CO5160296A1 - Nuevas formas de presentacion para agentes activos labiles en medio acido, unidad de agente activo y proceso para la produccion de dicha unidad de agente - Google Patents
Nuevas formas de presentacion para agentes activos labiles en medio acido, unidad de agente activo y proceso para la produccion de dicha unidad de agenteInfo
- Publication number
- CO5160296A1 CO5160296A1 CO00040091A CO00040091A CO5160296A1 CO 5160296 A1 CO5160296 A1 CO 5160296A1 CO 00040091 A CO00040091 A CO 00040091A CO 00040091 A CO00040091 A CO 00040091A CO 5160296 A1 CO5160296 A1 CO 5160296A1
- Authority
- CO
- Colombia
- Prior art keywords
- agent unit
- active
- active agent
- production
- agents
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a una forma de presentación para agentes activos lábiles en medio ácido, que contiene adyuvantes farmacéuticos y unidades individuales múltiples de agente activo, caracterizada porque el agente activo lábil en medio ácido se encuentra en las unidades individuales de agente activo en una matriz constituida por una mezcla que contiene al menos un alcohol graso y al menos una parafina sólida.Igualmente, se refiere a una unidad de agente activo que contiene un agente activo lábil en medio ácido y a un proceso para la producción de dicha una unidad de agente activo.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19925710A DE19925710C2 (de) | 1999-06-07 | 1999-06-07 | Neue Zubereitung und Darreichungsform enthaltend einen säurelabilen Protonenpumpenhemmer |
Publications (1)
Publication Number | Publication Date |
---|---|
CO5160296A1 true CO5160296A1 (es) | 2002-05-30 |
Family
ID=7910295
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO00040091A CO5160296A1 (es) | 1999-06-07 | 2000-05-30 | Nuevas formas de presentacion para agentes activos labiles en medio acido, unidad de agente activo y proceso para la produccion de dicha unidad de agente |
Country Status (6)
Country | Link |
---|---|
AR (1) | AR024310A1 (es) |
CO (1) | CO5160296A1 (es) |
DE (1) | DE19925710C2 (es) |
MY (1) | MY138975A (es) |
PE (1) | PE20010303A1 (es) |
TW (1) | TWI255720B (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10061135C1 (de) * | 2000-12-07 | 2002-11-07 | Byk Gulden Lomberg Chem Fab | Pharmazeutische Zubereitung in Form einer Paste enthaltend einen säurelabilen Wirkstoff |
DE10061138C1 (de) * | 2000-12-07 | 2002-08-14 | Byk Gulden Lomberg Chem Fab | Pharmazeutische Zubereitung in Form eines Saftes enthaltend einen säurelabilen Wirkstoff |
DE10061136C1 (de) * | 2000-12-07 | 2002-10-24 | Byk Gulden Lomberg Chem Fab | Schnell zerfallende Tablette enthaltend einen säurelabilen Protonenpumpenhemmer |
UA80393C2 (uk) * | 2000-12-07 | 2007-09-25 | Алтана Фарма Аг | Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці |
BR0115986A (pt) * | 2000-12-07 | 2003-12-23 | Altana Pharma Ag | Comprimido de desintegração rápida contendo um ingrediente ativo instável aos ácidos |
AU2002234545A1 (en) | 2000-12-07 | 2002-06-18 | Byk Gulden Lomberg Chemische Fabrik G.M.B.H. | Pharmaceutical preparation in the form of a suspension comprising an acid-labileactive ingredient |
BR0115985A (pt) | 2000-12-07 | 2003-12-23 | Altana Pharma Ag | Preparação farmacêutica em forma de uma pasta compreendendo um ingrediente ativo ácido-lábil |
DE10061137B4 (de) * | 2000-12-07 | 2016-10-06 | Takeda Gmbh | Neue pharmazeutische Zubereitung |
SE0101379D0 (sv) | 2001-04-18 | 2001-04-18 | Diabact Ab | Komposition som hämmar utsöndring av magsyra |
US20040213848A1 (en) | 2001-09-28 | 2004-10-28 | Shun-Por Li | Modified release dosage forms |
MY140561A (en) | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
EP1572151A1 (en) * | 2002-07-03 | 2005-09-14 | Abbott Laboratories | Liquid dosage forms of proton pump inhibitors |
DE10244129B4 (de) * | 2002-09-23 | 2006-04-20 | Iongate Biosciences Gmbh | H+-K+-ATPase-Assay |
SE0203065D0 (sv) | 2002-10-16 | 2002-10-16 | Diabact Ab | Gastric acid secretion inhibiting composition |
BRPI0406427B8 (pt) | 2003-03-10 | 2021-05-25 | Astrazeneca Ab | processo para a preparação de roflumilast |
TW200503783A (en) * | 2003-04-11 | 2005-02-01 | Altana Pharma Ag | Oral pharmaceutical preparation for proton pump antagonists |
DK1861074T3 (da) | 2005-03-16 | 2013-07-29 | Takeda Gmbh | Smagsmaskeret doseringsform indeholdende roflumilast |
US8673352B2 (en) | 2005-04-15 | 2014-03-18 | Mcneil-Ppc, Inc. | Modified release dosage form |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2725924C3 (de) * | 1977-06-08 | 1980-11-06 | Hobeg Hochtemperaturreaktor-Brennelement Gmbh, 6450 Hanau | Verfahren zur Herstellung kugelförmiger Teilchen aus niedrigschmelzenden organischen Substanzen |
DE3524572A1 (de) * | 1985-07-10 | 1987-01-15 | Thomae Gmbh Dr K | Feste arzneimittelformen zur peroralen anwendung enthaltend 9-deoxo-11-deoxy-9,11-(imino(2-(2-methoxyethoxy)ethyliden)-oxy)-(9s)-erythromycin und verfahren zu ihrer herstellung |
JP2681373B2 (ja) * | 1988-07-18 | 1997-11-26 | 塩野義製薬株式会社 | 徐放性製剤の製造法 |
-
1999
- 1999-06-07 DE DE19925710A patent/DE19925710C2/de not_active Expired - Fee Related
-
2000
- 2000-05-30 MY MYPI20002403A patent/MY138975A/en unknown
- 2000-05-30 CO CO00040091A patent/CO5160296A1/es unknown
- 2000-06-07 TW TW089111052A patent/TWI255720B/zh not_active IP Right Cessation
- 2000-06-07 AR ARP000102825A patent/AR024310A1/es unknown
- 2000-06-07 PE PE2000000565A patent/PE20010303A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DE19925710C2 (de) | 2002-10-10 |
AR024310A1 (es) | 2002-09-25 |
PE20010303A1 (es) | 2001-03-09 |
TWI255720B (en) | 2006-06-01 |
DE19925710A1 (de) | 2000-12-14 |
MY138975A (en) | 2009-08-28 |
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