NZ594044A - Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics - Google Patents

Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics

Info

Publication number
NZ594044A
NZ594044A NZ59404410A NZ59404410A NZ594044A NZ 594044 A NZ594044 A NZ 594044A NZ 59404410 A NZ59404410 A NZ 59404410A NZ 59404410 A NZ59404410 A NZ 59404410A NZ 594044 A NZ594044 A NZ 594044A
Authority
NZ
New Zealand
Prior art keywords
inhibitor
dpp
antidiabetic agent
linagliptin
optionally
Prior art date
Application number
NZ59404410A
Other languages
English (en)
Inventor
Hans-Juergen Woerle
Eva Ulrike Graefe-Mody
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42174359&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ594044(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Priority to NZ619520A priority Critical patent/NZ619520A/en
Publication of NZ594044A publication Critical patent/NZ594044A/en

Links

Classifications

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Physiology (AREA)
NZ59404410A 2009-02-13 2010-02-12 Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics NZ594044A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NZ619520A NZ619520A (en) 2009-02-13 2010-02-12 Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09152869 2009-02-13
PCT/EP2010/051817 WO2010092163A2 (en) 2009-02-13 2010-02-12 Antidiabetic medications

Publications (1)

Publication Number Publication Date
NZ594044A true NZ594044A (en) 2014-08-29

Family

ID=42174359

Family Applications (2)

Application Number Title Priority Date Filing Date
NZ59404410A NZ594044A (en) 2009-02-13 2010-02-12 Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics
NZ619520A NZ619520A (en) 2009-02-13 2010-02-12 Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics

Family Applications After (1)

Application Number Title Priority Date Filing Date
NZ619520A NZ619520A (en) 2009-02-13 2010-02-12 Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics

Country Status (14)

Country Link
US (6) US20120094894A1 (cg-RX-API-DMAC7.html)
EP (1) EP2395988A2 (cg-RX-API-DMAC7.html)
JP (3) JP2012517977A (cg-RX-API-DMAC7.html)
KR (2) KR20110115582A (cg-RX-API-DMAC7.html)
CN (3) CN102387795A (cg-RX-API-DMAC7.html)
AU (1) AU2010212823B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI1013639A2 (cg-RX-API-DMAC7.html)
CA (1) CA2752437C (cg-RX-API-DMAC7.html)
CL (1) CL2011001853A1 (cg-RX-API-DMAC7.html)
EA (1) EA029759B1 (cg-RX-API-DMAC7.html)
IL (1) IL213716A0 (cg-RX-API-DMAC7.html)
MX (2) MX387264B (cg-RX-API-DMAC7.html)
NZ (2) NZ594044A (cg-RX-API-DMAC7.html)
WO (1) WO2010092163A2 (cg-RX-API-DMAC7.html)

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* Cited by examiner, † Cited by third party
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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
JP5323684B2 (ja) 2006-05-04 2013-10-23 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 多形体
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
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US20150105318A1 (en) 2015-04-16
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JP2012517977A (ja) 2012-08-09
US20220088023A1 (en) 2022-03-24
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CA2752437A1 (en) 2010-08-19
KR20110115582A (ko) 2011-10-21
IL213716A0 (en) 2011-07-31
CN117547538A (zh) 2024-02-13
WO2010092163A2 (en) 2010-08-19
CN102387795A (zh) 2012-03-21
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JP2015044875A (ja) 2015-03-12
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US20120094894A1 (en) 2012-04-19
EA029759B1 (ru) 2018-05-31
US20200323861A1 (en) 2020-10-15
AU2010212823B2 (en) 2016-01-28
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