015500983B1 publication Critical patent/PH12015500983B1/en

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/84Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
PH12015500983A 2012-11-16 2015-05-04 Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections PH12015500983B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12192970 2012-11-16
PCT/EP2013/073901 WO2014076221A1 (en) 2012-11-16 2013-11-15 Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections

Publications (2)

Publication Number Publication Date
PH12015500983A1 true PH12015500983A1 (en) 2015-08-03
PH12015500983B1 PH12015500983B1 (en) 2015-08-03

Family

ID=47189782

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12015500983A PH12015500983B1 (en) 2012-11-16 2015-05-04 Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections

Country Status (21)

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US (3) US9663474B2 (US06894165-20050517-C00155.png)
EP (1) EP2925729B1 (US06894165-20050517-C00155.png)
JP (1) JP6297055B2 (US06894165-20050517-C00155.png)
KR (1) KR102253773B1 (US06894165-20050517-C00155.png)
CN (1) CN105051018B (US06894165-20050517-C00155.png)
AU (1) AU2013346793B2 (US06894165-20050517-C00155.png)
BR (1) BR112015011036B1 (US06894165-20050517-C00155.png)
CA (1) CA2886635C (US06894165-20050517-C00155.png)
CL (1) CL2015001265A1 (US06894165-20050517-C00155.png)
DK (1) DK2925729T3 (US06894165-20050517-C00155.png)
EA (1) EA035431B1 (US06894165-20050517-C00155.png)
ES (1) ES2655843T3 (US06894165-20050517-C00155.png)
IL (1) IL237864A (US06894165-20050517-C00155.png)
MX (1) MX361585B (US06894165-20050517-C00155.png)
MY (1) MY171115A (US06894165-20050517-C00155.png)
NZ (2) NZ706226A (US06894165-20050517-C00155.png)
PH (1) PH12015500983B1 (US06894165-20050517-C00155.png)
PL (1) PL2925729T3 (US06894165-20050517-C00155.png)
SG (1) SG11201503042QA (US06894165-20050517-C00155.png)
UA (1) UA118341C2 (US06894165-20050517-C00155.png)
WO (1) WO2014076221A1 (US06894165-20050517-C00155.png)

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