MX387264B - Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos. - Google Patents

Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos.

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Publication number
MX387264B
MX387264B MX2016013286A MX2016013286A MX387264B MX 387264 B MX387264 B MX 387264B MX 2016013286 A MX2016013286 A MX 2016013286A MX 2016013286 A MX2016013286 A MX 2016013286A MX 387264 B MX387264 B MX 387264B
Authority
MX
Mexico
Prior art keywords
dpp
inhibitor
combination
linagliptin
antidiabetics
Prior art date
Application number
MX2016013286A
Other languages
English (en)
Inventor
Eva Ulrike Graefe-Mody
Hans-Juergen Woerle
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42174359&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX387264(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MX387264B publication Critical patent/MX387264B/es

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    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
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  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Neurology (AREA)
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  • Oil, Petroleum & Natural Gas (AREA)
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Abstract

La invención se refiere a medicaciones antidiabéticas que son adecuadas en el tratamiento o la prevención de una o más condiciones, seleccionadas de entre diabetes mellitus tipo 1, diabetes mellitus tipo 2, tolerancia deteriorada a la glucosa e hiperglucemia, inter alia. Además, la presente invención se refiere a métodos para prevenir o tratar trastornos metabólicos y condiciones relacionadas. La medicación es un mono tratamiento con un inhibidor de DPP-4 (preferiblemente linagliptina) o un tratamiento de combinación con un inhibidor de DPP-4 y un segundo y/o un tercer antidiabético.
MX2016013286A 2009-02-13 2010-02-12 Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos. MX387264B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09152869 2009-02-13
PCT/EP2010/051817 WO2010092163A2 (en) 2009-02-13 2010-02-12 Antidiabetic medications

Publications (1)

Publication Number Publication Date
MX387264B true MX387264B (es) 2025-03-18

Family

ID=42174359

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2016013286A MX387264B (es) 2009-02-13 2010-02-12 Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos.
MX2011008416A MX2011008416A (es) 2009-02-13 2010-02-12 Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2011008416A MX2011008416A (es) 2009-02-13 2010-02-12 Medicaciones antidiabeticas que comprenden un inhibidor de dpp-4 (linagliptina) opcionalmente en combinacion con otros antidiabeticos.

Country Status (14)

Country Link
US (7) US20120094894A1 (es)
EP (1) EP2395988A2 (es)
JP (3) JP2012517977A (es)
KR (2) KR20110115582A (es)
CN (3) CN102387795A (es)
AU (1) AU2010212823B2 (es)
BR (1) BRPI1013639A2 (es)
CA (1) CA2752437C (es)
CL (1) CL2011001853A1 (es)
EA (1) EA029759B1 (es)
IL (1) IL213716A0 (es)
MX (2) MX387264B (es)
NZ (2) NZ619520A (es)
WO (1) WO2010092163A2 (es)

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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
CN102838599A (zh) 2006-05-04 2012-12-26 贝林格尔.英格海姆国际有限公司 多晶型
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
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KR20160143897A (ko) 2016-12-14
KR20110115582A (ko) 2011-10-21
AU2010212823A1 (en) 2011-08-18
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US20220088023A1 (en) 2022-03-24
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