PE20010303A1 - Nueva preparacion y forma de presentacion que contiene un agente activo labil en medio acido que consiste en un inhibidor de la bomba de protones labil en medio acido - Google Patents

Nueva preparacion y forma de presentacion que contiene un agente activo labil en medio acido que consiste en un inhibidor de la bomba de protones labil en medio acido

Info

Publication number
PE20010303A1
PE20010303A1 PE2000000565A PE0005652000A PE20010303A1 PE 20010303 A1 PE20010303 A1 PE 20010303A1 PE 2000000565 A PE2000000565 A PE 2000000565A PE 0005652000 A PE0005652000 A PE 0005652000A PE 20010303 A1 PE20010303 A1 PE 20010303A1
Authority
PE
Peru
Prior art keywords
acid medium
labil
inhibitor
presentation
proton pump
Prior art date
Application number
PE2000000565A
Other languages
English (en)
Spanish (es)
Inventor
Rudolf Linder
Rango Dietrich
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7910295&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20010303(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of PE20010303A1 publication Critical patent/PE20010303A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PE2000000565A 1999-06-07 2000-06-07 Nueva preparacion y forma de presentacion que contiene un agente activo labil en medio acido que consiste en un inhibidor de la bomba de protones labil en medio acido PE20010303A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19925710A DE19925710C2 (de) 1999-06-07 1999-06-07 Neue Zubereitung und Darreichungsform enthaltend einen säurelabilen Protonenpumpenhemmer

Publications (1)

Publication Number Publication Date
PE20010303A1 true PE20010303A1 (es) 2001-03-09

Family

ID=7910295

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2000000565A PE20010303A1 (es) 1999-06-07 2000-06-07 Nueva preparacion y forma de presentacion que contiene un agente activo labil en medio acido que consiste en un inhibidor de la bomba de protones labil en medio acido

Country Status (6)

Country Link
AR (1) AR024310A1 (de)
CO (1) CO5160296A1 (de)
DE (1) DE19925710C2 (de)
MY (1) MY138975A (de)
PE (1) PE20010303A1 (de)
TW (1) TWI255720B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2430816C (en) 2000-12-07 2012-05-15 Altana Pharma Ag Pharmaceutical preparation in the form of a paste comprising an acid-labile active ingredient
UA80393C2 (uk) * 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
WO2002045692A1 (en) * 2000-12-07 2002-06-13 Altana Pharma Ag Pharmaceutical preparation in the form of a suspension comprising an acid-labile active ingredient
DE10061138C1 (de) * 2000-12-07 2002-08-14 Byk Gulden Lomberg Chem Fab Pharmazeutische Zubereitung in Form eines Saftes enthaltend einen säurelabilen Wirkstoff
JP2004514737A (ja) * 2000-12-07 2004-05-20 アルタナ ファルマ アクチエンゲゼルシャフト 酸分解性活性成分を含有する迅速に崩壊する錠剤
DE10061136C1 (de) * 2000-12-07 2002-10-24 Byk Gulden Lomberg Chem Fab Schnell zerfallende Tablette enthaltend einen säurelabilen Protonenpumpenhemmer
DE10061137B4 (de) * 2000-12-07 2016-10-06 Takeda Gmbh Neue pharmazeutische Zubereitung
DE10061135C1 (de) * 2000-12-07 2002-11-07 Byk Gulden Lomberg Chem Fab Pharmazeutische Zubereitung in Form einer Paste enthaltend einen säurelabilen Wirkstoff
SE0101379D0 (sv) 2001-04-18 2001-04-18 Diabact Ab Komposition som hämmar utsöndring av magsyra
BR0212950A (pt) * 2001-09-28 2004-10-26 Mcneil Ppc Inc Formas de dosagens compósitas tendo uma porção inserida
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
CA2490142A1 (en) * 2002-07-03 2004-01-15 Abbott Laboratories Liquid dosage forms of proton pump inhibitors
DE10244129B4 (de) * 2002-09-23 2006-04-20 Iongate Biosciences Gmbh H+-K+-ATPase-Assay
SE0203065D0 (sv) 2002-10-16 2002-10-16 Diabact Ab Gastric acid secretion inhibiting composition
ME00524B (me) 2003-03-10 2011-10-10 Astrazeneca Ab Novi postupak za dobijanje roflumilasta
TW200503783A (en) * 2003-04-11 2005-02-01 Altana Pharma Ag Oral pharmaceutical preparation for proton pump antagonists
WO2006097456A1 (en) 2005-03-16 2006-09-21 Nycomed Gmbh Taste masked dosage form containing roflumilast
US8673352B2 (en) 2005-04-15 2014-03-18 Mcneil-Ppc, Inc. Modified release dosage form

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2725924C3 (de) * 1977-06-08 1980-11-06 Hobeg Hochtemperaturreaktor-Brennelement Gmbh, 6450 Hanau Verfahren zur Herstellung kugelförmiger Teilchen aus niedrigschmelzenden organischen Substanzen
DE3524572A1 (de) * 1985-07-10 1987-01-15 Thomae Gmbh Dr K Feste arzneimittelformen zur peroralen anwendung enthaltend 9-deoxo-11-deoxy-9,11-(imino(2-(2-methoxyethoxy)ethyliden)-oxy)-(9s)-erythromycin und verfahren zu ihrer herstellung
JP2681373B2 (ja) * 1988-07-18 1997-11-26 塩野義製薬株式会社 徐放性製剤の製造法

Also Published As

Publication number Publication date
AR024310A1 (es) 2002-09-25
CO5160296A1 (es) 2002-05-30
DE19925710A1 (de) 2000-12-14
TWI255720B (en) 2006-06-01
DE19925710C2 (de) 2002-10-10
MY138975A (en) 2009-08-28

Similar Documents

Publication Publication Date Title
PE20010303A1 (es) Nueva preparacion y forma de presentacion que contiene un agente activo labil en medio acido que consiste en un inhibidor de la bomba de protones labil en medio acido
UA74339C2 (uk) Форма для введення, що включає інгібітор протонної помпи у вигляді окремих одиниць, та спосіб їх одержання
CY1120513T1 (el) Υψηλης συμπυκνωσης συνθεση μινοξιδιλης
ES2542728T3 (es) Composiciones farmacéuticas que tienen la biodisponibilidad deseable
RU2005110945A (ru) Капсулы, содержащие водные наполняющие композиции, стабилизированные производным циклодекстрина
ES2155043B1 (es) Composiciones farmaceuticas comprendiendo acido pirimidin-5-il(3r, 5s)-3,5-dihidroxihept-6-enoico o una sal suya, su estabilizacion con sal fosfato tribasico y su preparacion.
AP2397A (en) Matrix for sustained, invariant and independent release of active compounds.
PE3296A1 (es) Composicion oral conteniendo un mucoadhesivo
JP2006328089A (ja) 安定な局所レチノイド組成物
CO5180575A1 (es) Composiciones antibacterianas orales de lupulona hidrogenda estable
PE20081365A1 (es) Formulaciones topicas para administracion local que contienen indoxacarb
CO5221123A1 (es) Desodorante con pequenas particulas de oxido de zinc
PT2116243E (pt) Composição de gel para tratamento de micoses
BR0007360A (pt) Composição de liberação controlada
AR055090A1 (es) Una presentacion farmaceutica de forma de dosificacion de liberacion modificada que comprende un inhibidor de la enzima ciclooxigenasa
PE20041024A1 (es) Sistema de liberacion controlada
AR038681A1 (es) Formulacion oral de solucion solida de una sustancia activa pobremente soluble en agua
NO20055601L (no) Farmasoytisk preparat i form av en hydrogel for transdermal administrasjon av aktive virkestoffer
NO820319L (no) Antimykotisk middel i form av stifter og med hoey virksom stoff frigjoering
CO5380014A1 (es) Formulacion farmaceuticas para la administracion oral o topica de compuestos hidrofobicos que no frma emulsion
PE20040545A1 (es) Formulaciones parasiticidas que comprenden benzoimidazoles o salicilanilidas en combinacion con lactonas macrociclicas
MY143793A (en) Non-tabletted, chewable, individually dosed administration forms
ES2460967T3 (es) Método para la prevención de la degradación de una sustancia térmicamente inestable
ES2530874T3 (es) Formulaciones de depósito de corta duración
CO5160318A1 (es) Composicion precursora para preparar un dialitico

Legal Events

Date Code Title Description
FG Grant, registration
FD Application declared void or lapsed