NZ249189A - Benzothiazepine derivatives and pharmaceutical compositions - Google Patents

Benzothiazepine derivatives and pharmaceutical compositions

Info

Publication number
NZ249189A
NZ249189A NZ249189A NZ24918993A NZ249189A NZ 249189 A NZ249189 A NZ 249189A NZ 249189 A NZ249189 A NZ 249189A NZ 24918993 A NZ24918993 A NZ 24918993A NZ 249189 A NZ249189 A NZ 249189A
Authority
NZ
New Zealand
Prior art keywords
compound
formula
solvate
functional derivative
butyl
Prior art date
Application number
NZ249189A
Other languages
English (en)
Inventor
Lawrence Edward Brieaddy
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of NZ249189A publication Critical patent/NZ249189A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
NZ249189A 1992-02-17 1993-02-16 Benzothiazepine derivatives and pharmaceutical compositions NZ249189A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929203347A GB9203347D0 (en) 1992-02-17 1992-02-17 Hypolipidaemic compounds

Publications (1)

Publication Number Publication Date
NZ249189A true NZ249189A (en) 1996-02-27

Family

ID=10710542

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ249189A NZ249189A (en) 1992-02-17 1993-02-16 Benzothiazepine derivatives and pharmaceutical compositions

Country Status (21)

Country Link
US (2) US5663165A (en:Method)
EP (1) EP0626952B1 (en:Method)
JP (1) JP2904926B2 (en:Method)
KR (1) KR100265529B1 (en:Method)
AT (1) ATE178897T1 (en:Method)
AU (1) AU675419B2 (en:Method)
CA (1) CA2117485A1 (en:Method)
DE (1) DE69324479T2 (en:Method)
DK (1) DK0626952T3 (en:Method)
ES (1) ES2131106T3 (en:Method)
FI (1) FI943775A7 (en:Method)
GB (1) GB9203347D0 (en:Method)
GR (1) GR3030491T3 (en:Method)
HU (1) HUT71487A (en:Method)
IL (1) IL104740A (en:Method)
MX (1) MX9300821A (en:Method)
MY (1) MY129970A (en:Method)
NZ (1) NZ249189A (en:Method)
TW (1) TW274547B (en:Method)
WO (1) WO1993016055A1 (en:Method)
ZA (1) ZA931073B (en:Method)

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* Cited by examiner, † Cited by third party
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KR20250110930A (ko) 2022-12-09 2025-07-21 알비레오 에이비 신장 질병 치료용 asbt 억제제
WO2025146508A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators
WO2025146507A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators

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EP0626952A1 (en) 1994-12-07
US5663165A (en) 1997-09-02
DE69324479D1 (de) 1999-05-20
FI943775L (fi) 1994-08-16
FI943775A0 (fi) 1994-08-16
CA2117485A1 (en) 1993-08-19
FI943775A7 (fi) 1994-08-16
US5859240A (en) 1999-01-12
JP2904926B2 (ja) 1999-06-14
ATE178897T1 (de) 1999-04-15
JPH07503724A (ja) 1995-04-20
MY129970A (en) 2007-05-31
WO1993016055A1 (en) 1993-08-19
ZA931073B (en) 1994-08-16
HK1004217A1 (en) 1998-11-20
ES2131106T3 (es) 1999-07-16
AU675419B2 (en) 1997-02-06
KR950700265A (ko) 1995-01-16
MX9300821A (es) 1993-09-01
AU3508293A (en) 1993-09-03
IL104740A0 (en) 1993-06-10
KR100265529B1 (ko) 2000-11-01
GB9203347D0 (en) 1992-04-01
HU9402365D0 (en) 1994-10-28
EP0626952B1 (en) 1999-04-14
IL104740A (en) 1996-09-12
DE69324479T2 (de) 1999-09-16
GR3030491T3 (en) 1999-10-29
DK0626952T3 (da) 1999-10-25
TW274547B (en:Method) 1996-04-21
HUT71487A (en) 1995-11-28

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