PH12014502597A1 - N-substituted benzamides and their use in the treatment of pain - Google Patents

N-substituted benzamides and their use in the treatment of pain

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Publication number
PH12014502597A1
PH12014502597A1 PH12014502597A PH12014502597A PH12014502597A1 PH 12014502597 A1 PH12014502597 A1 PH 12014502597A1 PH 12014502597 A PH12014502597 A PH 12014502597A PH 12014502597 A PH12014502597 A PH 12014502597A PH 12014502597 A1 PH12014502597 A1 PH 12014502597A1
Authority
PH
Philippines
Prior art keywords
pain
treatment
substituted benzamides
compounds
subscript
Prior art date
Application number
PH12014502597A
Other languages
English (en)
Inventor
Andrez Jean-Christophe
Chowdhury Sultan
Decker Shannon
Dehnhardt Christoph Martin
Focken Thilo
Grimwood Michael Edward
Hemeon Ivan William
Jia Qi
Jun Li
Daniel F Ortwine
Safina Brian
Sheng Tao
Sun Shaoyi
Daniel P Sutherlin
Wilson Michael Scott
Zenova Alla Yurevna
Original Assignee
Genentech Inc
Xenon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genentech Inc, Xenon Pharmaceuticals Inc filed Critical Genentech Inc
Publication of PH12014502597A1 publication Critical patent/PH12014502597A1/en

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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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